Title : Cholinesterase inhibitory activity of highly functionalized fluorinated spiropyrrolidine heterocyclic hybrids - Kumar_2021_Saudi.J.Biol.Sci_28_754 |
Author(s) : Kumar RS , Almansour AI , Arumugam N , Kotresha D , Manohar TS , Venketesh S |
Ref : Saudi J Biol Sci , 28 :754 , 2021 |
Abstract : Kumar_2021_Saudi.J.Biol.Sci_28_754 |
ESTHER : Kumar_2021_Saudi.J.Biol.Sci_28_754 |
PubMedSearch : Kumar_2021_Saudi.J.Biol.Sci_28_754 |
PubMedID: 33424364 |
Title : Design, synthesis and cholinesterase inhibitory activity of novel spiropyrrolidine tethered imidazole heterocyclic hybrids - Almansour_2019_Bioorg.Med.Chem.Lett__126789 |
Author(s) : Almansour AI , Arumugam N , Kumar RS , Kotresha D , Manohar TS , Venketesh S |
Ref : Bioorganic & Medicinal Chemistry Lett , :126789 , 2019 |
Abstract : Almansour_2019_Bioorg.Med.Chem.Lett__126789 |
ESTHER : Almansour_2019_Bioorg.Med.Chem.Lett__126789 |
PubMedSearch : Almansour_2019_Bioorg.Med.Chem.Lett__126789 |
PubMedID: 31753696 |
Title : Dispiropyrrolidinyl-piperidone embedded indeno[1,2-b]quinoxaline heterocyclic hybrids: Synthesis, cholinesterase inhibitory activity and their molecular docking simulation - Arumugam_2019_Bioorg.Med.Chem_27_2621 |
Author(s) : Arumugam N , Almansour AI , Kumar RS , Kotresha D , Saiswaroop R , Venketesh S |
Ref : Bioorganic & Medicinal Chemistry , 27 :2621 , 2019 |
Abstract : Arumugam_2019_Bioorg.Med.Chem_27_2621 |
ESTHER : Arumugam_2019_Bioorg.Med.Chem_27_2621 |
PubMedSearch : Arumugam_2019_Bioorg.Med.Chem_27_2621 |
PubMedID: 30952387 |
Title : Ionic liquid-enabled synthesis, cholinesterase inhibitory activity, and molecular docking study of highly functionalized tetrasubstituted pyrrolidines - Kumar_2018_Bioorg.Chem_77_263 |
Author(s) : Kumar RS , Almansour AI , Arumugam N , Althomili DMQ , Altaf M , Basiri A , D K , Sai Manohar T , S V |
Ref : Bioorg Chem , 77 :263 , 2018 |
Abstract : Kumar_2018_Bioorg.Chem_77_263 |
ESTHER : Kumar_2018_Bioorg.Chem_77_263 |
PubMedSearch : Kumar_2018_Bioorg.Chem_77_263 |
PubMedID: 29421701 |
Title : Highly functionalized 2-amino-4H-pyrans as potent cholinesterase inhibitors - Kumar_2018_Bioorg.Chem_81_134 |
Author(s) : Kumar RS , Almansour AI , Arumugam N , Al-Thamili DM , Basiri A , Kotresha D , Manohar TS , Venketesh S , Asad M , Asiri AM |
Ref : Bioorg Chem , 81 :134 , 2018 |
Abstract : Kumar_2018_Bioorg.Chem_81_134 |
ESTHER : Kumar_2018_Bioorg.Chem_81_134 |
PubMedSearch : Kumar_2018_Bioorg.Chem_81_134 |
PubMedID: 30121001 |
Title : Synthesis and cholinesterase inhibitory activity study of new piperidone grafted spiropyrrolidines - Basiri_2017_Bioorg.Chem_75_210 |
Author(s) : Basiri A , Abd Razik BM , Ezzat MO , Kia Y , Kumar RS , Almansour AI , Arumugam N , Murugaiyah V |
Ref : Bioorg Chem , 75 :210 , 2017 |
Abstract : Basiri_2017_Bioorg.Chem_75_210 |
ESTHER : Basiri_2017_Bioorg.Chem_75_210 |
PubMedSearch : Basiri_2017_Bioorg.Chem_75_210 |
PubMedID: 28987876 |
Title : A facile ionic liquid promoted synthesis, cholinesterase inhibitory activity and molecular modeling study of novel highly functionalized spiropyrrolidines - Almansour_2015_Molecules_20_2296 |
Author(s) : Almansour AI , Kumar RS , Arumugam N , Basiri A , Kia Y , Ali MA , Farooq M , Murugaiyah V |
Ref : Molecules , 20 :2296 , 2015 |
Abstract : Almansour_2015_Molecules_20_2296 |
ESTHER : Almansour_2015_Molecules_20_2296 |
PubMedSearch : Almansour_2015_Molecules_20_2296 |
PubMedID: 25642838 |
Title : An efficient ionic liquid mediated synthesis, cholinesterase inhibitory activity and molecular modeling study of novel piperidone embedded alpha,beta-unsaturated ketones - Kia_2014_Med.Chem_10_512 |
Author(s) : Kia Y , Osman H , Kumar RS , Murugaiyah V , Basiri A , Khaw KY , Rosli MM |
Ref : Med Chem , 10 :512 , 2014 |
Abstract : Kia_2014_Med.Chem_10_512 |
