Title : In vitro and in vivo metabolism of N-adamantyl substituted urea-based soluble epoxide hydrolase inhibitors - Liu_2015_Biochem.Pharmacol_98_718 |
Author(s) : Liu JY , Tsai HJ , Morisseau C , Lango J , Hwang SH , Watanabe T , Kim IH , Hammock BD |
Ref : Biochemical Pharmacology , 98 :718 , 2015 |
Abstract : |
PubMedSearch : Liu_2015_Biochem.Pharmacol_98_718 |
PubMedID: 26494425 |
Title : Soluble Epoxide Hydrolase Inhibition Exhibits Antihypertensive Actions Independently of Nitric Oxide in Mice with Renovascular Hypertension - Kopkan_2012_Kidney.Blood.Press.Res_35_595 |
Author(s) : Kopkan L , Huskova Z , Sporkova A , Varcabova S , Honetschlagerova Z , Hwang SH , Tsai HJ , Hammock BD , Imig JD , Kramer HJ , Burgelova M , Vojtiskova A , Kujal P , Vernerova Z , Cervenka L |
Ref : Kidney Blood Press Res , 35 :595 , 2012 |
Abstract : |
PubMedSearch : Kopkan_2012_Kidney.Blood.Press.Res_35_595 |
PubMedID: 22948718 |
Title : Renal mechanisms contributing to the antihypertensive action of soluble epoxide hydrolase inhibition in Ren-2 transgenic rats with inducible hypertension - Honetschlagerova_2011_J.Physiol_589_207 |
Author(s) : Honetschlagerova Z , Z ZH , Vanourkova Z , Sporkova A , Kramer HJ , Hwang SH , Tsai HJ , Hammock BD , Imig JD , Cervenka L , Kopkan L |
Ref : The Journal of Physiology , 589 :207 , 2011 |
Abstract : |
PubMedSearch : Honetschlagerova_2011_J.Physiol_589_207 |
PubMedID: 21078594 |
Title : Pharmacokinetic screening of soluble epoxide hydrolase inhibitors in dogs - Tsai_2010_Eur.J.Pharm.Sci_40_222 |
Author(s) : Tsai HJ , Hwang SH , Morisseau C , Yang J , Jones PD , Kasagami T , Kim IH , Hammock BD |
Ref : Eur J Pharm Sci , 40 :222 , 2010 |
Abstract : |
PubMedSearch : Tsai_2010_Eur.J.Pharm.Sci_40_222 |
PubMedID: 20359531 |
Title : Naturally occurring monoepoxides of eicosapentaenoic acid and docosahexaenoic acid are bioactive antihyperalgesic lipids - Morisseau_2010_J.Lipid.Res_51_3481 |
Author(s) : Morisseau C , Inceoglu B , Schmelzer K , Tsai HJ , Jinks SL , Hegedus CM , Hammock BD |
Ref : J Lipid Res , 51 :3481 , 2010 |
Abstract : |
PubMedSearch : Morisseau_2010_J.Lipid.Res_51_3481 |
PubMedID: 20664072 |
Title : Pharmacokinetic optimization of four soluble epoxide hydrolase inhibitors for use in a murine model of inflammation - Liu_2009_Br.J.Pharmacol_156_284 |
Author(s) : Liu JY , Tsai HJ , Hwang SH , Jones PD , Morisseau C , Hammock BD |
Ref : British Journal of Pharmacology , 156 :284 , 2009 |
Abstract : |
PubMedSearch : Liu_2009_Br.J.Pharmacol_156_284 |
PubMedID: 19154430 |
Title : Soluble epoxide hydrolase inhibitors reduce the development of atherosclerosis in apolipoprotein e-knockout mouse model - Ulu_2008_J.Cardiovasc.Pharmacol_52_314 |
Author(s) : Ulu A , Davis BB , Tsai HJ , Kim IH , Morisseau C , Inceoglu B , Fiehn O , Hammock BD , Weiss RH |
Ref : J Cardiovasc Pharmacol , 52 :314 , 2008 |
Abstract : |
PubMedSearch : Ulu_2008_J.Cardiovasc.Pharmacol_52_314 |
PubMedID: 18791465 |
Title : Inhibition of soluble epoxide hydrolase does not protect against endotoxin-mediated hepatic inflammation - Fife_2008_J.Pharmacol.Exp.Ther_327_707 |
Author(s) : Fife KL , Liu Y , Schmelzer KR , Tsai HJ , Kim IH , Morisseau C , Hammock BD , Kroetz DL |
Ref : Journal of Pharmacology & Experimental Therapeutics , 327 :707 , 2008 |
Abstract : |
PubMedSearch : Fife_2008_J.Pharmacol.Exp.Ther_327_707 |
PubMedID: 18815352 |
