Szymanski P

References (26)

Title : New cyclopentaquinoline and 3,5-dichlorobenzoic acid hybrids with neuroprotection against oxidative stress for the treatment of Alzheimer's disease - Czarnecka_2023_J.Enzyme.Inhib.Med.Chem_38_2158822
Author(s) : Czarnecka K , Girek M , Krecisz P , Skibinski R , Latka K , Jonczyk J , Bajda M , Szymczyk P , Galita G , Kabzinski J , Majsterek I , Espargaro A , Sabate R , Szymanski P
Ref : J Enzyme Inhib Med Chem , 38 :2158822 , 2023
PubMedID: 36629422

Title : Novel Cyclopentaquinoline and Acridine Analogs as Multifunctional, Potent Drug Candidates in Alzheimer's Disease - Maciejewska_2022_Int.J.Mol.Sci_23_
Author(s) : Maciejewska K , Czarnecka K , Krecisz P , Niedzialek D , Wieczorek G , Skibinski R , Szymanski P
Ref : Int J Mol Sci , 23 : , 2022
PubMedID: 35682556

Title : Synthesis and Biological Studies of Novel Aminophosphonates and Their Metal Carbonyl Complexes (Fe, Ru) - Kosinska_2022_Int.J.Mol.Sci_23_
Author(s) : Kosinska A , Virieux D , Pirat JL , Czarnecka K , Girek M , Szymanski P , Wojtulewski S , Vasudevan S , Chworos A , Rudolf B
Ref : Int J Mol Sci , 23 : , 2022
PubMedID: 35897660

Title : New Imaging Modality of COVID-19 Pneumonia Developed on the Basis of Alzheimer's Disease Research - Kozminski_2022_Int.J.Mol.Sci_23_
Author(s) : Kozminski P , Niedzialek D , Wieczorek G , Halik PK , Czarnecka K , Rogut A , Cheda L , Rogulski Z , Szymanski P , Gniazdowska E
Ref : Int J Mol Sci , 23 : , 2022
PubMedID: 35955536

Title : Biological evaluation and molecular docking of novel 1,3,4-thiadiazole-resorcinol conjugates as multifunctional cholinesterases inhibitors - Skrzypek_2021_Bioorg.Chem_107_104617
Author(s) : Skrzypek A , Matysiak J , Karpinska M , Czarnecka K , Krecisz P , Stary D , Kukulowicz J , Paw B , Bajda M , Szymanski P , Niewiadomy A
Ref : Bioorg Chem , 107 :104617 , 2021
PubMedID: 33444983

Title : New Tetrahydroacridine Hybrids with Dichlorobenzoic Acid Moiety Demonstrating Multifunctional Potential for the Treatment of Alzheimer's Disease - Czarnecka_2020_Int.J.Mol.Sci_21_
Author(s) : Czarnecka K , Girek M , Wojtowicz P , Krecisz P , Skibinski R , Jonczyk J , Latka K , Bajda M , Walczak A , Galita G , Kabzinski J , Majsterek I , Szymczyk P , Szymanski P
Ref : Int J Mol Sci , 21 : , 2020
PubMedID: 32466601

Title : Discovery of New Cyclopentaquinoline Analogues as Multifunctional Agents for the Treatment of Alzheimer's Disease - Czarnecka_2019_Int.J.Mol.Sci_20_
Author(s) : Czarnecka K , Girek M , Krecisz P , Skibinski R , Latka K , Jonczyk J , Bajda M , Kabzinski J , Majsterek I , Szymczyk P , Szymanski P
Ref : Int J Mol Sci , 20 : , 2019
PubMedID: 30678364

Title : Biological Evaluation, Molecular Docking, and SAR Studies of Novel 2-(2,4-Dihydroxyphenyl)-1H- Benzimidazole Analogues - Matysiak_2019_Biomolecules_9_
Author(s) : Matysiak J , Skrzypek A , Karpinska M , Czarnecka K , Szymanski P , Bajda M , Niewiadomy A
Ref : Biomolecules , 9 : , 2019
PubMedID: 31842463

