Title : Structure-activity studies of diazabicyclo[3.3.0]octane-substituted pyrazines and pyridines as potent alpha4beta2 nicotinic acetylcholine receptor ligands - Scanio_2011_J.Med.Chem_54_7678 |
Author(s) : Scanio MJ , Shi L , Bunnelle WH , Anderson DJ , Helfrich RJ , Malysz J , Thorin-Hagene KK , Van Handel CE , Marsh KC , Lee CH , Gopalakrishnan M |
Ref : Journal of Medicinal Chemistry , 54 :7678 , 2011 |
Abstract : Scanio_2011_J.Med.Chem_54_7678 |
ESTHER : Scanio_2011_J.Med.Chem_54_7678 |
PubMedSearch : Scanio_2011_J.Med.Chem_54_7678 |
PubMedID: 21962147 |
Title : Preclinical characterization of A-582941: a novel alpha7 neuronal nicotinic receptor agonist with broad spectrum cognition-enhancing properties - Tietje_2008_CNS.Neurosci.Ther_14_65 |
Author(s) : Tietje KR , Anderson DJ , Bitner RS , Blomme EA , Brackemeyer PJ , Briggs CA , Browman KE , Bury D , Curzon P , Drescher KU , Frost JM , Fryer RM , Fox GB , Gronlien JH , Hakerud M , Gubbins EJ , Halm S , Harris R , Helfrich RJ , Kohlhaas KL , Law D , Malysz J , Marsh KC , Martin RL , Meyer MD , Molesky AL , Nikkel AL , Otte S , Pan L , Puttfarcken PS , Radek RJ , Robb HM , Spies E , Thorin-Hagene K , Waring JF , Ween H , Xu H , Gopalakrishnan M , Bunnelle WH |
Ref : CNS Neurosci Ther , 14 :65 , 2008 |
Abstract : Tietje_2008_CNS.Neurosci.Ther_14_65 |
ESTHER : Tietje_2008_CNS.Neurosci.Ther_14_65 |
PubMedSearch : Tietje_2008_CNS.Neurosci.Ther_14_65 |
PubMedID: 18482100 |
Title : Comparative pharmacology of human dopamine D(2)-like receptor stable cell lines coupled to calcium flux through Galpha(qo5) - Moreland_2004_Biochem.Pharmacol_68_761 |
Author(s) : Moreland RB , Nakane M , Donnelly-Roberts D , Miller LN , Chang R , Uchic ME , Terranova MA , Gubbins EJ , Helfrich RJ , Namovic MT , El-Kouhen OF , Masters JN , Brioni JD |
Ref : Biochemical Pharmacology , 68 :761 , 2004 |
Abstract : Moreland_2004_Biochem.Pharmacol_68_761 |
ESTHER : Moreland_2004_Biochem.Pharmacol_68_761 |
PubMedSearch : Moreland_2004_Biochem.Pharmacol_68_761 |
PubMedID: 15276084 |
Title : A cell-based microarrayed compound screening format for identifying agonists of G-protein-coupled receptors - Gopalakrishnan_2003_Anal.Biochem_321_192 |
Author(s) : Gopalakrishnan SM , Moreland RB , Kofron JL , Helfrich RJ , Gubbins E , McGowen J , Masters JN , Donnelly-Roberts D , Brioni JD , Burns DJ , Warrior U |
Ref : Analytical Biochemistry , 321 :192 , 2003 |
Abstract : Gopalakrishnan_2003_Anal.Biochem_321_192 |
ESTHER : Gopalakrishnan_2003_Anal.Biochem_321_192 |
PubMedSearch : Gopalakrishnan_2003_Anal.Biochem_321_192 |
PubMedID: 14511684 |