| Title : Targeting Neuroinflammation and Cognitive Decline: First-in-Class Dual Butyrylcholinesterase and p38alpha Mitogen-Activated Protein Kinase Inhibitors - Ferjancic Benetik_2025_J.Med.Chem__ |
| Author(s) : Ferjancic Benetik S , Proj M , Knez D , Kosak U , Meden A , Krajsek K , Pislar A , Horvat S , Svajger U , Tesic N , Pulkrabkova L , Soukup O , Skarka A , Andrys R , Brazzolotto X , Igert A , Nachon F , Dias J , Detka J , Gdula-Argasinska J , Wyska E , Szafarz M , Manik A , Plachtij N , Musilek K , Salat K , Obreza A , Gobec S |
| Ref : Journal of Medicinal Chemistry , : , 2025 |
| Abstract : |
| PubMedSearch : Ferjancic Benetik_2025_J.Med.Chem__ |
| PubMedID: 40779804 |
| Title : Targeting Neuroinflammation and Cognitive Decline: First-in-Class Dual Butyrylcholinesterase and p38alpha Mitogen-Activated Protein Kinase Inhibitors - Ferjancic Benetik_2025_J.Med.Chem__ |
| Author(s) : Ferjancic Benetik S , Proj M , Knez D , Kosak U , Meden A , Krajsek K , Pislar A , Horvat S , Svajger U , Tesic N , Pulkrabkova L , Soukup O , Skarka A , Andrys R , Brazzolotto X , Igert A , Nachon F , Dias J , Detka J , Gdula-Argasinska J , Wyska E , Szafarz M , Manik A , Plachtij N , Musilek K , Salat K , Obreza A , Gobec S |
| Ref : Journal of Medicinal Chemistry , : , 2025 |
| Abstract : |
| PubMedSearch : Ferjancic Benetik_2025_J.Med.Chem__ |
| PubMedID: 40779804 |
| Title : N-Propargylpyrrolidine-based butyrylcholinesterase and monoamine oxidase inhibitors - Kosak_2025_Chem.Biol.Interact_15ChEPon_420_111681 |
| Author(s) : Kosak U , Knez D , Pislar A , Horvat S , Zakelj S , Igert A , Dias J , Nachon F , Brazzolotto X , Gobec S |
| Ref : Chemico-Biological Interactions , 420 :111681 , 2025 |
| Abstract : |
| PubMedSearch : Kosak_2025_Chem.Biol.Interact_15ChEPon_420_111681 |
| PubMedID: 40750068 |
| Gene_locus related to this paper: human-BCHE |
| Title : Chiral switch of a butyrylcholinesterase inhibitor for the treatment of Alzheimer's disease - Kosak_2025_Chem.Biol.Interact_15ChEPon_420_111670 |
| Author(s) : Kosak U , Knez D , Benetik SF , Sokolov PM , Pislar A , Horvat S , Stojan J , Lv B , Zhang W , Wang Y , Wang Q , Igert A , Dias J , Nachon F , Brazzolotto X , Sun H , Gobec S |
| Ref : Chemico-Biological Interactions , 420 :111670 , 2025 |
| Abstract : |
| PubMedSearch : Kosak_2025_Chem.Biol.Interact_15ChEPon_420_111670 |
| PubMedID: 40712769 |
| Gene_locus related to this paper: human-BCHE |
| Title : N-Propargylpyrrolidine-based butyrylcholinesterase and monoamine oxidase inhibitors - Kosak_2025_Chem.Biol.Interact_15ChEPon_420_111681 |
| Author(s) : Kosak U , Knez D , Pislar A , Horvat S , Zakelj S , Igert A , Dias J , Nachon F , Brazzolotto X , Gobec S |
| Ref : Chemico-Biological Interactions , 420 :111681 , 2025 |
| Abstract : |
| PubMedSearch : Kosak_2025_Chem.Biol.Interact_15ChEPon_420_111681 |
| PubMedID: 40750068 |
| Gene_locus related to this paper: human-BCHE |
| Title : Chiral switch of a butyrylcholinesterase inhibitor for the treatment of Alzheimer's disease - Kosak_2025_Chem.Biol.Interact_15ChEPon_420_111670 |
| Author(s) : Kosak U , Knez D , Benetik SF , Sokolov PM , Pislar A , Horvat S , Stojan J , Lv B , Zhang W , Wang Y , Wang Q , Igert A , Dias J , Nachon F , Brazzolotto X , Sun H , Gobec S |
| Ref : Chemico-Biological Interactions , 420 :111670 , 2025 |
| Abstract : |
| PubMedSearch : Kosak_2025_Chem.Biol.Interact_15ChEPon_420_111670 |
| PubMedID: 40712769 |
| Gene_locus related to this paper: human-BCHE |
| Title : N-Propargylpyrrolidine-based butyrylcholinesterase and monoamine oxidase inhibitors - Kosak_2025_Chem.Biol.Interact_15ChEPon_420_111681 |