Title : Synthesis, physicochemical and biological evaluation of tacrine derivative labeled with technetium-99m and gallium-68 as a prospective diagnostic tool for early diagnosis of Alzheimer's disease - Gniazdowska_2019_Bioorg.Chem_91_103136
Author(s) : Gniazdowska E , Kozminski P , Halik P , Bajda M , Czarnecka K , Mikiciuk-Olasik E , Maslowska K , Rogulski Z , Cheda L , Kilian K , Szymanski P
Ref : Bioorg Chem , 91 :103136 , 2019
PubMedID: 31374521

Title : New tacrine-acridine hybrids as promising multifunctional drugs for potential treatment of Alzheimer's disease - Chufarova_2018_Arch.Pharm.(Weinheim)__e1800050
Author(s) : Chufarova N , Czarnecka K , Skibinski R , Cuchra M , Majsterek I , Szymanski P
Ref : Arch Pharm (Weinheim) , :e1800050 , 2018
PubMedID: 29870588

Title : Tetrahydroacridine derivatives with dichloronicotinic acid moiety as attractive, multipotent agents for Alzheimer's disease treatment - Czarnecka_2018_Eur.J.Med.Chem_145_760
Author(s) : Czarnecka K , Chufarova N , Halczuk K , Maciejewska K , Girek M , Skibinski R , Jonczyk J , Bajda M , Kabzinski J , Majsterek I , Szymanski P
Ref : Eur Journal of Medicinal Chemistry , 145 :760 , 2018
PubMedID: 29353726

Title : Novel tetrahydroacridine derivatives with iodobenzoic acid moiety as multifunctional acetylcholinesterase inhibitors - Skibinski_2018_Chem.Biol.Drug.Des_91_505
Author(s) : Skibinski R , Czarnecka K , Girek M , Bilichowski I , Chufarova N , Mikiciuk-Olasik E , Szymanski P
Ref : Chemical Biology Drug Des , 91 :505 , 2018
PubMedID: 28944565

Title : New cyclopentaquinoline hybrids with multifunctional capacities for the treatment of Alzheimer's disease - Czarnecka_2017_J.Enzyme.Inhib.Med.Chem_33_158
Author(s) : Czarnecka K , Girek M , Maciejewska K , Skibinski R , Jonczyk J , Bajda M , Kabzinski J , Solowiej P , Majsterek I , Szymanski P
Ref : J Enzyme Inhib Med Chem , 33 :158 , 2017
PubMedID: 29210299

Title : Tetrahydroacridine derivatives with fluorobenzoic acid moiety as multifunctional agents for Alzheimer's disease treatment - Czarnecka_2017_Bioorg.Chem_72_315
Author(s) : Czarnecka K , Szymanski P , Girek M , Mikiciuk-Olasik E , Skibinski R , Kabzinski J , Majsterek I , Malawska B , Jonczyk J , Bajda M
Ref : Bioorg Chem , 72 :315 , 2017
PubMedID: 28501648

Title : Synthesis, physicochemical and biological studies of technetium-99m labeled tacrine derivative as a diagnostic tool for evaluation of cholinesterase level - Gniazdowska_2017_Bioorg.Med.Chem_25_912
Author(s) : Gniazdowska E , Kozminski P , Wasek M , Bajda M , Sikora J , Mikiciuk-Olasik E , Szymanski P
Ref : Bioorganic & Medicinal Chemistry , 25 :912 , 2017
PubMedID: 27998671

Title : Taxodione and Extracts from Salvia austriaca Roots as Human Cholinesterase Inhibitors - Kuzma_2016_Phytother.Res_30_234
Author(s) : Kuzma L , Wysokinska H , Sikora J , Olszewska P , Mikiciuk-Olasik E , Szymanski P
Ref : Phytother Res , 30 :234 , 2016
PubMedID: 26621777

