Title : Novel 6-alkyl-bridged 4-arylalkylpiperazin-1-yl derivatives of azepino[4,3-b]indol-1(2H)-one as potent BChE-selective inhibitors showing protective effects against neurodegenerative insults - Samarelli_2024_Eur.J.Med.Chem_270_116353 |
Author(s) : Samarelli F , Purgatorio R , Lopopolo G , Deruvo C , Catto M , Andresini M , Carrieri A , Nicolotti O , De Palma A , Miniero DV , de Candia M , Altomare CD |
Ref : Eur Journal of Medicinal Chemistry , 270 :116353 , 2024 |
Abstract : Samarelli_2024_Eur.J.Med.Chem_270_116353 |
ESTHER : Samarelli_2024_Eur.J.Med.Chem_270_116353 |
PubMedSearch : Samarelli_2024_Eur.J.Med.Chem_270_116353 |
PubMedID: 38579622 |
Samarelli F, Purgatorio R, Lopopolo G, Deruvo C, Catto M, Andresini M, Carrieri A, Nicolotti O, De Palma A, Miniero DV, de Candia M, Altomare CD (2024)
Novel 6-alkyl-bridged 4-arylalkylpiperazin-1-yl derivatives of azepino[4,3-b]indol-1(2H)-one as potent BChE-selective inhibitors showing protective effects against neurodegenerative insults
Eur Journal of Medicinal Chemistry
270 :116353
Samarelli F, Purgatorio R, Lopopolo G, Deruvo C, Catto M, Andresini M, Carrieri A, Nicolotti O, De Palma A, Miniero DV, de Candia M, Altomare CD (2024)
Eur Journal of Medicinal Chemistry
270 :116353