Full name : Spilling Christopher D
First name : Christopher D
Mail : Department of Chemistry and Biochemistry and the Center for Nanoscience, University of Missouri-St. Louis, One University Boulevard, St. Louis, MO 63121
Zip Code :
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Country : USA
Email : cspill@umsl.edu
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| Title : Direct capture, inhibition and crystal structure of HsaD (Rv3569c) from M. tuberculosis - Barelier_2022_FEBS.J__ |
| Author(s) : Barelier S , Avellan R , Gnawali GR , Fourquet P , Roig-Zamboni V , Poncin I , Point V , Bourne Y , Audebert S , Camoin L , Spilling CD , Canaan S , Cavalier JF , Sulzenbacher G |
| Ref : Febs J , : , 2022 |
| Abstract : |
| PubMedSearch : Barelier_2022_FEBS.J__ |
| PubMedID: 36197115 |
| Gene_locus related to this paper: myctu-Rv3569c |
| Title : Lipolytic enzymes inhibitors: A new way for antibacterial drugs discovery - Cavalier_2021_Eur.J.Med.Chem_209_112908 |
| Author(s) : Cavalier JF , Spilling CD , Durand T , Camoin L , Canaan S |
| Ref : Eur Journal of Medicinal Chemistry , 209 :112908 , 2021 |
| Abstract : |
| PubMedSearch : Cavalier_2021_Eur.J.Med.Chem_209_112908 |
| PubMedID: 33071055 |
| Title : Cyclophostin and Cyclipostins analogues, new promising molecules to treat mycobacterial-related diseases - Nguyen_2018_Int.J.Antimicrob.Agents_51_651 |
| Author(s) : Nguyen PC , Madani A , Santucci P , Martin BP , Paudel RR , Delattre S , Herrmann JL , Spilling CD , Kremer L , Canaan S , Cavalier JF |
| Ref : Int J Antimicrob Agents , 51 :651 , 2018 |
| Abstract : |
| PubMedSearch : Nguyen_2018_Int.J.Antimicrob.Agents_51_651 |
| PubMedID: 29241819 |
| Title : Biochemical and Structural Characterization of TesA, a Major Thioesterase Required for Outer-Envelope Lipid Biosynthesis in Mycobacterium tuberculosis - Nguyen_2018_J.Mol.Biol_430_5120 |
| Author(s) : Nguyen PC , Nguyen VS , Martin BP , Fourquet P , Camoin L , Spilling CD , Cavalier JF , Cambillau C , Canaan S |
| Ref : Journal of Molecular Biology , 430 :5120 , 2018 |
| Abstract : |
| PubMedSearch : Nguyen_2018_J.Mol.Biol_430_5120 |
| PubMedID: 30292819 |
| Gene_locus related to this paper: myctu-yt28 |
| Title : Cyclipostins and cyclophostin analogs inhibit the antigen 85C from Mycobacterium tuberculosis both in vitro and in vivo - Viljoen_2018_J.Biol.Chem_293_2755 |
| Author(s) : Viljoen A , Richard M , Nguyen PC , Fourquet P , Camoin L , Paudal RR , Gnawali GR , Spilling CD , Cavalier JF , Canaan S , Blaise M , Kremer L |
| Ref : Journal of Biological Chemistry , 293 :2755 , 2018 |
| Abstract : |
| PubMedSearch : Viljoen_2018_J.Biol.Chem_293_2755 |
| PubMedID: 29301937 |
| Gene_locus related to this paper: myctu-a85c |
| Title : Cyclipostins and Cyclophostin analogs as promising compounds in the fight against tuberculosis - Nguyen_2017_Sci.Rep_7_11751 |
| Author(s) : Nguyen PC , Delorme V , Benarouche A , Martin BP , Paudel R , Gnawali GR , Madani A , Puppo R , Landry V , Kremer L , Brodin P , Spilling CD , Cavalier JF , Canaan S |
| Ref : Sci Rep , 7 :11751 , 2017 |
| Abstract : |