Title : Synthesis, biological evaluation and molecular modeling of new tetrahydroacridine derivatives as potential multifunctional agents for the treatment of Alzheimer's disease - Bajda_2015_Bioorg.Med.Chem_23_5610
Author(s) : Bajda M , Jonczyk J , Malawska B , Czarnecka K , Girek M , Olszewska P , Sikora J , Mikiciuk-Olasik E , Skibinski R , Gumieniczek A , Szymanski P
Ref : Bioorganic & Medicinal Chemistry , 23 :5610 , 2015
PubMedID: 26242241

Title : Synthesis and biological evaluation of 1,3,4-thiadiazole analogues as novel AChE and BCHE inhibitors - Skrzypek_2013_Eur.J.Med.Chem_62C_311
Author(s) : Skrzypek A , Matysiak J , Niewiadomy A , Bajda M , Szymanski P
Ref : Eur Journal of Medicinal Chemistry , 62C :311 , 2013
PubMedID: 23376249

Title : New tacrine analogs as acetylcholinesterase inhibitors - theoretical study with chemometric analysis - Szymanski_2013_Molecules_18_2878
Author(s) : Szymanski P , Skibinski R , Inglot T , Bajda M , Jonczyk J , Malawska B , Mikiciuk-Olasik E
Ref : Molecules , 18 :2878 , 2013
PubMedID: 23459299

Title : Synthesis and biological activity of new donepezil-hydrazinonicotinamide hybrids - Zurek_2013_Drug.Res.(Stuttg)_63_137
Author(s) : Zurek E , Szymanski P , Mikiciuk-Olasik E
Ref : Drug Res (Stuttg) , 63 :137 , 2013
PubMedID: 23447117

Title : 2,3-dihydro-1H-cyclopenta[b]quinoline derivatives as acetylcholinesterase inhibitors-synthesis, radiolabeling and biodistribution - Szymanski_2012_Int.J.Mol.Sci_13_10067
Author(s) : Szymanski P , Laznickova A , Laznicek M , Bajda M , Malawska B , Markowicz M , Mikiciuk-Olasik E
Ref : Int J Mol Sci , 13 :10067 , 2012
PubMedID: 22949848

Title : Synthesis, biological activity and molecular modeling of 4-fluoro-N-[omega-(1,2,3,4-tetrahydroacridin-9-ylamino)-alkyl]-benzamide derivatives as cholinesterase inhibitors - Szymanski_2012_Arzneimittelforschung_62_655
Author(s) : Szymanski P , Markowicz M , Bajda M , Malawska B , Mikiciuk-Olasik E
Ref : Arzneimittelforschung , 62 :655 , 2012
PubMedID: 23154886

Title : Design, synthesis and biological evaluation of new 2-benzoxazolinone derivatives as potential cholinesterase inhibitors for therapy of alzheimer's disease - Szymanski_2011_Pharmazie_66_399
Author(s) : Szymanski P , Janik A , Zurek E , Mikiciuk-Olasik E
Ref : Pharmazie , 66 :399 , 2011
PubMedID: 21699076

Title : Synthesis, biological activity and HPLC validation of 1,2,3,4-tetrahydroacridine derivatives as acetylcholinesterase inhibitors - Szymanski_2011_Eur.J.Med.Chem_46_3250
Author(s) : Szymanski P , Karpinski A , Mikiciuk-Olasik E
Ref : Eur Journal of Medicinal Chemistry , 46 :3250 , 2011
PubMedID: 21570751

Title : Synthesis and biological activity of derivatives of tetrahydroacridine as acetylcholinesterase inhibitors - Szymanski_2011_Bioorg.Chem_39_138
Author(s) : Szymanski P , Markowicz M , Mikiciuk-Olasik E
Ref : Bioorg Chem , 39 :138 , 2011
PubMedID: 21621811

Title : New tacrine-hydrazinonicotinamide hybrids as acetylcholinesterase inhibitors of potential interest for the early diagnostics of Alzheimer's disease - Szymanski_2006_Pharmazie_61_269
Author(s) : Szymanski P , Zurek E , Mikiciuk-Olasik E
Ref : Pharmazie , 61 :269 , 2006
PubMedID: 16649535