Title : Chemoproteomics-Enabled Identification of 4-Oxo-beta-Lactams as Inhibitors of Dipeptidyl Peptidases 8 and 9 - Carvalho_2022_Angew.Chem.Int.Ed.Engl_61_e202210498 |
Author(s) : Carvalho LAR , Ross B , Fehr L , Bolgi O , Wohrle S , Lum KM , Podlesainski D , Vieira AC , Kiefersauer R , Felix R , Rodrigues T , Lucas SD , Gross O , Geiss-Friedlander R , Cravatt BF , Huber R , Kaiser M , Moreira R |
Ref : Angew Chem Int Ed Engl , : , 2022 |
Abstract : |
PubMedSearch : Carvalho_2022_Angew.Chem.Int.Ed.Engl_61_e202210498 |
PubMedID: 36089535 |
Gene_locus related to this paper: human-DPP8 , human-DPP9 |
Title : Synthesis, Biological Evaluation, and Docking Studies of Open-chain Carbohydrate Amides as Acetylcholinesterase Inhibitors - Goncalves-Pereira_2022_Med.Chem__ |
Author(s) : Goncalves-Pereira R , Figueiredo JA , Lucas SD , Garcia-Moreno MI , Mellet CO , Rauter AP , Ismael MI |
Ref : Med Chem , : , 2022 |
Abstract : |
PubMedSearch : Goncalves-Pereira_2022_Med.Chem__ |
PubMedID: 36476428 |
Title : 3-Oxo-beta-sultam as a Sulfonylating Chemotype for Inhibition of Serine Hydrolases and Activity-Based Protein Profiling - Carvalho_2020_ACS.Chem.Biol_15_878 |
Author(s) : Carvalho LAR , Almeida VT , Brito JA , Lum KM , Oliveira TF , Guedes RC , Goncalves LM , Lucas SD , Cravatt BF , Archer M , Moreira R |
Ref : ACS Chemical Biology , 15 :878 , 2020 |
Abstract : |
PubMedSearch : Carvalho_2020_ACS.Chem.Biol_15_878 |
PubMedID: 32176480 |
Title : Ursolic and oleanolic acid derivatives with cholinesterase inhibiting potential - Loesche_2018_Bioorg.Chem_85_23 |
Author(s) : Loesche A , Kowitsch A , Lucas SD , Al-Halabi Z , Sippl W , Al-Harrasi A , Csuk R |
Ref : Bioorg Chem , 85 :23 , 2018 |
Abstract : |
PubMedSearch : Loesche_2018_Bioorg.Chem_85_23 |
PubMedID: 30599410 |
Title : Converting maslinic acid into an effective inhibitor of acylcholinesterases - Schwarz_2015_Eur.J.Med.Chem_103_438 |
Author(s) : Schwarz S , Loesche A , Lucas SD , Sommerwerk S , Serbian I , Siewert B , Pianowski E , Csuk R |
Ref : Eur Journal of Medicinal Chemistry , 103 :438 , 2015 |
Abstract : |
PubMedSearch : Schwarz_2015_Eur.J.Med.Chem_103_438 |
PubMedID: 26383128 |
Title : Amino derivatives of glycyrrhetinic acid as potential inhibitors of cholinesterases - Schwarz_2014_Bioorg.Med.Chem_22_3370 |
Author(s) : Schwarz S , Lucas SD , Sommerwerk S , Csuk R |
Ref : Bioorganic & Medicinal Chemistry , 22 :3370 , 2014 |
Abstract : |
PubMedSearch : Schwarz_2014_Bioorg.Med.Chem_22_3370 |
PubMedID: 24853320 |