Title : Design of bioavailable derivatives of 12-(3-adamantan-1-yl-ureido)dodecanoic acid, a potent inhibitor of the soluble epoxide hydrolase - Kim_2007_Bioorg.Med.Chem_15_312 |
Author(s) : Kim IH , Nishi K , Tsai HJ , Bradford T , Koda Y , Watanabe T , Morisseau C , Blanchfield J , Toth I , Hammock BD |
Ref : Bioorganic & Medicinal Chemistry , 15 :312 , 2007 |
Abstract : |
PubMedSearch : Kim_2007_Bioorg.Med.Chem_15_312 |
PubMedID: 17046265 |
Gene_locus related to this paper: human-EPHX2 |
Title : Soluble epoxide hydrolase: a novel therapeutic target in stroke - Zhang_2007_J.Cereb.Blood.Flow.Metab_27_1931 |
Author(s) : Zhang W , Koerner IP , Noppens R , Grafe M , Tsai HJ , Morisseau C , Luria A , Hammock BD , Falck JR , Alkayed NJ |
Ref : Journal of Cerebral Blood Flow & Metabolism , 27 :1931 , 2007 |
Abstract : |
PubMedSearch : Zhang_2007_J.Cereb.Blood.Flow.Metab_27_1931 |
PubMedID: 17440491 |
Gene_locus related to this paper: human-EPHX2 |
Title : Orally bioavailable potent soluble epoxide hydrolase inhibitors - Hwang_2007_J.Med.Chem_50_3825 |
Author(s) : Hwang SH , Tsai HJ , Liu JY , Morisseau C , Hammock BD |
Ref : Journal of Medicinal Chemistry , 50 :3825 , 2007 |
Abstract : |
PubMedSearch : Hwang_2007_J.Med.Chem_50_3825 |
PubMedID: 17616115 |
Title : 1,3-disubstituted ureas functionalized with ether groups are potent inhibitors of the soluble epoxide hydrolase with improved pharmacokinetic properties - Kim_2007_J.Med.Chem_50_5217 |
Author(s) : Kim IH , Tsai HJ , Nishi K , Kasagami T , Morisseau C , Hammock BD |
Ref : Journal of Medicinal Chemistry , 50 :5217 , 2007 |
Abstract : |
PubMedSearch : Kim_2007_J.Med.Chem_50_5217 |
PubMedID: 17894481 |
Title : The soluble epoxide hydrolase as a pharmaceutical target for hypertension - Chiamvimonvat_2007_J.Cardiovasc.Pharmacol_50_225 |
Author(s) : Chiamvimonvat N , Ho CM , Tsai HJ , Hammock BD |
Ref : J Cardiovasc Pharmacol , 50 :225 , 2007 |
Abstract : |
PubMedSearch : Chiamvimonvat_2007_J.Cardiovasc.Pharmacol_50_225 |
PubMedID: 17878749 |
Title : Optimization of amide-based inhibitors of soluble epoxide hydrolase with improved water solubility - Kim_2005_J.Med.Chem_48_3621 |
Author(s) : Kim IH , Heirtzler FR , Morisseau C , Nishi K , Tsai HJ , Hammock BD |
Ref : Journal of Medicinal Chemistry , 48 :3621 , 2005 |
Abstract : |
PubMedSearch : Kim_2005_J.Med.Chem_48_3621 |
PubMedID: 15887969 |
Title : Quantitative structure-activity relationships for the pre-steady state acetylcholinesterase inhibition by carbamates - Lin_2004_J.Biochem.Mol.Toxicol_18_353 |
Author(s) : Lin G , Liao WC , Chan CH , Wu YH , Tsai HJ , Hsieh CW |
Ref : J Biochem Mol Toxicol , 18 :353 , 2004 |
Abstract : |
PubMedSearch : Lin_2004_J.Biochem.Mol.Toxicol_18_353 |
PubMedID: 15674842 |
Title : Cage amines as the stopper inhibitors of cholinesterases - Lin_2003_Bioorg.Med.Chem.Lett_13_2887 |
Author(s) : Lin G , Tsai HJ , Tsai YH |
Ref : Bioorganic & Medicinal Chemistry Lett , 13 :2887 , 2003 |
Abstract : |
PubMedSearch : Lin_2003_Bioorg.Med.Chem.Lett_13_2887 |
PubMedID: 14611850 |
Title : Transgenic zebrafish with fluorescent germ cell: a useful tool to visualize germ cell proliferation and juvenile hermaphroditism in vivo - Hsiao_2003_Dev.Biol_262_313 |
Author(s) : Hsiao CD , Tsai HJ |
Ref : Developmental Biology , 262 :313 , 2003 |
Abstract : |
PubMedSearch : Hsiao_2003_Dev.Biol_262_313 |
PubMedID: 14550794 |
