Title : Novel multifunctional tacrine-donepezil hybrids against Alzheimer's disease: Design synthesis and bioactivity studies - Bayraktar_2024_Arch.Pharm.(Weinheim)__e2300575 |
Author(s) : Bayraktar G , Bartolini M , Bolognesi ML , Erdogan MA , Armagan G , Bayir E , Sendemir A , Bagetta D , Alcaro S , Alptuzun V |
Ref : Arch Pharm (Weinheim) , :e2300575 , 2024 |
Abstract : |
PubMedSearch : Bayraktar_2024_Arch.Pharm.(Weinheim)__e2300575 |
PubMedID: 38593283 |
Title : Evaluation of chromane derivatives: Promising privileged scaffolds for lead discovery within Alzheimer's disease - Moutayakine_2022_Bioorg.Med.Chem_68_116807 |
Author(s) : Moutayakine A , Marques C , Lopez O , Bagetta D , Leitzbach L , Hagenow S , Carreiro EP , Stark H , Alcaro S , Fernandez-Bolanos JG , Burke AJ |
Ref : Bioorganic & Medicinal Chemistry , 68 :116807 , 2022 |
Abstract : |
PubMedSearch : Moutayakine_2022_Bioorg.Med.Chem_68_116807 |
PubMedID: 35653868 |
Title : N-1,2,3-triazole-isatin derivatives for cholinesterase and beta-amyloid aggregation inhibition: A comprehensive bioassay study - Marques_2020_Bioorg.Chem_98_103753 |
Author(s) : Marques CS , Lopez O , Bagetta D , Carreiro EP , Petralla S , Bartolini M , Hoffmann M , Alcaro S , Monti B , Bolognesi ML , Decker M , Fernandez-Bolanos JG , Burke AJ |
Ref : Bioorg Chem , 98 :103753 , 2020 |
Abstract : |
PubMedSearch : Marques_2020_Bioorg.Chem_98_103753 |
PubMedID: 32200328 |
Title : New deferiprone derivatives as multi-functional cholinesterase inhibitors: design, synthesis and in vitro evaluation - Bortolami_2020_Eur.J.Med.Chem_198_112350 |
Author(s) : Bortolami M , Pandolfi F , De Vita D , Carafa C , Messore A , Di Santo R , Feroci M , Costi R , Chiarotto I , Bagetta D , Alcaro S , Colone M , Stringaro A , Scipione L |
Ref : Eur Journal of Medicinal Chemistry , 198 :112350 , 2020 |
Abstract : |
PubMedSearch : Bortolami_2020_Eur.J.Med.Chem_198_112350 |
PubMedID: 32380385 |
Title : 4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis - Secci_2019_J.Enzyme.Inhib.Med.Chem_34_597 |
Author(s) : Secci D , Carradori S , Petzer A , Guglielmi P , D'Ascenzio M , Chimenti P , Bagetta D , Alcaro S , Zengin G , Petzer JP , Ortuso F |
Ref : J Enzyme Inhib Med Chem , 34 :597 , 2019 |
Abstract : |
PubMedSearch : Secci_2019_J.Enzyme.Inhib.Med.Chem_34_597 |
PubMedID: 30727777 |
Title : Benzoic acid-derived nitrones: A new class of potential acetylcholinesterase inhibitors and neuroprotective agents - Oliveira_2019_Eur.J.Med.Chem_174_116 |
Author(s) : Oliveira C , Bagetta D , Cagide F , Teixeira J , Amorim R , Silva T , Garrido J , Remiao F , Uriarte E , Oliveira PJ , Alcaro S , Ortuso F , Borges F |
Ref : Eur Journal of Medicinal Chemistry , 174 :116 , 2019 |
Abstract : |
PubMedSearch : Oliveira_2019_Eur.J.Med.Chem_174_116 |
PubMedID: 31029943 |
Title : Multi-target-directed ligands for Alzheimer's disease: Discovery of chromone-based monoamine oxidase\/cholinesterase inhibitors - Reis_2018_Eur.J.Med.Chem_158_781 |
Author(s) : Reis J , Cagide F , Valencia ME , Teixeira J , Bagetta D , Perez C , Uriarte E , Oliveira PJ , Ortuso F , Alcaro S , Rodriguez-Franco MI , Borges F |
Ref : Eur Journal of Medicinal Chemistry , 158 :781 , 2018 |
Abstract : |
PubMedSearch : Reis_2018_Eur.J.Med.Chem_158_781 |
PubMedID: 30245401 |
Title : Design, synthesis and biochemical evaluation of novel multi-target inhibitors as potential anti-Parkinson agents - Carradori_2018_Eur.J.Med.Chem_143_1543 |
Author(s) : Carradori S , Ortuso F , Petzer A , Bagetta D , De Monte C , Secci D , De Vita D , Guglielmi P , Zengin G , Aktumsek A , Alcaro S , Petzer JP |
Ref : Eur Journal of Medicinal Chemistry , 143 :1543 , 2018 |
Abstract : |
PubMedSearch : Carradori_2018_Eur.J.Med.Chem_143_1543 |
PubMedID: 29126727 |