Tetracaine
Local anesthetic, substrate as well as inhibitor, C15H24N2O2,[94-24-6],264.3. Tetracaine is an allosteric blocker of channel function
General
Type : Local anesthetic, Drug, Not A\/B H target
Chemical_Nomenclature : 4-(Butylamino)benzoicacid 2-(dimethylamino)ehtyl ester
Canonical SMILES : CCCCNC1=CC=C(C=C1)C(=O)OCCN(C)C
InChI : InChI=1S\/C15H24N2O2\/c1-4-5-10-16-14-8-6-13(7-9-14)15(18)19-12-11-17(2)3\/h6-9,16H,4-5,10-12H2,1-3H3
InChIKey : GKCBAIGFKIBETG-UHFFFAOYSA-N
Other name(s) : Amethocaine, Uromucaesthin, Contralgin, Fissucain, Intercain, Laudocaine, Medicaine, Meethobalm, Metraspray, Cetacaine, Pontocain
MW : 300.83
Formula : C15H25ClN2O2
CAS_number : 136-47-0
PubChem : 5411
UniChem : GKCBAIGFKIBETG-UHFFFAOYSA-N
Wikipedia : Tetracaine
Target
Families : Tetracaine ligand of proteins in family
BCHE
References (3)
| Title : Genetic variants of human serum cholinesterase influence metabolism of the muscle relaxant succinylcholine. - Lockridge_1990_Pharmacol.Ther_47_35 |
| Author(s) : Lockridge O |
| Ref : Pharmacol Ther , 47 :35 , 1990 |
| PubMedID: 2195556 |
| Gene_locus related to this paper: human-BCHE |
| Title : Differential inhibition of plasma cholinesterase variants using the dibutyrate analogue of pancuronium bromide - Whittaker_1981_Hum.Hered_31_242 |
| Author(s) : Whittaker M , Britten JJ |
| Ref : Hum Hered , 31 :242 , 1981 |
| PubMedID: 7287015 |