Title : The complex of a bivalent derivative of galanthamine with torpedo acetylcholinesterase displays drastic deformation of the active-site gorge: implications for structure-based drug design - Greenblatt_2004_J.Am.Chem.Soc_126_15405 |
Author(s) : Greenblatt HM , Guillou C , Guenard D , Argaman A , Botti SA , Badet B , Thal C , Silman I , Sussman JL |
Ref : Journal of the American Chemical Society , 126 :15405 , 2004 |
Abstract : |
PubMedSearch : Greenblatt_2004_J.Am.Chem.Soc_126_15405 |
PubMedID: 15563167 |
Gene_locus related to this paper: torca-ACHE |
Title : Synthesis and structure-activity relationships of open D-Ring galanthamine analogues - Herlem_2003_Bioorg.Med.Chem.Lett_13_2389 |
Author(s) : Herlem D , Martin MT , Thal C , Guillou C |
Ref : Bioorganic & Medicinal Chemistry Lett , 13 :2389 , 2003 |
Abstract : |
PubMedSearch : Herlem_2003_Bioorg.Med.Chem.Lett_13_2389 |
PubMedID: 12824041 |
Title : (-)-9-Dehydrogalanthaminium bromide, a new cholinesterase inhibitor, enhances place and object recognition memory in young and old rats - Lamirault_2003_Neurobiol.Learn.Mem_80_113 |
Author(s) : Lamirault L , Guillou C , Thal C , Simon H |
Ref : Neurobiol Learn Mem , 80 :113 , 2003 |
Abstract : |
PubMedSearch : Lamirault_2003_Neurobiol.Learn.Mem_80_113 |
PubMedID: 12932426 |
Title : Combined treatment with galanthaminium bromide, a new cholinesterase inhibitor, and RS 67333, a partial agonist of 5-HT4 receptors, enhances place and object recognition in young adult and old rats - Lamirault_2003_Prog.Neuropsychopharmacol.Biol.Psychiatry_27_185 |
Author(s) : Lamirault L , Guillou C , Thal C , Simon H |
Ref : Prog Neuropsychopharmacol Biological Psychiatry , 27 :185 , 2003 |
Abstract : |
PubMedSearch : Lamirault_2003_Prog.Neuropsychopharmacol.Biol.Psychiatry_27_185 |
PubMedID: 12551743 |
Title : Potent acetylcholinesterase inhibitors: design, synthesis and structure-activity relationships of alkylene linked bis-galanthamine and galanthamine-galanthaminium salts - Guillou_2000_Bioorg.Med.Chem.Lett_10_637 |
Author(s) : Guillou C , Mary A , Renko DZ , Gras E , Thal C |
Ref : Bioorganic & Medicinal Chemistry Lett , 10 :637 , 2000 |
Abstract : |
PubMedSearch : Guillou_2000_Bioorg.Med.Chem.Lett_10_637 |
PubMedID: 10762042 |
Title : Potent acetylcholinesterase inhibitors: design, synthesis, and structure-activity relationships of bis-interacting ligands in the galanthamine series - Mary_1998_Bioorg.Med.Chem_6_1835 |
Author(s) : Mary A , Renko DZ , Guillou C , Thal C |
Ref : Bioorganic & Medicinal Chemistry , 6 :1835 , 1998 |
Abstract : |
PubMedSearch : Mary_1998_Bioorg.Med.Chem_6_1835 |
PubMedID: 9839013 |