Title : Direct capture, inhibition and crystal structure of HsaD (Rv3569c) from M. tuberculosis - Barelier_2022_FEBS.J__ |
Author(s) : Barelier S , Avellan R , Gnawali GR , Fourquet P , Roig-Zamboni V , Poncin I , Point V , Bourne Y , Audebert S , Camoin L , Spilling CD , Canaan S , Cavalier JF , Sulzenbacher G |
Ref : Febs J , : , 2022 |
Abstract : |
PubMedSearch : Barelier_2022_FEBS.J__ |
PubMedID: 36197115 |
Gene_locus related to this paper: myctu-Rv3569c |
Title : Identification of cell wall synthesis inhibitors active against Mycobacterium tuberculosis by competitive activity-based protein profiling - Li_2022_Cell.Chem.Biol_29_883 |
Author(s) : Li M , Patel HV , Cognetta AB, 3rd , Smith TC, 2nd , Mallick I , Cavalier JF , Previti ML , Canaan S , Aldridge BB , Cravatt BF , Seeliger JC |
Ref : Cell Chemical Biology , 29 :883 , 2022 |
Abstract : |
PubMedSearch : Li_2022_Cell.Chem.Biol_29_883 |
PubMedID: 34599873 |
Title : Lipolytic enzymes inhibitors: A new way for antibacterial drugs discovery - Cavalier_2021_Eur.J.Med.Chem_209_112908 |
Author(s) : Cavalier JF , Spilling CD , Durand T , Camoin L , Canaan S |
Ref : Eur Journal of Medicinal Chemistry , 209 :112908 , 2021 |
Abstract : |
PubMedSearch : Cavalier_2021_Eur.J.Med.Chem_209_112908 |
PubMedID: 33071055 |
Title : Dissecting the antibacterial activity of oxadiazolone-core derivatives against Mycobacterium abscessus - Madani_2020_PLoS.One_15_e0238178 |
Author(s) : Madani A , Mallick I , Guy A , Crauste C , Durand T , Fourquet P , Audebert S , Camoin L , Canaan S , Cavalier JF |
Ref : PLoS ONE , 15 :e0238178 , 2020 |
Abstract : |
PubMedSearch : Madani_2020_PLoS.One_15_e0238178 |
PubMedID: 32946441 |
Title : Dissecting the membrane lipid binding properties and lipase activity of Mycobacterium tuberculosis LipY domains - Santucci_2019_Febs.j_286_3164 |
Author(s) : Santucci P , Smichi N , Diomande S , Poncin I , Point V , Gaussier H , Cavalier JF , Kremer L , Canaan S |
Ref : Febs J , 286 :3164 , 2019 |
Abstract : |
PubMedSearch : Santucci_2019_Febs.j_286_3164 |
PubMedID: 31034693 |
Gene_locus related to this paper: myctu-Rv3097c |
Title : Cyclophostin and Cyclipostins analogues, new promising molecules to treat mycobacterial-related diseases - Nguyen_2018_Int.J.Antimicrob.Agents_51_651 |
Author(s) : Nguyen PC , Madani A , Santucci P , Martin BP , Paudel RR , Delattre S , Herrmann JL , Spilling CD , Kremer L , Canaan S , Cavalier JF |
Ref : Int J Antimicrob Agents , 51 :651 , 2018 |
Abstract : |
PubMedSearch : Nguyen_2018_Int.J.Antimicrob.Agents_51_651 |
PubMedID: 29241819 |
Title : Cyclipostins and cyclophostin analogs inhibit the antigen 85C from Mycobacterium tuberculosis both in vitro and in vivo - Viljoen_2018_J.Biol.Chem_293_2755 |
Author(s) : Viljoen A , Richard M , Nguyen PC , Fourquet P , Camoin L , Paudal RR , Gnawali GR , Spilling CD , Cavalier JF , Canaan S , Blaise M , Kremer L |
Ref : Journal of Biological Chemistry , 293 :2755 , 2018 |
Abstract : |
PubMedSearch : Viljoen_2018_J.Biol.Chem_293_2755 |
PubMedID: 29301937 |
Gene_locus related to this paper: myctu-a85c |
Title : Oxadiazolone derivatives, new promising multi-target inhibitors against M. tuberculosis - Nguyen_2018_Bioorg.Chem_81_414 |
Author(s) : Nguyen PC , Delorme V , Benarouche A , Guy A , Landry V , Audebert S , Pophillat M , Camoin L , Crauste C , Galano JM , Durand T , Brodin P , Canaan S , Cavalier JF |
Ref : Bioorg Chem , 81 :414 , 2018 |
Abstract : |
PubMedSearch : Nguyen_2018_Bioorg.Chem_81_414 |
