Title : N,N'-Alkane-diyl-bis-3-picoliniums as nicotinic receptor antagonists: inhibition of nicotine-evoked dopamine release and hyperactivity - Dwoskin_2008_J.Pharmacol.Exp.Ther_326_563 |
Author(s) : Dwoskin LP , Wooters TE , Sumithran SP , Siripurapu KB , Joyce BM , Lockman PR , Manda VK , Ayers JT , Zhang Z , Deaciuc AG , McIntosh JM , Crooks PA , Bardo MT |
Ref : Journal of Pharmacology & Experimental Therapeutics , 326 :563 , 2008 |
Abstract : |
PubMedSearch : Dwoskin_2008_J.Pharmacol.Exp.Ther_326_563 |
PubMedID: 18460644 |
Title : QSAR modeling of mono- and bis-quaternary ammonium salts that act as antagonists at neuronal nicotinic acetylcholine receptors mediating dopamine release - Zheng_2006_Bioorg.Med.Chem_14_3017 |
Author(s) : Zheng F , Bayram E , Sumithran SP , Ayers JT , Zhan CG , Schmitt JD , Dwoskin LP , Crooks PA |
Ref : Bioorganic & Medicinal Chemistry , 14 :3017 , 2006 |
Abstract : |
PubMedSearch : Zheng_2006_Bioorg.Med.Chem_14_3017 |
PubMedID: 16431111 |
Title : N-n-alkylnicotinium analogs, a novel class of antagonists at alpha 4 beta 2* nicotinic acetylcholine receptors: inhibition of S(-)-nicotine-evoked 86Rb+ efflux from rat thalamic synaptosomes - Wilkins_2005_AAPS.J_7_E922 |
Author(s) : Wilkins LH, Jr. , Miller DK , Ayers JT , Crooks PA , Dwoskin LP |
Ref : AAPS J , 7 :E922 , 2005 |
Abstract : |
PubMedSearch : Wilkins_2005_AAPS.J_7_E922 |
PubMedID: 16594645 |
Title : Molecular modeling of mono- and bis-quaternary ammonium salts as ligands at the alpha4beta2 nicotinic acetylcholine receptor subtype using nonlinear techniques - Ayers_2005_AAPS.J_7_E678 |
Author(s) : Ayers JT , Clauset A , Schmitt JD , Dwoskin LP , Crooks PA |
Ref : AAPS J , 7 :E678 , 2005 |
Abstract : |
PubMedSearch : Ayers_2005_AAPS.J_7_E678 |
PubMedID: 16353944 |
Title : A general procedure for the enantioselective synthesis of the minor tobacco alkaloids nornicotine, anabasine, and anatabine - Ayers_2005_AAPS.J_7_E752 |
Author(s) : Ayers JT , Xu R , Dwoskin LP , Crooks PA |
Ref : AAPS J , 7 :E752 , 2005 |
Abstract : |
PubMedSearch : Ayers_2005_AAPS.J_7_E752 |
PubMedID: 16353951 |
Title : Development of subtype-selective ligands as antagonists at nicotinic receptors mediating nicotine-evoked dopamine release - Crooks_2004_Bioorg.Med.Chem.Lett_14_1869 |
Author(s) : Crooks PA , Ayers JT , Xu R , Sumithran SP , Grinevich VP , Wilkins LH , Deaciuc AG , Allen DD , Dwoskin LP |
Ref : Bioorganic & Medicinal Chemistry Lett , 14 :1869 , 2004 |
Abstract : |
PubMedSearch : Crooks_2004_Bioorg.Med.Chem.Lett_14_1869 |
PubMedID: 15050618 |
Title : Subtype-selective nicotinic receptor antagonists: potential as tobacco use cessation agents - Dwoskin_2004_Bioorg.Med.Chem.Lett_14_1863 |
Author(s) : Dwoskin LP , Sumithran SP , Zhu J , Deaciuc AG , Ayers JT , Crooks PA |
Ref : Bioorganic & Medicinal Chemistry Lett , 14 :1863 , 2004 |
Abstract : |
PubMedSearch : Dwoskin_2004_Bioorg.Med.Chem.Lett_14_1863 |
PubMedID: 15050617 |
Title : N-n-alkylnicotinium analogs, a novel class of nicotinic receptor antagonists: interaction with alpha4beta2* and alpha7* neuronal nicotinic receptors - Wilkins_2003_J.Pharmacol.Exp.Ther_304_400 |
Author(s) : Wilkins LH, Jr. , Grinevich VP , Ayers JT , Crooks PA , Dwoskin LP |
Ref : Journal of Pharmacology & Experimental Therapeutics , 304 :400 , 2003 |
Abstract : |
PubMedSearch : Wilkins_2003_J.Pharmacol.Exp.Ther_304_400 |
PubMedID: 12490617 |
Title : N-n-alkylpyridinium analogs, a novel class of nicotinic receptor antagonists: selective inhibition of nicotine-evoked [3H] dopamine overflow from superfused rat striatal slices - Grinevich_2003_J.Pharmacol.Exp.Ther_306_1011 |
Author(s) : Grinevich VP , Crooks PA , Sumithran SP , Haubner AJ , Ayers JT , Dwoskin LP |
Ref : Journal of Pharmacology & Experimental Therapeutics , 306 :1011 , 2003 |
Abstract : |
PubMedSearch : Grinevich_2003_J.Pharmacol.Exp.Ther_306_1011 |
PubMedID: 12766255 |
Title : N-n-alkylnicotinium analogs, a novel class of nicotinic receptor antagonist: inhibition of S(-)-nicotine-evoked [(3)H]dopamine overflow from superfused rat striatal slices - Wilkins_2002_J.Pharmacol.Exp.Ther_301_1088 |
Author(s) : Wilkins LH, Jr. , Haubner A , Ayers JT , Crooks PA , Dwoskin LP |
Ref : Journal of Pharmacology & Experimental Therapeutics , 301 :1088 , 2002 |
Abstract : |
PubMedSearch : Wilkins_2002_J.Pharmacol.Exp.Ther_301_1088 |
PubMedID: 12023541 |
Title : bis-Azaaromatic quaternary ammonium analogues: ligands for alpha4beta2* and alpha7* subtypes of neuronal nicotinic receptors - Ayers_2002_Bioorg.Med.Chem.Lett_12_3067 |
Author(s) : Ayers JT , Dwoskin LP , Deaciuc AG , Grinevich VP , Zhu J , Crooks PA |
Ref : Bioorganic & Medicinal Chemistry Lett , 12 :3067 , 2002 |
Abstract : |
PubMedSearch : Ayers_2002_Bioorg.Med.Chem.Lett_12_3067 |
PubMedID: 12372503 |