Title : Turning Donepezil into a Multi-Target-Directed Ligand through a Merging Strategy - Perone_2021_ChemMedChem_16_187 |
Author(s) : Perone R , Albertini C , Uliassi E , Di Pietri F , de Sena Murteira Pinheiro P , Petralla S , Rizzardi N , Fato R , Pulkrabkova L , Soukup O , Tramarin A , Bartolini M , Bolognesi ML |
Ref : ChemMedChem , 16 :187 , 2021 |
Abstract : |
PubMedSearch : Perone_2021_ChemMedChem_16_187 |
PubMedID: 32716144 |
Title : Tackling neuroinflammation and cholinergic deficit in Alzheimer's disease: Multi-target inhibitors of cholinesterases, cyclooxygenase-2 and 15-lipoxygenase - AlFadly_2019_Eur.J.Med.Chem_167_161 |
Author(s) : AlFadly ED , Elzahhar PA , Tramarin A , Elkazaz S , Shaltout H , Abu-Serie MM , Janockova J , Soukup O , Ghareeb DA , El-Yazbi AF , Rafeh RW , Bakkar NZ , Kobeissy F , Iriepa I , Moraleda I , Saudi MNS , Bartolini M , Belal ASF |
Ref : Eur Journal of Medicinal Chemistry , 167 :161 , 2019 |
Abstract : |
PubMedSearch : AlFadly_2019_Eur.J.Med.Chem_167_161 |
PubMedID: 30771604 |
Title : Combination of human acetylcholinesterase and serum albumin sensing surfaces as highly informative analytical tool for inhibitor screening - Fabini_2018_J.Pharm.Biomed.Anal_155_177 |
Author(s) : Fabini E , Tramarin A , Bartolini M |
Ref : J Pharm Biomed Anal , 155 :177 , 2018 |
Abstract : |
PubMedSearch : Fabini_2018_J.Pharm.Biomed.Anal_155_177 |
PubMedID: 29635172 |
Title : Tacripyrimidines, the first tacrine-dihydropyrimidine hybrids, as multi-target-directed ligands for Alzheimer's disease - Chioua_2018_Eur.J.Med.Chem_155_839 |
Author(s) : Chioua M , Buzzi E , Moraleda I , Iriepa I , Maj M , Wnorowski A , Giovannini C , Tramarin A , Portali F , Ismaili L , Lopez-Alvarado P , Bolognesi ML , Jozwiak K , Menendez JC , Marco-Contelles J , Bartolini M |
Ref : Eur Journal of Medicinal Chemistry , 155 :839 , 2018 |
Abstract : |
PubMedSearch : Chioua_2018_Eur.J.Med.Chem_155_839 |
PubMedID: 29958119 |