| Author(s) : Kosak U , Knez D , Pislar A , Horvat S , Zakelj S , Igert A , Dias J , Nachon F , Brazzolotto X , Gobec S |
| Ref : Chemico-Biological Interactions , 420 :111681 , 2025 |
| Abstract : |
| PubMedSearch : Kosak_2025_Chem.Biol.Interact_15ChEPon_420_111681 |
| PubMedID: 40750068 |
| Gene_locus related to this paper: human-BCHE |
| Title : Chiral switch of a butyrylcholinesterase inhibitor for the treatment of Alzheimer's disease - Kosak_2025_Chem.Biol.Interact_15ChEPon_420_111670 |
| Author(s) : Kosak U , Knez D , Benetik SF , Sokolov PM , Pislar A , Horvat S , Stojan J , Lv B , Zhang W , Wang Y , Wang Q , Igert A , Dias J , Nachon F , Brazzolotto X , Sun H , Gobec S |
| Ref : Chemico-Biological Interactions , 420 :111670 , 2025 |
| Abstract : |
| PubMedSearch : Kosak_2025_Chem.Biol.Interact_15ChEPon_420_111670 |
| PubMedID: 40712769 |
| Gene_locus related to this paper: human-BCHE |
| Title : Targeting Neuroinflammation and Cognitive Decline: First-in-Class Dual Butyrylcholinesterase and p38alpha Mitogen-Activated Protein Kinase Inhibitors - Ferjancic Benetik_2025_J.Med.Chem__ |
| Author(s) : Ferjancic Benetik S , Proj M , Knez D , Kosak U , Meden A , Krajsek K , Pislar A , Horvat S , Svajger U , Tesic N , Pulkrabkova L , Soukup O , Skarka A , Andrys R , Brazzolotto X , Igert A , Nachon F , Dias J , Detka J , Gdula-Argasinska J , Wyska E , Szafarz M , Manik A , Plachtij N , Musilek K , Salat K , Obreza A , Gobec S |
| Ref : Journal of Medicinal Chemistry , : , 2025 |
| Abstract : |
| PubMedSearch : Ferjancic Benetik_2025_J.Med.Chem__ |
| PubMedID: 40779804 |
| Title : Characterization of four BCHE mutations associated with prolonged effect of suxamethonium - Brazzolotto_2021_Pharmacogenomics.J_21_165 |
| Author(s) : Brazzolotto X , Courcelle S , Sauvanet C , Guillon V , Igert A , Kononchik J , Nachon F , Ceppa F , Delacour H |
| Ref : Pharmacogenomics J , 21(2):165-173 : , 2021 |
| Abstract : |
| PubMedSearch : Brazzolotto_2021_Pharmacogenomics.J_21_165 |
| PubMedID: 33024248 |
| Title : Discovery of drug-like acetylcholinesterase inhibitors by rapid virtual screening of a 6.9 million compound database - Miles_2021_Chem.Biol.Drug.Des__ |
| Author(s) : Miles JA , Ng JH , Sreenivas BY , Courageux C , Igert A , Dias J , McGeary RP , Brazzolotto X , Ross BP |
| Ref : Chemical Biology Drug Des , : , 2021 |
| Abstract : |
| PubMedSearch : Miles_2021_Chem.Biol.Drug.Des__ |
| PubMedID: 33455074 |
| Title : Discovery of drug-like acetylcholinesterase inhibitors by rapid virtual screening of a 6.9 million compound database - Miles_2021_Chem.Biol.Drug.Des__ |
| Author(s) : Miles JA , Ng JH , Sreenivas BY , Courageux C , Igert A , Dias J , McGeary RP , Brazzolotto X , Ross BP |
| Ref : Chemical Biology Drug Des , : , 2021 |
| Abstract : |
| PubMedSearch : Miles_2021_Chem.Biol.Drug.Des__ |
| PubMedID: 33455074 |
| Title : Diisopropylfluorophosphate-induced status epilepticus drives complex glial cell phenotypes in adult male mice - Maupu_2021_Neurobiol.Dis__105276 |
| Author(s) : Maupu C , Enderlin J , Igert A , Oger M , Auvin S , Hassan-Abdi R , Soussi-Yanicostas N , Brazzolotto X , Nachon F , Bo GD , Dupuis N |
| Ref : Neurobiol Dis , :105276 , 2021 |
| Abstract : |
| PubMedSearch : Maupu_2021_Neurobiol.Dis__105276 |
| PubMedID: 33529768 |
| Title : Diisopropylfluorophosphate-induced status epilepticus drives complex glial cell phenotypes in adult male mice - Maupu_2021_Neurobiol.Dis__105276 |