PubMedID: 30212765 |
Title : Biochemical and Structural Characterization of TesA, a Major Thioesterase Required for Outer-Envelope Lipid Biosynthesis in Mycobacterium tuberculosis - Nguyen_2018_J.Mol.Biol_430_5120 |
Author(s) : Nguyen PC , Nguyen VS , Martin BP , Fourquet P , Camoin L , Spilling CD , Cavalier JF , Cambillau C , Canaan S |
Ref : Journal of Molecular Biology , 430 :5120 , 2018 |
Abstract : |
PubMedSearch : Nguyen_2018_J.Mol.Biol_430_5120 |
PubMedID: 30292819 |
Gene_locus related to this paper: myctu-yt28 |
Title : Cyclipostins and Cyclophostin analogs as promising compounds in the fight against tuberculosis - Nguyen_2017_Sci.Rep_7_11751 |
Author(s) : Nguyen PC , Delorme V , Benarouche A , Martin BP , Paudel R , Gnawali GR , Madani A , Puppo R , Landry V , Kremer L , Brodin P , Spilling CD , Cavalier JF , Canaan S |
Ref : Sci Rep , 7 :11751 , 2017 |
Abstract : |
PubMedSearch : Nguyen_2017_Sci.Rep_7_11751 |
PubMedID: 28924204 |
Gene_locus related to this paper: mycle-ML2603 , myctu-a85a , myctu-a85c , myctu-Rv1399c , myctu-Rv2970c , myctu-Rv3569c , myctu-yt28 |
Title : Studying Gastric Lipase Adsorption Onto Phospholipid Monolayers by Surface Tensiometry, Ellipsometry, and Atomic Force Microscopy - Benarouche_2017_Methods.Enzymol_583_255 |
Author(s) : Benarouche A , Sams L , Bourlieu C , Vie V , Point V , Cavalier JF , Carriere F |
Ref : Methods Enzymol , 583 :255 , 2017 |
Abstract : |
PubMedSearch : Benarouche_2017_Methods.Enzymol_583_255 |
PubMedID: 28063494 |
Title : Efficient synthesis of novel dialkyl-3-cyanopropylphosphate derivatives and evaluation of their anticholinesterase activity - Aouani_2017_Bioorg.Chem_72_301 |
Author(s) : Aouani I , Sellami B , Lahbib K , Cavalier JF , Touil S |
Ref : Bioorg Chem , 72 :301 , 2017 |
Abstract : |
PubMedSearch : Aouani_2017_Bioorg.Chem_72_301 |
PubMedID: 28500956 |
Title : Slowing down fat digestion and absorption by an oxadiazolone inhibitor targeting selectively gastric lipolysis - Point_2016_Eur.J.Med.Chem_123_834 |
Author(s) : Point V , Benarouche A , Zarrillo J , Guy A , Magnez R , Fonseca L , Raux B , Leclaire J , Buono G , Fotiadu F , Durand T , Carriere F , Vaysse C , Couedelo L , Cavalier JF |
Ref : Eur Journal of Medicinal Chemistry , 123 :834 , 2016 |
Abstract : |
PubMedSearch : Point_2016_Eur.J.Med.Chem_123_834 |
PubMedID: 27543878 |
Gene_locus related to this paper: canfa-1lipg , human-LIPF |
Title : Effect of preduodenal lipase inhibition in suckling rats on dietary octanoic acid (C8:0) gastric absorption and plasma octanoylated ghrelin concentration - Lemarie_2016_Biochim.Biophys.Acta_1861_1111 |
Author(s) : Lemarie F , Cavalier JF , Garcia C , Boissel F , Point V , Catheline D , Legrand P , Carriere F , Rioux V |
Ref : Biochimica & Biophysica Acta , 1861 :1111 , 2016 |
Abstract : |
PubMedSearch : Lemarie_2016_Biochim.Biophys.Acta_1861_1111 |
PubMedID: 27317984 |
Title : New lipase assay using Pomegranate oil coating in microtiter plates - Ulker_2016_Biochimie_120_110 |
Author(s) : Ulker S , Placidi C , Point V , Gadenne B , Serveau-Avesque C , Canaan S , Carriere F , Cavalier JF |
Ref : Biochimie , 120 :110 , 2016 |
Abstract : |
PubMedSearch : Ulker_2016_Biochimie_120_110 |
PubMedID: 26343557 |
Title : Adsorption of gastric lipase onto multicomponent model lipid monolayers with phase separation - Bourlieu_2016_Colloids.Surf.B.Biointerfaces_143_97 |
Author(s) : Bourlieu C , Paboeuf G , Chever S , Pezennec S , Cavalier JF , Guyomarc'h F , Deglaire A , Bouhallab S , Dupont D , Carriere F , Vie V |
