Report for Espargaro A

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References (14)

Title : Novel drug-like fluorenyl derivatives as selective butyrylcholinesterase and beta-amyloid inhibitors for the treatment of Alzheimer's disease - Pasieka_2023_Bioorg.Med.Chem_88-89_117333
Author(s) : Pasieka A , Panek D , Zareba P , Slugocka E , Gucwa N , Espargaro A , Latacz G , Khan N , Bucki A , Sabate R , Wieckowska A , Malawska B
Ref : Bioorganic & Medicinal Chemistry , 88-89 :117333 , 2023
Abstract : Pasieka_2023_Bioorg.Med.Chem_88-89_117333
ESTHER : Pasieka_2023_Bioorg.Med.Chem_88-89_117333
PubMedSearch : Pasieka_2023_Bioorg.Med.Chem_88-89_117333
PubMedID: 37236021

Title : Discovery of novel multifunctional ligands targeting GABA transporters, butyrylcholinesterase, beta-secretase, and amyloid beta aggregation as potential treatment of Alzheimer's disease - Zareba_2023_Eur.J.Med.Chem_261_115832
Author(s) : Zareba P , Latka K , Mazur G , Gryzlo B , Pasieka A , Godyn J , Panek D , Skrzypczak-Wiercioch A , Hofner GC , Latacz G , Maj M , Espargaro A , Sabate R , Jozwiak K , Wanner KT , Salat K , Malawska B , Kulig K , Bajda M
Ref : Eur Journal of Medicinal Chemistry , 261 :115832 , 2023
Abstract : Zareba_2023_Eur.J.Med.Chem_261_115832
ESTHER : Zareba_2023_Eur.J.Med.Chem_261_115832
PubMedSearch : Zareba_2023_Eur.J.Med.Chem_261_115832
PubMedID: 37837674

Title : New cyclopentaquinoline and 3,5-dichlorobenzoic acid hybrids with neuroprotection against oxidative stress for the treatment of Alzheimer's disease - Czarnecka_2023_J.Enzyme.Inhib.Med.Chem_38_2158822
Author(s) : Czarnecka K , Girek M , Krecisz P , Skibinski R , Latka K , Jonczyk J , Bajda M , Szymczyk P , Galita G , Kabzinski J , Majsterek I , Espargaro A , Sabate R , Szymanski P
Ref : J Enzyme Inhib Med Chem , 38 :2158822 , 2023
Abstract : Czarnecka_2023_J.Enzyme.Inhib.Med.Chem_38_2158822
ESTHER : Czarnecka_2023_J.Enzyme.Inhib.Med.Chem_38_2158822
PubMedSearch : Czarnecka_2023_J.Enzyme.Inhib.Med.Chem_38_2158822
PubMedID: 36629422

Title : Three to Tango: Inhibitory Effect of Quercetin and Apigenin on Acetylcholinesterase, Amyloid- Aggregation and Acetylcholinesterase-Amyloid Interaction - Alvarez-Berbel_2022_Pharmaceutics_14_
Author(s) : Alvarez-Berbel I , Espargaro A , Viayna A , Caballero AB , Busquets MA , Gamez P , Luque FJ , Sabate R
Ref : Pharmaceutics , 14 : , 2022
Abstract : Alvarez-Berbel_2022_Pharmaceutics_14_
ESTHER : Alvarez-Berbel_2022_Pharmaceutics_14_
PubMedSearch : Alvarez-Berbel_2022_Pharmaceutics_14_
PubMedID: 36365159