ESTHER : Kia_2014_Med.Chem_10_512 |
PubMedSearch : Kia_2014_Med.Chem_10_512 |
PubMedID: 24138113 |
Title : An expedient synthesis and screening for antiacetylcholinesterase activity of piperidine embedded novel pentacyclic cage compounds - Kumar_2014_Med.Chem_10_228 |
Author(s) : Kumar RS , Almansour AI , Arumugam N , Osman H , Ali MA , Basiri A , Kia Y |
Ref : Med Chem , 10 :228 , 2014 |
Abstract : Kumar_2014_Med.Chem_10_228 |
ESTHER : Kumar_2014_Med.Chem_10_228 |
PubMedSearch : Kumar_2014_Med.Chem_10_228 |
PubMedID: 23627271 |
Title : Cholinesterase inhibitory activity versus aromatic core multiplicity: A facile green synthesis and molecular docking study of novel piperidone embedded thiazolopyrimidines - Basiri_2014_Bioorg.Med.Chem_22_906 |
Author(s) : Basiri A , Murugaiyah V , Osman H , Kumar RS , Kia Y , Hooda A , Parsons RB |
Ref : Bioorganic & Medicinal Chemistry , 22 :906 , 2014 |
Abstract : Basiri_2014_Bioorg.Med.Chem_22_906 |
ESTHER : Basiri_2014_Bioorg.Med.Chem_22_906 |
PubMedSearch : Basiri_2014_Bioorg.Med.Chem_22_906 |
PubMedID: 24369842 |
Title : Ionic liquid mediated synthesis of mono- and bis-spirooxindole-hexahydropyrrolidines as cholinesterase inhibitors and their molecular docking studies - Kia_2014_Bioorg.Med.Chem_22_1318 |
Author(s) : Kia Y , Osman H , Kumar RS , Basiri A , Murugaiyah V |
Ref : Bioorganic & Medicinal Chemistry , 22 :1318 , 2014 |
Abstract : Kia_2014_Bioorg.Med.Chem_22_1318 |
ESTHER : Kia_2014_Bioorg.Med.Chem_22_1318 |
PubMedSearch : Kia_2014_Bioorg.Med.Chem_22_1318 |
PubMedID: 24461561 |
Title : Synthesis and discovery of novel piperidone-grafted mono- and bis-spirooxindole-hexahydropyrrolizines as potent cholinesterase inhibitors - Kia_2013_Bioorg.Med.Chem_21_1696 |
Author(s) : Kia Y , Osman H , Kumar RS , Murugaiyah V , Basiri A , Perumal S , Wahab HA , Bing CS |
Ref : Bioorganic & Medicinal Chemistry , 21 :1696 , 2013 |
Abstract : Kia_2013_Bioorg.Med.Chem_21_1696 |
ESTHER : Kia_2013_Bioorg.Med.Chem_21_1696 |
PubMedSearch : Kia_2013_Bioorg.Med.Chem_21_1696 |
PubMedID: 23454132 |
Title : An expedient, ionic liquid mediated multi-component synthesis of novel piperidone grafted cholinesterase enzymes inhibitors and their molecular modeling study - Basiri_2013_Eur.J.Med.Chem_67C_221 |
Author(s) : Basiri A , Murugaiyah V , Osman H , Kumar RS , Kia Y , Awang KB , Ali MA |
Ref : Eur Journal of Medicinal Chemistry , 67C :221 , 2013 |
Abstract : Basiri_2013_Eur.J.Med.Chem_67C_221 |
ESTHER : Basiri_2013_Eur.J.Med.Chem_67C_221 |
PubMedSearch : Basiri_2013_Eur.J.Med.Chem_67C_221 |
PubMedID: 23871902 |
Title : AChE inhibitor: a regio- and stereo-selective 1,3-dipolar cycloaddition for the synthesis of novel substituted 5,6-dimethoxy spiro[5.3']-oxindole-spiro-[6.3'']-2,3-dihydro-1H-inden-1''-one-7-(substituted aryl)-tetrahydro-1H-pyrrolo[1,2-c][1,3]thiazole - Ashraf_2012_Bioorg.Med.Chem.Lett_22_508 |
Author(s) : Ashraf Ali M , Ismail R , Choon TS , Kumar RS , Osman H , Arumugam N , Almansour AI , Elumalai K , Singh A |
Ref : Bioorganic & Medicinal Chemistry Lett , 22 :508 , 2012 |
Abstract : Ashraf_2012_Bioorg.Med.Chem.Lett_22_508 |
ESTHER : Ashraf_2012_Bioorg.Med.Chem.Lett_22_508 |
PubMedSearch : Ashraf_2012_Bioorg.Med.Chem.Lett_22_508 |
PubMedID: 22142546 |
Title : Substituted spiro [2.3'] oxindolespiro [3.2'']-5,6-dimethoxy-indane-1''-one-pyrrolidine analogue as inhibitors of acetylcholinesterase - Ali_2010_Bioorg.Med.Chem.Lett_20_7064 |
Author(s) : Ali MA , Ismail R , Choon TS , Yoon YK , Wei AC , Pandian S , Kumar RS , Osman H , Manogaran E |
Ref : Bioorganic & Medicinal Chemistry Lett , 20 :7064 , 2010 |
Abstract : Ali_2010_Bioorg.Med.Chem.Lett_20_7064 |
ESTHER : Ali_2010_Bioorg.Med.Chem.Lett_20_7064 |
PubMedSearch : Ali_2010_Bioorg.Med.Chem.Lett_20_7064 |
PubMedID: 20951037 |