| Author(s) : Maupu C , Enderlin J , Igert A , Oger M , Auvin S , Hassan-Abdi R , Soussi-Yanicostas N , Brazzolotto X , Nachon F , Bo GD , Dupuis N |
| Ref : Neurobiol Dis , :105276 , 2021 |
| Abstract : |
| PubMedSearch : Maupu_2021_Neurobiol.Dis__105276 |
| PubMedID: 33529768 |
| Title : Characterization of four BCHE mutations associated with prolonged effect of suxamethonium - Brazzolotto_2021_Pharmacogenomics.J_21_165 |
| Author(s) : Brazzolotto X , Courcelle S , Sauvanet C , Guillon V , Igert A , Kononchik J , Nachon F , Ceppa F , Delacour H |
| Ref : Pharmacogenomics J , 21(2):165-173 : , 2021 |
| Abstract : |
| PubMedSearch : Brazzolotto_2021_Pharmacogenomics.J_21_165 |
| PubMedID: 33024248 |
| Title : Discovery of drug-like acetylcholinesterase inhibitors by rapid virtual screening of a 6.9 million compound database - Miles_2021_Chem.Biol.Drug.Des__ |
| Author(s) : Miles JA , Ng JH , Sreenivas BY , Courageux C , Igert A , Dias J , McGeary RP , Brazzolotto X , Ross BP |
| Ref : Chemical Biology Drug Des , : , 2021 |
| Abstract : |
| PubMedSearch : Miles_2021_Chem.Biol.Drug.Des__ |
| PubMedID: 33455074 |
| Title : Characterization of four BCHE mutations associated with prolonged effect of suxamethonium - Brazzolotto_2021_Pharmacogenomics.J_21_165 |
| Author(s) : Brazzolotto X , Courcelle S , Sauvanet C , Guillon V , Igert A , Kononchik J , Nachon F , Ceppa F , Delacour H |
| Ref : Pharmacogenomics J , 21(2):165-173 : , 2021 |
| Abstract : |
| PubMedSearch : Brazzolotto_2021_Pharmacogenomics.J_21_165 |
| PubMedID: 33024248 |
| Title : Diisopropylfluorophosphate-induced status epilepticus drives complex glial cell phenotypes in adult male mice - Maupu_2021_Neurobiol.Dis__105276 |
| Author(s) : Maupu C , Enderlin J , Igert A , Oger M , Auvin S , Hassan-Abdi R , Soussi-Yanicostas N , Brazzolotto X , Nachon F , Bo GD , Dupuis N |
| Ref : Neurobiol Dis , :105276 , 2021 |
| Abstract : |
| PubMedSearch : Maupu_2021_Neurobiol.Dis__105276 |
| PubMedID: 33529768 |
| Title : Organophosphorus diisopropylfluorophosphate (DFP) intoxication in zebrafish larvae causes behavioral defects, neuronal hyperexcitation and neuronal death - Brenet_2020_Sci.Rep_10_19228 |
| Author(s) : Brenet A , Somkhit J , Hassan-Abdi R , Yanicostas C , Romain C , Bar O , Igert A , Saurat D , Taudon N , Dal Bo G , Nachon F , Dupuis N , Soussi-Yanicostas N |
| Ref : Sci Rep , 10 :19228 , 2020 |
| Abstract : |
| PubMedSearch : Brenet_2020_Sci.Rep_10_19228 |
| PubMedID: 33154418 |
| Gene_locus related to this paper: danre-ACHE |
| Title : Organophosphorus diisopropylfluorophosphate (DFP) intoxication in zebrafish larvae causes behavioral defects, neuronal hyperexcitation and neuronal death - Brenet_2020_Sci.Rep_10_19228 |
| Author(s) : Brenet A , Somkhit J , Hassan-Abdi R , Yanicostas C , Romain C , Bar O , Igert A , Saurat D , Taudon N , Dal Bo G , Nachon F , Dupuis N , Soussi-Yanicostas N |
| Ref : Sci Rep , 10 :19228 , 2020 |
| Abstract : |
| PubMedSearch : Brenet_2020_Sci.Rep_10_19228 |
| PubMedID: 33154418 |
| Gene_locus related to this paper: danre-ACHE |
| Title : Characterization of organophosphate-induced brain injuries in a convulsive mouse model of diisopropylfluorophosphate exposure - Enderlin_2020_Epilepsia__ |
| Author(s) : Enderlin J , Igert A , Auvin S , Nachon F , Dal Bo G , Dupuis N |
| Ref : Epilepsia , : , 2020 |
| Abstract : |
| PubMedSearch : Enderlin_2020_Epilepsia__ |
| PubMedID: 32359085 |
| Title : Organophosphorus diisopropylfluorophosphate (DFP) intoxication in zebrafish larvae causes behavioral defects, neuronal hyperexcitation and neuronal death - Brenet_2020_Sci.Rep_10_19228 |