Title : Molecular structure and developmental expression of three muscle-type troponin T genes in zebrafish - Hsiao_2003_Dev.Dyn_227_266 |
Author(s) : Hsiao CD , Tsai WY , Horng LS , Tsai HJ |
Ref : Developmental Dynamics , 227 :266 , 2003 |
Abstract : |
PubMedSearch : Hsiao_2003_Dev.Dyn_227_266 |
PubMedID: 12761854 |
Title : Novel regulatory sequence -82\/-62 functions as a key element to drive the somite-specificity of zebrafish myf-5 - Chen_2003_Dev.Dyn_228_41 |
Author(s) : Chen YH , Lee HC , Liu CF , Lin CY , Tsai HJ |
Ref : Developmental Dynamics , 228 :41 , 2003 |
Abstract : |
PubMedSearch : Chen_2003_Dev.Dyn_228_41 |
PubMedID: 12950078 |
Title : Functional analysis of the proximal promoter regions of fish rhodopsin and myf-5 genes using transgenesis - Wang_2002_Mar.Biotechnol.(NY)_4_247 |
Author(s) : Wang TM , Chen YH , Liu CF , Tsai HJ |
Ref : Mar Biotechnol (NY) , 4 :247 , 2002 |
Abstract : |
PubMedSearch : Wang_2002_Mar.Biotechnol.(NY)_4_247 |
PubMedID: 14961258 |
Title : Expression, purification and DNA-binding activity of tilapia muscle-specific transcription factor, MyoD, produced in Escherichia coli - Chen_2002_Comp.Biochem.Physiol.B.Biochem.Mol.Biol_131_795 |
Author(s) : Chen YH , Liang CT , Tsai HJ |
Ref : Comparative Biochemistry & Physiology B Biochem Mol Biol , 131 :795 , 2002 |
Abstract : |
PubMedSearch : Chen_2002_Comp.Biochem.Physiol.B.Biochem.Mol.Biol_131_795 |
PubMedID: 11923092 |
Title : Treatment with Myf5-morpholino results in somite patterning and brain formation defects in zebrafish - Chen_2002_Differentiation_70_447 |
Author(s) : Chen YH , Tsai HJ |
Ref : Differentiation , 70 :447 , 2002 |
Abstract : |
PubMedSearch : Chen_2002_Differentiation_70_447 |
PubMedID: 12366382 |
Title : Reversal of mivacurium chloride: edrophonium of spontaneous recovery in microscopic laryngeal surgery - Ting_2001_Acta.Anaesthesiol.Sin_39_157 |
Author(s) : Ting CK , Lin SM , Yang YW , Tsai HJ , Lao HC , Chu YC , Tsai SK |
Ref : Acta Anaesthesiol Sin , 39 :157 , 2001 |
Abstract : |
PubMedSearch : Ting_2001_Acta.Anaesthesiol.Sin_39_157 |
PubMedID: 11840581 |
Title : Molecular structure, dynamic expression, and promoter analysis of zebrafish (Danio rerio) myf-5 gene - Chen_2001_Genesis_29_22 |
Author(s) : Chen YH , Lee WC , Liu CF , Tsai HJ |
Ref : Genesis , 29 :22 , 2001 |
Abstract : |
PubMedSearch : Chen_2001_Genesis_29_22 |
PubMedID: 11135459 |
Title : Uniform GFP-expression in transgenic medaka (Oryzias latipes) at the F0 generation - Chou_2001_Transgenic.Res_10_303 |
Author(s) : Chou CY , Horng LS , Tsai HJ |
Ref : Transgenic Res , 10 :303 , 2001 |
Abstract : |
PubMedSearch : Chou_2001_Transgenic.Res_10_303 |
PubMedID: 11592710 |
Title : Muscle regulatory factor gene: zebrafish (Danio rerio) myogenin cDNA - Chen_2000_Comp.Biochem.Physiol.B.Biochem.Mol.Biol_127_97 |
Author(s) : Chen YH , Lee WC , Cheng CH , Tsai HJ |
Ref : Comparative Biochemistry & Physiology B Biochem Mol Biol , 127 :97 , 2000 |
Abstract : |
PubMedSearch : Chen_2000_Comp.Biochem.Physiol.B.Biochem.Mol.Biol_127_97 |
PubMedID: 11126756 |
Title : Effects of choline and other nicotinic agonists on the tectum of juvenile and adult Xenopus frogs: a patch-clamp study - Titmus_1999_Neurosci_91_753 |
Author(s) : Titmus MJ , Tsai HJ , Lima R , Udin SB |
Ref : Neuroscience , 91 :753 , 1999 |
Abstract : |
PubMedSearch : Titmus_1999_Neurosci_91_753 |
PubMedID: 10366031 |