Title : Design, Synthesis, and In Vitro, In Silico and In Cellulo Evaluation of New Pyrimidine and Pyridine Amide and Carbamate Derivatives as Multi-Functional Cholinesterase Inhibitors - Bortolami_2022_Pharmaceuticals.(Basel)_15_
Author(s) : Bortolami M , Pandolfi F , Tudino V , Messore A , Madia VN , De Vita D , Di Santo R , Costi R , Romeo I , Alcaro S , Colone M , Stringaro A , Espargaro A , Sabate R , Scipione L
Ref : Pharmaceuticals (Basel) , 15 : , 2022
Abstract : Bortolami_2022_Pharmaceuticals.(Basel)_15_
ESTHER : Bortolami_2022_Pharmaceuticals.(Basel)_15_
PubMedSearch : Bortolami_2022_Pharmaceuticals.(Basel)_15_
PubMedID: 35745594

Title : Azobioisosteres of Curcumin with Pronounced Activity against Amyloid Aggregation, Intracellular Oxidative Stress, and Neuroinflammation - Hofmann_2021_Chemistry_27_6015
Author(s) : Hofmann J , Ginex T , Espargaro A , Scheiner M , Gunesch S , Arago M , Stigloher C , Sabate R , Luque FJ , Decker M
Ref : Chemistry , 27 :6015 , 2021
Abstract : Hofmann_2021_Chemistry_27_6015
ESTHER : Hofmann_2021_Chemistry_27_6015
PubMedSearch : Hofmann_2021_Chemistry_27_6015
PubMedID: 33666306

Title : Dual Effect of Prussian Blue Nanoparticles on Abeta40 Aggregation: beta-Sheet Fibril Reduction and Copper Dyshomeostasis Regulation - Kowalczyk_2021_Biomacromolecules__
Author(s) : Kowalczyk J , Grapsi E , Espargaro A , Caballero AB , Juarez-Jimenez J , Busquets MA , Gamez P , Sabate R , Estelrich J
Ref : Biomacromolecules , : , 2021
Abstract : Kowalczyk_2021_Biomacromolecules__
ESTHER : Kowalczyk_2021_Biomacromolecules__
PubMedSearch : Kowalczyk_2021_Biomacromolecules__
PubMedID: 33416315

Title : New Pyrimidine and Pyridine Derivatives as Multitarget Cholinesterase Inhibitors: Design, Synthesis, and In Vitro and In Cellulo Evaluation - Bortolami_2021_ACS.Chem.Neurosci__
Author(s) : Bortolami M , Pandolfi F , Tudino V , Messore A , Madia VN , De Vita D , Di Santo R , Costi R , Romeo I , Alcaro S , Colone M , Stringaro A , Espargaro A , Sabate R , Scipione L
Ref : ACS Chem Neurosci , : , 2021
Abstract : Bortolami_2021_ACS.Chem.Neurosci__
ESTHER : Bortolami_2021_ACS.Chem.Neurosci__
PubMedSearch : Bortolami_2021_ACS.Chem.Neurosci__
PubMedID: 34652128

Title : Centrally Active Multitarget Anti-Alzheimer Agents Derived from the Antioxidant Lead CR-6 - Perez-Areales_2020_J.Med.Chem_63_9360
Author(s) : Perez-Areales FJ , Garrido M , Aso E , Bartolini M , De Simone A , Espargaro A , Ginex T , Sabate R , Perez B , Andrisano V , Puigoriol-Illamola D , Pallas M , Luque FJ , Loza MI , Brea J , Ferrer I , Ciruela F , Messeguer A , Munoz-Torrero D
Ref : Journal of Medicinal Chemistry , 63 :9360 , 2020
Abstract : Perez-Areales_2020_J.Med.Chem_63_9360
ESTHER : Perez-Areales_2020_J.Med.Chem_63_9360
PubMedSearch : Perez-Areales_2020_J.Med.Chem_63_9360
PubMedID: 32706255