| Author(s) : Brenet A , Somkhit J , Hassan-Abdi R , Yanicostas C , Romain C , Bar O , Igert A , Saurat D , Taudon N , Dal Bo G , Nachon F , Dupuis N , Soussi-Yanicostas N |
| Ref : Sci Rep , 10 :19228 , 2020 |
| Abstract : |
| PubMedSearch : Brenet_2020_Sci.Rep_10_19228 |
| PubMedID: 33154418 |
| Gene_locus related to this paper: danre-ACHE |
| Title : Rapid discovery of a selective butyrylcholinesterase inhibitor using structure-based virtual screening - Miles_2020_Bioorg.Med.Chem.Lett__127609 |
| Author(s) : Miles JA , Kapure JS , Singh Deora G , Courageux C , Igert A , Dias J , McGeary RP , Brazzolotto X , Ross BP |
| Ref : Bioorganic & Medicinal Chemistry Lett , :127609 , 2020 |
| Abstract : |
| PubMedSearch : Miles_2020_Bioorg.Med.Chem.Lett__127609 |
| PubMedID: 33039562 |
| Title : Characterization of organophosphate-induced brain injuries in a convulsive mouse model of diisopropylfluorophosphate exposure - Enderlin_2020_Epilepsia__ |
| Author(s) : Enderlin J , Igert A , Auvin S , Nachon F , Dal Bo G , Dupuis N |
| Ref : Epilepsia , : , 2020 |
| Abstract : |
| PubMedSearch : Enderlin_2020_Epilepsia__ |
| PubMedID: 32359085 |
| Title : Characterization of organophosphate-induced brain injuries in a convulsive mouse model of diisopropylfluorophosphate exposure - Enderlin_2020_Epilepsia__ |
| Author(s) : Enderlin J , Igert A , Auvin S , Nachon F , Dal Bo G , Dupuis N |
| Ref : Epilepsia , : , 2020 |
| Abstract : |
| PubMedSearch : Enderlin_2020_Epilepsia__ |
| PubMedID: 32359085 |
| Title : Rapid discovery of a selective butyrylcholinesterase inhibitor using structure-based virtual screening - Miles_2020_Bioorg.Med.Chem.Lett__127609 |
| Author(s) : Miles JA , Kapure JS , Singh Deora G , Courageux C , Igert A , Dias J , McGeary RP , Brazzolotto X , Ross BP |
| Ref : Bioorganic & Medicinal Chemistry Lett , :127609 , 2020 |
| Abstract : |
| PubMedSearch : Miles_2020_Bioorg.Med.Chem.Lett__127609 |
| PubMedID: 33039562 |
| Title : Rapid discovery of a selective butyrylcholinesterase inhibitor using structure-based virtual screening - Miles_2020_Bioorg.Med.Chem.Lett__127609 |
| Author(s) : Miles JA , Kapure JS , Singh Deora G , Courageux C , Igert A , Dias J , McGeary RP , Brazzolotto X , Ross BP |
| Ref : Bioorganic & Medicinal Chemistry Lett , :127609 , 2020 |
| Abstract : |
| PubMedSearch : Miles_2020_Bioorg.Med.Chem.Lett__127609 |
| PubMedID: 33039562 |
| Title : Bacterial Expression of Human Butyrylcholinesterase as a Tool for Nerve Agent Bioscavengers Development - Brazzolotto_2017_Molecules_22_ |
| Author(s) : Brazzolotto X , Igert A , Guillon V , Santoni G , Nachon F |
| Ref : Molecules , 22 : , 2017 |
| Abstract : |
| PubMedSearch : Brazzolotto_2017_Molecules_22_ |
| PubMedID: 29077024 |
| Gene_locus related to this paper: human-BCHE |
| Title : Bacterial Expression of Human Butyrylcholinesterase as a Tool for Nerve Agent Bioscavengers Development - Brazzolotto_2017_Molecules_22_ |
| Author(s) : Brazzolotto X , Igert A , Guillon V , Santoni G , Nachon F |
| Ref : Molecules , 22 : , 2017 |
| Abstract : |
| PubMedSearch : Brazzolotto_2017_Molecules_22_ |
| PubMedID: 29077024 |
| Gene_locus related to this paper: human-BCHE |
| Title : Bacterial Expression of Human Butyrylcholinesterase as a Tool for Nerve Agent Bioscavengers Development - Brazzolotto_2017_Molecules_22_ |
| Author(s) : Brazzolotto X , Igert A , Guillon V , Santoni G , Nachon F |
| Ref : Molecules , 22 : , 2017 |
| Abstract : |
| PubMedSearch : Brazzolotto_2017_Molecules_22_ |
| PubMedID: 29077024 |
| Gene_locus related to this paper: human-BCHE |