Thakur GA

General

Full name : Thakur Ganeshsingh A

First name : Ganeshsingh A

Mail : Dept. of Pharmaceutical Sciences and Center for Drug Discovery, Northeastern University, Boston, MA 02115

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Country : USA

Email : g.thakur@neu.edu

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Comment

References (8)

Title : Heteromeric Neuronal Nicotinic Acetylcholine Receptors with Mutant beta Subunits Acquire Sensitivity to alpha7-Selective Positive Allosteric Modulators - Stokes_2019_J.Pharmacol.Exp.Ther_370_252
Author(s) : Stokes C , Garai S , Kulkarni AR , Cantwell LN , Noviello CM , Hibbs RE , Horenstein NA , Abboud KA , Thakur GA , Papke RL
Ref : Journal of Pharmacology & Experimental Therapeutics , 370 :252 , 2019
Abstract :
PubMedSearch : Stokes_2019_J.Pharmacol.Exp.Ther_370_252
PubMedID: 31175218

Title : The Activity of GAT107, an Allosteric Activator and Positive Modulator of alpha7 Nicotinic Acetylcholine Receptors (nAChR), Is Regulated by Aromatic Amino Acids That Span the Subunit Interface - Papke_2014_J.Biol.Chem_289_4515
Author(s) : Papke RL , Horenstein NA , Kulkarni AR , Stokes C , Corrie LW , Maeng CY , Thakur GA
Ref : Journal of Biological Chemistry , 289 :4515 , 2014
Abstract :
PubMedSearch : Papke_2014_J.Biol.Chem_289_4515
PubMedID: 24362025

Title : Novel adamantyl cannabinoids as CB1 receptor probes - Thakur_2013_J.Med.Chem_56_3904
Author(s) : Thakur GA , Bajaj S , Paronis C , Peng Y , Bowman AL , Barak LS , Caron MG , Parrish D , Deschamps JR , Makriyannis A
Ref : Journal of Medicinal Chemistry , 56 :3904 , 2013
Abstract :
PubMedSearch : Thakur_2013_J.Med.Chem_56_3904
PubMedID: 23621789

Title : Expeditious synthesis, enantiomeric resolution, and enantiomer functional characterization of (4-(4-bromophenyl)-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-8-sulfonamide (4BP-TQS): an allosteric agonist-positive allosteric modulator of alpha7 nicotinic acetylcholine receptors - Thakur_2013_J.Med.Chem_56_8943
Author(s) : Thakur GA , Kulkarni AR , Deschamps JR , Papke RL
Ref : Journal of Medicinal Chemistry , 56 :8943 , 2013
Abstract :
PubMedSearch : Thakur_2013_J.Med.Chem_56_8943
PubMedID: 24090443

Title : Analysis of tolerance and behavioral\/physical dependence during chronic CB1 agonist treatment: effects of CB1 agonists, antagonists, and noncannabinoid drugs - Desai_2013_J.Pharmacol.Exp.Ther_344_319
Author(s) : Desai RI , Thakur GA , Vemuri VK , Bajaj S , Makriyannis A , Bergman J
Ref : Journal of Pharmacology & Experimental Therapeutics , 344 :319 , 2013
Abstract :
PubMedSearch : Desai_2013_J.Pharmacol.Exp.Ther_344_319
PubMedID: 23197773

Title : The novel cannabinoid CB1 receptor neutral antagonist AM4113 suppresses food intake and food-reinforced behavior but does not induce signs of nausea in rats - Sink_2008_Neuropsychopharmacology_33_946
Author(s) : Sink KS , McLaughlin PJ , Wood JA , Brown C , Fan P , Vemuri VK , Peng Y , Olszewska T , Thakur GA , Makriyannis A , Parker LA , Salamone JD
Ref : Neuropsychopharmacology , 33 :946 , 2008
Abstract :
PubMedSearch : Sink_2008_Neuropsychopharmacology_33_946
PubMedID: 17581535

Title : Cannabilactones: a novel class of CB2 selective agonists with peripheral analgesic activity - Khanolkar_2007_J.Med.Chem_50_6493
Author(s) : Khanolkar AD , Lu D , Ibrahim M , Duclos RI, Jr. , Thakur GA , Malan TP, Jr. , Porreca F , Veerappan V , Tian X , George C , Parrish DA , Papahatjis DP , Makriyannis A
Ref : Journal of Medicinal Chemistry , 50 :6493 , 2007
Abstract :
PubMedSearch : Khanolkar_2007_J.Med.Chem_50_6493
PubMedID: 18038967

Title : Adamantyl cannabinoids: a novel class of cannabinergic ligands - Lu_2005_J.Med.Chem_48_4576
Author(s) : Lu D , Meng Z , Thakur GA , Fan P , Steed J , Tartal CL , Hurst DP , Reggio PH , Deschamps JR , Parrish DA , George C , Jarbe TU , Lamb RJ , Makriyannis A
Ref : Journal of Medicinal Chemistry , 48 :4576 , 2005
Abstract :
PubMedSearch : Lu_2005_J.Med.Chem_48_4576
PubMedID: 15999995