Title : Predictive screening model for potential vector-mediated transport of cationic substrates at the blood-brain barrier choline transporter - Geldenhuys_2010_Bioorg.Med.Chem.Lett_20_870 |
Author(s) : Geldenhuys WJ , Manda VK , Mittapalli RK , Van der Schyf CJ , Crooks PA , Dwoskin LP , Allen DD , Lockman PR |
Ref : Bioorganic & Medicinal Chemistry Lett , 20 :870 , 2010 |
Abstract : |
PubMedSearch : Geldenhuys_2010_Bioorg.Med.Chem.Lett_20_870 |
PubMedID: 20053562 |
Title : N,N'-Alkane-diyl-bis-3-picoliniums as nicotinic receptor antagonists: inhibition of nicotine-evoked dopamine release and hyperactivity - Dwoskin_2008_J.Pharmacol.Exp.Ther_326_563 |
Author(s) : Dwoskin LP , Wooters TE , Sumithran SP , Siripurapu KB , Joyce BM , Lockman PR , Manda VK , Ayers JT , Zhang Z , Deaciuc AG , McIntosh JM , Crooks PA , Bardo MT |
Ref : Journal of Pharmacology & Experimental Therapeutics , 326 :563 , 2008 |
Abstract : |
PubMedSearch : Dwoskin_2008_J.Pharmacol.Exp.Ther_326_563 |
PubMedID: 18460644 |
Title : Carrier-mediated transport of the quaternary ammonium neuronal nicotinic receptor antagonist n,n'-dodecylbispicolinium dibromide at the blood-brain barrier - Lockman_2008_J.Pharmacol.Exp.Ther_324_244 |
Author(s) : Lockman PR , Manda VK , Geldenhuys WJ , Mittapalli RK , Thomas F , Albayati ZF , Crooks PA , Dwoskin LP , Allen DD |
Ref : Journal of Pharmacology & Experimental Therapeutics , 324 :244 , 2008 |
Abstract : |
PubMedSearch : Lockman_2008_J.Pharmacol.Exp.Ther_324_244 |
PubMedID: 17921191 |
Title : Discovery of a novel nicotinic receptor antagonist for the treatment of nicotine addiction: 1-(3-Picolinium)-12-triethylammonium-dodecane dibromide (TMPD) - Dwoskin_2007_Biochem.Pharmacol_74(8)_1271 |
Author(s) : Dwoskin LP , Joyce BM , Zheng G , Neugebauer NM , Manda VK , Lockman P , Papke RL , Bardo MT , Crooks PA |
Ref : Biochemical Pharmacology , 74 :1271 , 2007 |
Abstract : |
PubMedSearch : Dwoskin_2007_Biochem.Pharmacol_74(8)_1271 |
PubMedID: 17727820 |