Title : Novel insights into m3 muscarinic acetylcholine receptor physiology and structure - Kruse_2014_J.Mol.Neurosci_53_316 |
Author(s) : Kruse AC , Li J , Hu J , Kobilka BK , Wess J |
Ref : Journal of Molecular Neuroscience , 53 :316 , 2014 |
Abstract : |
PubMedSearch : Kruse_2014_J.Mol.Neurosci_53_316 |
PubMedID: 24068573 |
Title : Muscarinic acetylcholine receptor X-ray structures: potential implications for drug development - Kruse_2014_Curr.Opin.Pharmacol_16_24 |
Author(s) : Kruse AC , Hu J , Kobilka BK , Wess J |
Ref : Curr Opin Pharmacol , 16 :24 , 2014 |
Abstract : |
PubMedSearch : Kruse_2014_Curr.Opin.Pharmacol_16_24 |
PubMedID: 24662799 |
Title : Muscarinic acetylcholine receptors: novel opportunities for drug development - Kruse_2014_Nat.Rev.Drug.Discov_13_549 |
Author(s) : Kruse AC , Kobilka BK , Gautam D , Sexton PM , Christopoulos A , Wess J |
Ref : Nat Rev Drug Discov , 13 :549 , 2014 |
Abstract : |
PubMedSearch : Kruse_2014_Nat.Rev.Drug.Discov_13_549 |
PubMedID: 24903776 |
Title : Activation and allosteric modulation of a muscarinic acetylcholine receptor - Kruse_2013_Nature_504_101 |
Author(s) : Kruse AC , Ring AM , Manglik A , Hu J , Hu K , Eitel K , Hubner H , Pardon E , Valant C , Sexton PM , Christopoulos A , Felder CC , Gmeiner P , Steyaert J , Weis WI , Garcia KC , Wess J , Kobilka BK |
Ref : Nature , 504 :101 , 2013 |
Abstract : |
PubMedSearch : Kruse_2013_Nature_504_101 |
PubMedID: 24256733 |
Title : Muscarinic receptors as model targets and antitargets for structure-based ligand discovery - Kruse_2013_Mol.Pharmacol_84_528 |
Author(s) : Kruse AC , Weiss DR , Rossi M , Hu J , Hu K , Eitel K , Gmeiner P , Wess J , Kobilka BK , Shoichet BK |
Ref : Molecular Pharmacology , 84 :528 , 2013 |
Abstract : |
PubMedSearch : Kruse_2013_Mol.Pharmacol_84_528 |
PubMedID: 23887926 |
Title : Structure of the human M2 muscarinic acetylcholine receptor bound to an antagonist - Haga_2012_Nature_482_547 |
Author(s) : Haga K , Kruse AC , Asada H , Yurugi-Kobayashi T , Shiroishi M , Zhang C , Weis WI , Okada T , Kobilka BK , Haga T , Kobayashi T |
Ref : Nature , 482 :547 , 2012 |
Abstract : |
PubMedSearch : Haga_2012_Nature_482_547 |
PubMedID: 22278061 |
Title : Structure and dynamics of the M3 muscarinic acetylcholine receptor - Kruse_2012_Nature_482_552 |
Author(s) : Kruse AC , Hu J , Pan AC , Arlow DH , Rosenbaum DM , Rosemond E , Green HF , Liu T , Chae PS , Dror RO , Shaw DE , Weis WI , Wess J , Kobilka BK |
Ref : Nature , 482 :552 , 2012 |
Abstract : |
PubMedSearch : Kruse_2012_Nature_482_552 |
PubMedID: 22358844 |