| Title : Discovery of Highly Selective and Nanomolar Carbamate-Based Butyrylcholinesterase Inhibitors by Rational Investigation into Their Inhibition Mode - Sawatzky_2016_J.Med.Chem_59_2067 |
| Author(s) : Sawatzky E , Wehle S , Kling B , Wendrich J , Bringmann G , Sotriffer CA , Heilmann J , Decker M |
| Ref : Journal of Medicinal Chemistry , 59 :2067 , 2016 |
| Abstract : |
| PubMedSearch : Sawatzky_2016_J.Med.Chem_59_2067 |
| PubMedID: 26886849 |
| Title : Amine substitution of quinazolinones leads to selective nanomolar AChE inhibitors with 'inverted' binding mode - Darras_2014_Bioorg.Med.Chem_22_4867 |
| Author(s) : Darras FH , Wehle S , Huang G , Sotriffer CA , Decker M |
| Ref : Bioorganic & Medicinal Chemistry , 22 :4867 , 2014 |
| Abstract : |
| PubMedSearch : Darras_2014_Bioorg.Med.Chem_22_4867 |
| PubMedID: 25047936 |
| Title : Synthesis, Biological Evaluation, and Computational Studies of Tri- and Tetracyclic Nitrogen-Bridgehead Compounds as Potent Dual-Acting AChE Inhibitors and hH3 Receptor Antagonists - Darras_2014_ACS.Chem.Neurosci_5_225 |
| Author(s) : Darras FH , Pockes S , Huang G , Wehle S , Strasser A , Wittmann HJ , Nimczick M , Sotriffer CA , Decker M |
| Ref : ACS Chem Neurosci , 5 :225 , 2014 |
| Abstract : |
| PubMedSearch : Darras_2014_ACS.Chem.Neurosci_5_225 |
| PubMedID: 24422467 |
| Title : Acetylcholinesterase inhibitors with photoswitchable inhibition of beta-amyloid aggregation - Chen_2014_ACS.Chem.Neurosci_5_377 |
| Author(s) : Chen X , Wehle S , Kuzmanovic N , Merget B , Holzgrabe U , Konig B , Sotriffer CA , Decker M |
| Ref : ACS Chem Neurosci , 5 :377 , 2014 |
| Abstract : |
| PubMedSearch : Chen_2014_ACS.Chem.Neurosci_5_377 |
| PubMedID: 24628027 |
| Title : 1,4-Substituted 4-(1H)-pyridylene-hydrazone-type inhibitors of AChE, BCHE, and amyloid-beta aggregation crossing the blood-brain barrier - Prinz_2013_Eur.J.Pharm.Sci_49_603 |
| Author(s) : Prinz M , Parlar S , Bayraktar G , Alptuzun V , Erciyas E , Fallarero A , Karlsson D , Vuorela P , Burek M , Forster C , Turunc E , Armagan G , Yalcin A , Schiller C , Leuner K , Krug M , Sotriffer CA , Holzgrabe U |
| Ref : Eur J Pharm Sci , 49 :603 , 2013 |
| Abstract : |
| PubMedSearch : Prinz_2013_Eur.J.Pharm.Sci_49_603 |
| PubMedID: 23643737 |
| Title : Structure-based search for new inhibitors of cholinesterases - Bajda_2013_Int.J.Mol.Sci_14_5608 |
| Author(s) : Bajda M , Wieckowska A , Hebda M , Guzior N , Sotriffer CA , Malawska B |
| Ref : Int J Mol Sci , 14 :5608 , 2013 |
| Abstract : |
| PubMedSearch : Bajda_2013_Int.J.Mol.Sci_14_5608 |
| PubMedID: 23478436 |