Ref : Colloids Surf B Biointerfaces , 143 :97 , 2016 |
Abstract : |
PubMedSearch : Bourlieu_2016_Colloids.Surf.B.Biointerfaces_143_97 |
PubMedID: 27011347 |
Title : Biochemical characterization of Yarrowia lipolytica LIP8, a secreted lipase with a cleavable C-terminal region - Kamoun_2015_Biochim.Biophys.Acta_1851_129 |
Author(s) : Kamoun J , Schue M , Messaoud W , Baignol J , Point V , Mateos-Diaz E , Mansuelle P , Gargouri Y , Parsiegla G , Cavalier JF , Carriere F , Aloulou A |
Ref : Biochimica & Biophysica Acta , 1851 :129 , 2015 |
Abstract : |
PubMedSearch : Kamoun_2015_Biochim.Biophys.Acta_1851_129 |
PubMedID: 25449652 |
Gene_locus related to this paper: yarli-LIP8 |
Title : An interfacial and comparative in vitro study of gastrointestinal lipases and Yarrowia lipolytica LIP2 lipase, a candidate for enzyme replacement therapy - Benarouche_2014_Biochimie_102_145 |
Author(s) : Benarouche A , Point V , Carriere F , Cavalier JF |
Ref : Biochimie , 102 :145 , 2014 |
Abstract : |
PubMedSearch : Benarouche_2014_Biochimie_102_145 |
PubMedID: 24650780 |
Title : Using the reversible inhibition of gastric lipase by Orlistat for investigating simultaneously lipase adsorption and substrate hydrolysis at the lipid-water interface - Benarouche_2014_Biochimie_101_221 |
Author(s) : Benarouche A , Point V , Carriere F , Cavalier JF |
Ref : Biochimie , 101 :221 , 2014 |
Abstract : |
PubMedSearch : Benarouche_2014_Biochimie_101_221 |
PubMedID: 24508576 |
Title : Supported inhibitor for fishing lipases in complex biological media and mass spectrometry identification - Delorme_2014_Biochimie_107 Pt A_124 |
Author(s) : Delorme V , Raux B , Puppo R , Leclaire J , Cavalier JF , Marc S , Kamarajugadda PK , Buono G , Fotiadu F , Canaan S , Carriere F |
Ref : Biochimie , 107 Pt A :124 , 2014 |
Abstract : |
PubMedSearch : Delorme_2014_Biochimie_107 Pt A_124 |
PubMedID: 25064360 |
Title : New insights into the pH-dependent interfacial adsorption of dog gastric lipase using the monolayer technique - Benarouche_2013_Colloids.Surf.B.Biointerfaces_111_306 |
Author(s) : Benarouche A , Point V , Parsiegla G , Carriere F , Cavalier JF |
Ref : Colloids Surf B Biointerfaces , 111 :306 , 2013 |
Abstract : |
PubMedSearch : Benarouche_2013_Colloids.Surf.B.Biointerfaces_111_306 |
PubMedID: 23838197 |
Title : Effects of the propeptide of group X secreted phospholipase A(2) on substrate specificity and interfacial activity on phospholipid monolayers - Point_2013_Biochimie_95_51 |
Author(s) : Point V , Benarouche A , Jemel I , Parsiegla G , Lambeau G , Carriere F , Cavalier JF |
Ref : Biochimie , 95 :51 , 2013 |
Abstract : |
PubMedSearch : Point_2013_Biochimie_95_51 |
PubMedID: 22967966 |
Title : Biochemical and structural characterization of non-glycosylated Yarrowia lipolytica LIP2 lipase - Aloulou_2013_Eur.J.Lipid.Sci.Tech_115_429 |
Author(s) : Aloulou A , Benarouche A , Puccinelli D , Spinelli S , Cavalier JF , Cambillau C , Carriere F |
Ref : Eur.J.Lipid.Sci.Tech , 115 :429 , 2013 |
Abstract : |
PubMedSearch : Aloulou_2013_Eur.J.Lipid.Sci.Tech_115_429 |
PubMedID: |
Gene_locus related to this paper: yarli-lip2 |
Title : Enantioselective inhibition of microbial lipolytic enzymes by nonracemic monocyclic enolphosphonate analogues of cyclophostin - Point_2013_J.Med.Chem_56_4393 |
Author(s) : Point V , Malla RK , Carriere F , Canaan S , Spilling CD , Cavalier JF |
Ref : Journal of Medicinal Chemistry , 56 :4393 , 2013 |
