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Title : Selective Inhibitors of Fibroblast Activation Protein (FAP) with a (4-Quinolinoyl)-glycyl-2-cyanopyrrolidine Scaffold - Jansen_2013_ACS.Med.Chem.Lett_4_491 |
Author(s) : Jansen K , Heirbaut L , Cheng JD , Joossens J , Ryabtsova O , Cos P , Maes L , Lambeir AM , De Meester I , Augustyns K , Van der Veken P |
Ref : ACS Med Chem Lett , 4 :491 , 2013 |
Abstract : Jansen_2013_ACS.Med.Chem.Lett_4_491 |
ESTHER : Jansen_2013_ACS.Med.Chem.Lett_4_491 |
PubMedSearch : Jansen_2013_ACS.Med.Chem.Lett_4_491 |
PubMedID: 24900696 |
Title : Acylated Gly-(2-cyano)pyrrolidines as inhibitors of fibroblast activation protein (FAP) and the issue of FAP\/prolyl oligopeptidase (PREP)-selectivity - Ryabtsova_2012_Bioorg.Med.Chem.Lett_22_3412 |
Author(s) : Ryabtsova O , Jansen K , Van Goethem S , Joossens J , Cheng JD , Lambeir AM , De Meester I , Augustyns K , Van der Veken P |
Ref : Bioorganic & Medicinal Chemistry Lett , 22 :3412 , 2012 |
Abstract : Ryabtsova_2012_Bioorg.Med.Chem.Lett_22_3412 |
ESTHER : Ryabtsova_2012_Bioorg.Med.Chem.Lett_22_3412 |
PubMedSearch : Ryabtsova_2012_Bioorg.Med.Chem.Lett_22_3412 |
PubMedID: 22525314 |