Title : A novel class of multitarget anti-Alzheimer benzohomoadamantanechlorotacrine hybrids modulating cholinesterases and glutamate NMDA receptors - Perez-Areales_2019_Eur.J.Med.Chem_180_613
Author(s) : Perez-Areales FJ , Turcu AL , Barniol-Xicota M , Pont C , Pivetta D , Espargaro A , Bartolini M , De Simone A , Andrisano V , Perez B , Sabate R , Sureda FX , Vazquez S , Munoz-Torrero D
Ref : Eur Journal of Medicinal Chemistry , 180 :613 , 2019
Abstract : Perez-Areales_2019_Eur.J.Med.Chem_180_613
ESTHER : Perez-Areales_2019_Eur.J.Med.Chem_180_613
PubMedSearch : Perez-Areales_2019_Eur.J.Med.Chem_180_613
PubMedID: 31351393

Title : Design, synthesis and multitarget biological profiling of second-generation anti-Alzheimer rhein-huprine hybrids - Perez-Areales_2017_Future.Med.Chem_9_965
Author(s) : Perez-Areales FJ , Betari N , Viayna A , Pont C , Espargaro A , Bartolini M , De Simone A , Rinaldi Alvarenga JF , Perez B , Sabate R , Lamuela-Raventos RM , Andrisano V , Luque FJ , Munoz-Torrero D
Ref : Future Med Chem , 9 :965 , 2017
Abstract : Perez-Areales_2017_Future.Med.Chem_9_965
ESTHER : Perez-Areales_2017_Future.Med.Chem_9_965
PubMedSearch : Perez-Areales_2017_Future.Med.Chem_9_965
PubMedID: 28632395

Title : Novel Levetiracetam Derivatives That Are Effective against the Alzheimer-like Phenotype in Mice: Synthesis, in Vitro, ex Vivo, and in Vivo Efficacy Studies - Sola_2015_J.Med.Chem_58_6018
Author(s) : Sola I , Aso E , Frattini D , Lopez-Gonzalez I , Espargaro A , Sabate R , Di Pietro O , Luque FJ , Clos MV , Ferrer I , Munoz-Torrero D
Ref : Journal of Medicinal Chemistry , 58 :6018 , 2015
Abstract : Sola_2015_J.Med.Chem_58_6018
ESTHER : Sola_2015_J.Med.Chem_58_6018
PubMedSearch : Sola_2015_J.Med.Chem_58_6018
PubMedID: 26181606

Title : Shogaol-huprine hybrids: Dual antioxidant and anticholinesterase agents with beta-amyloid and tau anti-aggregating properties - Perez-Areales_2014_Bioorg.Med.Chem_22_5298
Author(s) : Perez-Areales FJ , Di Pietro O , Espargaro A , Vallverdu-Queralt A , Galdeano C , Ragusa IM , Viayna E , Guillou C , Clos MV , Perez B , Sabate R , Lamuela-Raventos RM , Luque FJ , Munoz-Torrero D
Ref : Bioorganic & Medicinal Chemistry , 22 :5298 , 2014
Abstract : Perez-Areales_2014_Bioorg.Med.Chem_22_5298
ESTHER : Perez-Areales_2014_Bioorg.Med.Chem_22_5298
PubMedSearch : Perez-Areales_2014_Bioorg.Med.Chem_22_5298
PubMedID: 25156301

Title : Tetrahydrobenzo[h][1,6]naphthyridine-6-chlorotacrine hybrids as a new family of anti-Alzheimer agents targeting beta-amyloid, tau, and cholinesterase pathologies - Di Pietro_2014_Eur.J.Med.Chem_84C_107
Author(s) : Di Pietro O , Perez-Areales FJ , Juarez-Jimenez J , Espargaro A , Clos MV , Perez B , Lavilla R , Sabate R , Luque FJ , Munoz-Torrero D
Ref : Eur Journal of Medicinal Chemistry , 84C :107 , 2014
Abstract : Di Pietro_2014_Eur.J.Med.Chem_84C_107
ESTHER : Di Pietro_2014_Eur.J.Med.Chem_84C_107
PubMedSearch : Di Pietro_2014_Eur.J.Med.Chem_84C_107
PubMedID: 25016233