Abstract : |
PubMedSearch : Point_2013_J.Med.Chem_56_4393 |
PubMedID: 23651298 |
Title : Analysis of the discriminative inhibition of mammalian digestive lipases by 3-phenyl substituted 1,3,4-oxadiazol-2(3H)-ones. - Point_2012_Eur.J.Med.Chem_58_452 |
Author(s) : Point V , Pavan Kumar KV , Marc S , Delorme V , Parsiegla G , Amara S , Carriere F , Buono G , Fotiadu F , Canaan S , Leclaire J , Cavalier JF |
Ref : Eur Journal of Medicinal Chemistry , 58 :452 , 2012 |
Abstract : |
PubMedSearch : Point_2012_Eur.J.Med.Chem_58_452 |
PubMedID: 23153815 |
Gene_locus related to this paper: canfa-1lipg , cavpo-2plrp , human-CEL , human-PNLIP , human-PNLIPRP2 , pig-1plip |
Title : MmPPOX inhibits Mycobacterium tuberculosis lipolytic enzymes belonging to the hormone-sensitive lipase family and alters mycobacterial growth - Delorme_2012_PLoS.One_7_e46493 |
Author(s) : Delorme V , Diomande SV , Dedieu L , Cavalier JF , Carriere F , Kremer L , Leclaire J , Fotiadu F , Canaan S |
Ref : PLoS ONE , 7 :e46493 , 2012 |
Abstract : |
PubMedSearch : Delorme_2012_PLoS.One_7_e46493 |
PubMedID: 23029536 |
Gene_locus related to this paper: myctu-Rv2970c |
Title : Synthesis and kinetic evaluation of cyclophostin and cyclipostins phosphonate analogs as selective and potent inhibitors of microbial lipases - Point_2012_J.Med.Chem_55_10204 |
Author(s) : Point V , Malla RK , Diomande S , Martin BP , Delorme V , Carriere F , Canaan S , Rath NP , Spilling CD , Cavalier JF |
Ref : Journal of Medicinal Chemistry , 55 :10204 , 2012 |
Abstract : |
PubMedSearch : Point_2012_J.Med.Chem_55_10204 |
PubMedID: 23095026 |
Title : Effects of surfactants on lipase structure, activity, and inhibition - Delorme_2011_Pharm.Res_28_1831 |
Author(s) : Delorme V , Dhouib R , Canaan S , Fotiadu F , Carriere F , Cavalier JF |
Ref : Pharm Res , 28 :1831 , 2011 |
Abstract : |
PubMedSearch : Delorme_2011_Pharm.Res_28_1831 |
PubMedID: 21234659 |
Title : Validation of lipolysis product extraction from aqueous\/biological samples, separation and quantification by thin-layer chromatography with flame ionization detection analysis using O-cholesteryl ethylene glycol as a new internal standard - Cavalier_2009_J.Chromatogr.A_1216_6543 |
Author(s) : Cavalier JF , Lafont D , Boullanger P , Houisse D , Giallo J , Ballester JM , Carriere F |
Ref : Journal of Chromatography A , 1216 :6543 , 2009 |
Abstract : |
PubMedSearch : Cavalier_2009_J.Chromatogr.A_1216_6543 |
PubMedID: 19671473 |
Title : Discrimination between closed and open forms of lipases using electrophoretic techniques - Miled_2005_Anal.Biochem_338_171 |
Author(s) : Miled N , Riviere M , Cavalier JF , Buono G , Berti L , Verger R |
Ref : Analytical Biochemistry , 338 :171 , 2005 |
Abstract : |
PubMedSearch : Miled_2005_Anal.Biochem_338_171 |
PubMedID: 15745736 |
Title : Covalent inhibition of digestive lipases by chiral phosphonates - Cavalier_2000_Acc.Chem.Res_33_579 |
Author(s) : Cavalier JF , Buono G , Verger R |
Ref : Acc Chem Res , 33 :579 , 2000 |
Abstract : |
PubMedSearch : Cavalier_2000_Acc.Chem.Res_33_579 |
PubMedID: 10995195 |
Title : Inhibition of human gastric and pancreatic lipases by chiral alkylphosphonates. A kinetic study with 1,2-didecanoyl-sn-glycerol monolayer - Cavalier_1999_Chem.Phys.Lipids_100_3 |
Author(s) : Cavalier JF , Ransac S , Verger R , Buono G |
Ref : Chemistry & Physic of Lipids , 100 :3 , 1999 |
Abstract : |
PubMedSearch : Cavalier_1999_Chem.Phys.Lipids_100_3 |
PubMedID: 10640192 |