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| Title : Inhibitors of the Thioesterase Activity of Mycobacterium tuberculosis Pks13 Discovered Using DNA-Encoded Chemical Library Screening - Krieger_2024_ACS.Infect.Dis__ |
| Author(s) : Krieger IV , Yalamanchili S , Dickson P , Engelhart CA , Zimmerman MD , Wood J , Clary E , Nguyen J , Thornton N , Centrella PA , Chan B , Cuozzo JW , Gengenbacher M , Guie MA , Guilinger JP , Bienstock C , Hartl H , Hupp CD , Jetson R , Satoh T , Yeoman JTS , Zhang Y , Dartois V , Schnappinger D , Keefe AD , Sacchettini JC |
| Ref : ACS Infect Dis , : , 2024 |
| Abstract : Krieger_2024_ACS.Infect.Dis__ |
| ESTHER : Krieger_2024_ACS.Infect.Dis__ |
| PubMedSearch : Krieger_2024_ACS.Infect.Dis__ |
| PubMedID: 38577994 |
| Title : Identification and Optimization of Novel Inhibitors of the Polyketide Synthase 13 Thioesterase Domain with Antitubercular Activity - Green_2023_J.Med.Chem__ |
| Author(s) : Green SR , Wilson C , Eadsforth TC , Punekar AS , Tamaki FK , Wood G , Caldwell N , Forte B , Norcross NR , Kiczun M , Post JM , Lopez-Roman EM , Engelhart CA , Lukac I , Zuccotto F , Epemolu O , Boshoff HIM , Schnappinger D , Walpole C , Gilbert IH , Read KD , Wyatt PG , Baragana B |
| Ref : Journal of Medicinal Chemistry , : , 2023 |
| Abstract : Green_2023_J.Med.Chem__ |
| ESTHER : Green_2023_J.Med.Chem__ |
| PubMedSearch : Green_2023_J.Med.Chem__ |
| PubMedID: 37948640 |
| Gene_locus related to this paper: myctu-PKS13 |
| Title : Optimization of TAM16, a Benzofuran That Inhibits the Thioesterase Activity of Pks13\; Evaluation toward a Preclinical Candidate for a Novel Antituberculosis Clinical Target - Wilson_2022_J.Med.Chem_65_409 |
| Author(s) : Wilson C , Ray P , Zuccotto F , Hernandez J , Aggarwal A , Mackenzie C , Caldwell N , Taylor M , Huggett M , Mathieson M , Murugesan D , Smith A , Davis S , Cocco M , Parai MK , Acharya A , Tamaki F , Scullion P , Epemolu O , Riley J , Stojanovski L , Lopez-Roman EM , Torres-Gomez PA , Toledo AM , Guijarro-Lopez L , Camino I , Engelhart CA , Schnappinger D , Massoudi LM , Lenaerts A , Robertson GT , Walpole C , Matthews D , Floyd D , Sacchettini JC , Read KD , Encinas L , Bates RH , Green SR , Wyatt PG |
| Ref : Journal of Medicinal Chemistry , 65 :409 , 2022 |
| Abstract : Wilson_2022_J.Med.Chem_65_409 |
| ESTHER : Wilson_2022_J.Med.Chem_65_409 |
| PubMedSearch : Wilson_2022_J.Med.Chem_65_409 |
| PubMedID: 34910486 |
| Gene_locus related to this paper: myctu-PKS13 |
| Title : Inhibition of respiration by nitric oxide induces a Mycobacterium tuberculosis dormancy program - Voskuil_2003_J.Exp.Med_198_705 |
| Author(s) : Voskuil MI , Schnappinger D , Visconti KC , Harrell MI , Dolganov GM , Sherman DR , Schoolnik GK |
| Ref : J Exp Med , 198 :705 , 2003 |
| Abstract : Voskuil_2003_J.Exp.Med_198_705 |
| ESTHER : Voskuil_2003_J.Exp.Med_198_705 |
| PubMedSearch : Voskuil_2003_J.Exp.Med_198_705 |
| PubMedID: 12953092 |
| Gene_locus related to this paper: myctu-RV2627C , myctu-y0571 |