| PubMedSearch : Nguyen_2017_Sci.Rep_7_11751 |
| PubMedID: 28924204 |
| Gene_locus related to this paper: mycle-ML2603 , myctu-a85a , myctu-a85c , myctu-Rv1399c , myctu-Rv2970c , myctu-Rv3569c , myctu-yt28 |
| Title : Synthesis and comparison of the biological activity of monocyclic phosphonate, difluorophosphonate and phosphate analogs of the natural AChE inhibitor cyclophostin - Martin_2015_Bioorg.Med.Chem_23_7529 |
| Author(s) : Martin BP , Vasilieva E , Dupureur CM , Spilling CD |
| Ref : Bioorganic & Medicinal Chemistry , 23 :7529 , 2015 |
| Abstract : |
| PubMedSearch : Martin_2015_Bioorg.Med.Chem_23_7529 |
| PubMedID: 26585276 |
| Title : Rat hormone sensitive lipase inhibition by cyclipostins and their analogs - Vasilieva_2015_Bioorg.Med.Chem_23_944 |
| Author(s) : Vasilieva E , Dutta S , Malla RK , Martin BP , Spilling CD , Dupureur CM |
| Ref : Bioorganic & Medicinal Chemistry , 23 :944 , 2015 |
| Abstract : |
| PubMedSearch : Vasilieva_2015_Bioorg.Med.Chem_23_944 |
| PubMedID: 25678014 |
| Gene_locus related to this paper: ratno-hslip |
| Title : Enantioselective inhibition of microbial lipolytic enzymes by nonracemic monocyclic enolphosphonate analogues of cyclophostin - Point_2013_J.Med.Chem_56_4393 |
| Author(s) : Point V , Malla RK , Carriere F , Canaan S , Spilling CD , Cavalier JF |
| Ref : Journal of Medicinal Chemistry , 56 :4393 , 2013 |
| Abstract : |
| PubMedSearch : Point_2013_J.Med.Chem_56_4393 |
| PubMedID: 23651298 |
| Title : Synthesis and kinetic evaluation of cyclophostin and cyclipostins phosphonate analogs as selective and potent inhibitors of microbial lipases - Point_2012_J.Med.Chem_55_10204 |
| Author(s) : Point V , Malla RK , Diomande S , Martin BP , Delorme V , Carriere F , Canaan S , Rath NP , Spilling CD , Cavalier JF |
| Ref : Journal of Medicinal Chemistry , 55 :10204 , 2012 |
| Abstract : |
| PubMedSearch : Point_2012_J.Med.Chem_55_10204 |
| PubMedID: 23095026 |
| Title : The first total synthesis of (+\/-)-cyclophostin and (+\/-)-cyclipostin P: inhibitors of the serine hydrolases acetyl cholinesterase and hormone sensitive lipase - Malla_2011_Org.Lett_13_3094 |
| Author(s) : Malla RK , Bandyopadhyay S , Spilling CD , Dutta S , Dupureur CM |
| Ref : Org Lett , 13 :3094 , 2011 |
| Abstract : |
| PubMedSearch : Malla_2011_Org.Lett_13_3094 |
| PubMedID: 21591624 |
| Title : Synthesis and kinetic analysis of some phosphonate analogs of cyclophostin as inhibitors of human acetylcholinesterase - Dutta_2010_Bioorg.Med.Chem_18_2265 |
| Author(s) : Dutta S , Malla RK , Bandyopadhyay S , Spilling CD , Dupureur CM |
| Ref : Bioorganic & Medicinal Chemistry , 18 :2265 , 2010 |
| Abstract : |
| PubMedSearch : Dutta_2010_Bioorg.Med.Chem_18_2265 |
| PubMedID: 20189400 |
| Title : Synthesis and biological evaluation of a phosphonate analog of the natural acetyl cholinesterase inhibitor cyclophostin - Bandyopadhyay_2008_J.Org.Chem_73_8386 |
| Author(s) : Bandyopadhyay S , Dutta S , Spilling CD , Dupureur CM , Rath NP |
| Ref : J Org Chem , 73 :8386 , 2008 |
| Abstract : |
| PubMedSearch : Bandyopadhyay_2008_J.Org.Chem_73_8386 |
| PubMedID: 18821801 |