Wieckowska A

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Title : Design, Synthesis, and Biological Evaluation of 1-Benzylamino-2-hydroxyalkyl Derivatives as New Potential Disease-Modifying Multifunctional Anti-Alzheimer's Agents - Panek_2018_ACS.Chem.Neurosci_9_1074
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Title : Design, synthesis and biological evaluation of new phthalimide and saccharin derivatives with alicyclic amines targeting cholinesterases, beta-secretase and amyloid beta aggregation - Panek_2016_Eur.J.Med.Chem_125_676
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Title : Novel multi-target-directed ligands for Alzheimer's disease: Combining cholinesterase inhibitors and 5-HT6 receptor antagonists. Design, synthesis and biological evaluation - Wieckowska_2016_Eur.J.Med.Chem_124_63
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Title : Cholinesterase inhibitory activity of chlorophenoxy derivatives-Histamine H3 receptor ligands - Lazewska_2016_Bioorg.Med.Chem.Lett_26_4140
Author(s) : Lazewska D , Jonczyk J , Bajda M , Szalaj N , Wieckowska A , Panek D , Moore C , Kuder K , Malawska B , Kiec-Kononowicz K
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Title : Synthesis, Molecular Modelling and Biological Evaluation of Novel Heterodimeric, Multiple Ligands Targeting Cholinesterases and Amyloid Beta - Hebda_2016_Molecules_21_
Author(s) : Hebda M , Bajda M , Wieckowska A , Szalaj N , Pasieka A , Panek D , Godyn J , Wichur T , Knez D , Gobec S , Malawska B
Ref : Molecules , 21 : , 2016
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Title : Development of an in-vivo active reversible butyrylcholinesterase inhibitor - Kosak_2016_Sci.Rep_6_39495
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Gene_locus related to this paper: human-BCHE

Title : SEARCH FOR POTENTIAL CHOLINESTERASE INHIBITORS FROM THE ZINC DATABASE BY VIRTUAL SCREENING METHOD - Bajda_2015_Acta.Pol.Pharm_72_737
Author(s) : Bajda M , Panek D , Hebda M , Wieckowska A , Guzior N , Malawska B
Ref : Acta Pol Pharm , 72 :737 , 2015
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Title : Recent development of multifunctional agents as potential drug candidates for the treatment of Alzheimer's disease - Guzior_2015_Curr.Med.Chem_22_373
Author(s) : Guzior N , Wieckowska A , Panek D , Malawska B
Ref : Curr Med Chem , 22 :373 , 2015
PubMedID: 25386820

Title : Synthesis of new N-benzylpiperidine derivatives as cholinesterase inhibitors with beta-amyloid anti-aggregation properties and beneficial effects on memory in vivo - Wieckowska_2015_Bioorg.Med.Chem_23_2445
Author(s) : Wieckowska A , Wieckowski K , Bajda M , Brus B , Salat K , Czerwinska P , Gobec S , Filipek B , Malawska B
Ref : Bioorganic & Medicinal Chemistry , 23 :2445 , 2015
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Title : Structure-based search for new inhibitors of cholinesterases - Bajda_2013_Int.J.Mol.Sci_14_5608
Author(s) : Bajda M , Wieckowska A , Hebda M , Guzior N , Sotriffer CA , Malawska B
Ref : Int J Mol Sci , 14 :5608 , 2013
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Title : Novel alkyl- and arylcarbamate derivatives with N-benzylpiperidine and N-benzylpiperazine moieties as cholinesterases inhibitors - Wieckowska_2010_Eur.J.Med.Chem_45_5602
Author(s) : Wieckowska A , Bajda M , Guzior N , Malawska B
Ref : Eur Journal of Medicinal Chemistry , 45 :5602 , 2010
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Title : Electrophoretically mediated microanalysis technique as a tool for the rapid screening of novel acetylcholinesterase inhibitors - Bajda_2009_Acta.Pol.Pharm_66_357
Author(s) : Bajda M , Wieckowska A , Malawska B
Ref : Acta Pol Pharm , 66 :357 , 2009
PubMedID: 19702166