| Title : Novel 6-alkyl-bridged 4-arylalkylpiperazin-1-yl derivatives of azepino[4,3-b]indol-1(2H)-one as potent BChE-selective inhibitors showing protective effects against neurodegenerative insults - Samarelli_2024_Eur.J.Med.Chem_270_116353 |
| Author(s) : Samarelli F , Purgatorio R , Lopopolo G , Deruvo C , Catto M , Andresini M , Carrieri A , Nicolotti O , De Palma A , Miniero DV , de Candia M , Altomare CD |
| Ref : Eur Journal of Medicinal Chemistry , 270 :116353 , 2024 |
| Abstract : Samarelli_2024_Eur.J.Med.Chem_270_116353 |
| ESTHER : Samarelli_2024_Eur.J.Med.Chem_270_116353 |
| PubMedSearch : Samarelli_2024_Eur.J.Med.Chem_270_116353 |
| PubMedID: 38579622 |
| Title : Scouting around 1,2,3,4-Tetrahydrochromeno[3,2-c]pyridin-10-ones for Single- and Multi-target Ligands Directed towards Relevant Alzheimer's Targets - Purgatorio_2020_ChemMedChem_15_1947 |
| Author(s) : Purgatorio R , Kulikova L , Pisani L , Catto M , de Candia M , Carrieri A , Cellamare S , De Palma A , Beloglazkin A , Raesi GR , Voskressensky L , Altomare CD |
| Ref : ChemMedChem , 15 :1947 , 2020 |
| Abstract : Purgatorio_2020_ChemMedChem_15_1947 |
| ESTHER : Purgatorio_2020_ChemMedChem_15_1947 |
| PubMedSearch : Purgatorio_2020_ChemMedChem_15_1947 |
| PubMedID: 32716595 |
| Title : Investigating 1,2,3,4,5,6-hexahydroazepino[4,3-b]indole as scaffold of butyrylcholinesterase-selective inhibitors with additional neuroprotective activities for Alzheimer's disease - Purgatorio_2019_Eur.J.Med.Chem_177_414 |
| Author(s) : Purgatorio R , de Candia M , Catto M , Carrieri A , Pisani L , De Palma A , Toma M , Ivanova OA , Voskressensky LG , Altomare CD |
| Ref : Eur Journal of Medicinal Chemistry , 177 :414 , 2019 |
| Abstract : Purgatorio_2019_Eur.J.Med.Chem_177_414 |
| ESTHER : Purgatorio_2019_Eur.J.Med.Chem_177_414 |
| PubMedSearch : Purgatorio_2019_Eur.J.Med.Chem_177_414 |
| PubMedID: 31158754 |
| Title : Discovery of Potent Dual Binding Site Acetylcholinesterase Inhibitors via Homo- and Heterodimerization of Coumarin-Based Moieties - Pisani_2017_ChemMedChem_12_1349 |
| Author(s) : Pisani L , Catto M , De Palma A , Farina R , Cellamare S , Altomare CD |
| Ref : ChemMedChem , 12 :1349 , 2017 |
| Abstract : Pisani_2017_ChemMedChem_12_1349 |
| ESTHER : Pisani_2017_ChemMedChem_12_1349 |
| PubMedSearch : Pisani_2017_ChemMedChem_12_1349 |
| PubMedID: 28570763 |
| Title : Mannich base approach to 5-methoxyisatin 3-(4-isopropylphenyl)hydrazone: A water-soluble prodrug for a multitarget inhibition of cholinesterases, beta-amyloid fibrillization and oligomer-induced cytotoxicity - Pisani_2017_Eur.J.Pharm.Sci_109_381 |
| Author(s) : Pisani L , De Palma A , Giangregorio N , Miniero DV , Pesce P , Nicolotti O , Campagna F , Altomare CD , Catto M |
| Ref : Eur J Pharm Sci , 109 :381 , 2017 |
| Abstract : Pisani_2017_Eur.J.Pharm.Sci_109_381 |
| ESTHER : Pisani_2017_Eur.J.Pharm.Sci_109_381 |
| PubMedSearch : Pisani_2017_Eur.J.Pharm.Sci_109_381 |
| PubMedID: 28801274 |