Title : Assessing the Potential of 1,2,3-Triazole-Dihydropyrimidinone Hybrids Against Cholinesterases: In Silico, In Vitro, and In Vivo Studies - Gastalho_2024_Int.J.Mol.Sci_25_ |
Author(s) : Gastalho CM , Sena AM , Lopez O , Fernandez-Bolanos JG , Garcia-Sosa AT , Pereira F , Antunes CM , Costa AR , Burke AJ , Carreiro EP |
Ref : Int J Mol Sci , 25 : , 2024 |
Abstract : |
PubMedSearch : Gastalho_2024_Int.J.Mol.Sci_25_ |
PubMedID: 39456935 |
Title : Quercetin-1,2,3-Triazole Hybrids as Multifunctional Anti-Alzheimer's Agents - Carreiro_2023_Molecules_28_ |
Author(s) : Carreiro EP , Costa AR , Antunes CM , Ernesto S , Pinto F , Rodrigues B , Burke AJ |
Ref : Molecules , 28 : , 2023 |
Abstract : |
PubMedSearch : Carreiro_2023_Molecules_28_ |
PubMedID: 38005217 |
Title : Evaluation of chromane derivatives: Promising privileged scaffolds for lead discovery within Alzheimer's disease - Moutayakine_2022_Bioorg.Med.Chem_68_116807 |
Author(s) : Moutayakine A , Marques C , Lopez O , Bagetta D , Leitzbach L , Hagenow S , Carreiro EP , Stark H , Alcaro S , Fernandez-Bolanos JG , Burke AJ |
Ref : Bioorganic & Medicinal Chemistry , 68 :116807 , 2022 |
Abstract : |
PubMedSearch : Moutayakine_2022_Bioorg.Med.Chem_68_116807 |
PubMedID: 35653868 |
Title : Ugi Reaction Synthesis of Oxindole-Lactam Hybrids as Selective Butyrylcholinesterase Inhibitors - Brandao_2021_ACS.Med.Chem.Lett_12_1718 |
Author(s) : Brandao P , Lopez O , Leitzbach L , Stark H , Fernandez-Bolanos JG , Burke AJ , Pineiro M |
Ref : ACS Med Chem Lett , 12 :1718 , 2021 |
Abstract : |
PubMedSearch : Brandao_2021_ACS.Med.Chem.Lett_12_1718 |
PubMedID: 34795859 |
Title : N-1,2,3-triazole-isatin derivatives for cholinesterase and beta-amyloid aggregation inhibition: A comprehensive bioassay study - Marques_2020_Bioorg.Chem_98_103753 |
Author(s) : Marques CS , Lopez O , Bagetta D , Carreiro EP , Petralla S , Bartolini M , Hoffmann M , Alcaro S , Monti B , Bolognesi ML , Decker M , Fernandez-Bolanos JG , Burke AJ |
Ref : Bioorg Chem , 98 :103753 , 2020 |
Abstract : |
PubMedSearch : Marques_2020_Bioorg.Chem_98_103753 |
PubMedID: 32200328 |
Title : In silico, NMR and pharmacological evaluation of an hydroxyoxindole cholinesterase inhibitor - Bacalhau_2019_Bioorg.Med.Chem_27_354 |
Author(s) : Bacalhau P , Fernandes L , Rosario Martins M , Candeias F , Carreiro EP , Lopez O , Teresa Caldeira A , Totobenazara J , Guedes RC , Burke AJ |
Ref : Bioorganic & Medicinal Chemistry , 27 :354 , 2019 |
Abstract : |
PubMedSearch : Bacalhau_2019_Bioorg.Med.Chem_27_354 |
PubMedID: 30578075 |
Title : Insights into (S)-rivastigmine inhibition of butyrylcholinesterase (BuChE): Molecular docking and saturation transfer difference NMR (STD-NMR) - Bacalhau_2016_Bioorg.Chem_67_105 |
Author(s) : Bacalhau P , San Juan AA , Goth A , Caldeira AT , Martins R , Burke AJ |
Ref : Bioorg Chem , 67 :105 , 2016 |
Abstract : |
PubMedSearch : Bacalhau_2016_Bioorg.Chem_67_105 |
PubMedID: 27317888 |
Title : New cholinesterase inhibitors for Alzheimer's disease: Structure Activity Studies (SARs) and molecular docking of isoquinolone and azepanone derivatives - Bacalhau_2016_Bioorg.Chem_67_1 |
Author(s) : Bacalhau P , San Juan AA , Marques CS , Peixoto D , Goth A , Guarda C , Silva M , Arantes S , Caldeira AT , Martins R , Burke AJ |
Ref : Bioorg Chem , 67 :1 , 2016 |
Abstract : |
PubMedSearch : Bacalhau_2016_Bioorg.Chem_67_1 |
PubMedID: 27231829 |