Tetracaine

Local anesthetic, substrate as well as inhibitor, C15H24N2O2,[94-24-6],264.3. Tetracaine is an allosteric blocker of channel function

General

Type : Local anesthetic, Drug, Not AlphaBeta Hydrolase target, Organochlorine

Chemical_Nomenclature : 4-(Butylamino)benzoicacid 2-(dimethylamino)ehtyl ester

Canonical SMILES :

InChI :

InChIKey :

Other name(s) : Amethocaine  ||  Uromucaesthin  ||  Contralgin  ||  Fissucain  ||  Intercain  ||  Laudocaine  ||  Medicaine  ||  Meethobalm  ||  Metraspray  ||  Cetacaine  ||  Pontocain


MW : 300.83

Formula : C15H25ClN2O2

CAS_number : 136-47-0

PubChem : 5411

UniChem :

Wikipedia : Tetracaine

Target

Families : Tetracaine ligand of proteins in family
BCHE

References (3)

Title : Genetic variants of human serum cholinesterase influence metabolism of the muscle relaxant succinylcholine. - Lockridge_1990_Pharmacol.Ther_47_35
Author(s) : Lockridge O
Ref : Pharmacol Ther , 47 :35 , 1990
Abstract :
PubMedSearch : Lockridge_1990_Pharmacol.Ther_47_35
PubMedID: 2195556
Gene_locus related to this paper: human-BCHE

Title : Differential inhibition of plasma cholinesterase variants using the dibutyrate analogue of pancuronium bromide - Whittaker_1981_Hum.Hered_31_242
Author(s) : Whittaker M , Britten JJ
Ref : Hum Hered , 31 :242 , 1981
Abstract :
PubMedSearch : Whittaker_1981_Hum.Hered_31_242
PubMedID: 7287015

Title : The activity of various esterase inhibitors towards atypical human serum cholinesterase -
Author(s) : Kalow W , Davies R0
Ref : Biochemical Pharmacology , 1 :183 , 1958
PubMedID: