Kumar RS

References (15)

Title : Cholinesterase inhibitory activity of highly functionalized fluorinated spiropyrrolidine heterocyclic hybrids - Kumar_2021_Saudi.J.Biol.Sci_28_754
Author(s) : Kumar RS , Almansour AI , Arumugam N , Kotresha D , Manohar TS , Venketesh S
Ref : Saudi J Biol Sci , 28 :754 , 2021
Abstract : Kumar_2021_Saudi.J.Biol.Sci_28_754
ESTHER : Kumar_2021_Saudi.J.Biol.Sci_28_754
PubMedSearch : Kumar_2021_Saudi.J.Biol.Sci_28_754
PubMedID: 33424364

Title : Design, synthesis and cholinesterase inhibitory activity of novel spiropyrrolidine tethered imidazole heterocyclic hybrids - Almansour_2019_Bioorg.Med.Chem.Lett__126789
Author(s) : Almansour AI , Arumugam N , Kumar RS , Kotresha D , Manohar TS , Venketesh S
Ref : Bioorganic & Medicinal Chemistry Lett , :126789 , 2019
Abstract : Almansour_2019_Bioorg.Med.Chem.Lett__126789
ESTHER : Almansour_2019_Bioorg.Med.Chem.Lett__126789
PubMedSearch : Almansour_2019_Bioorg.Med.Chem.Lett__126789
PubMedID: 31753696

Title : Dispiropyrrolidinyl-piperidone embedded indeno[1,2-b]quinoxaline heterocyclic hybrids: Synthesis, cholinesterase inhibitory activity and their molecular docking simulation - Arumugam_2019_Bioorg.Med.Chem_27_2621
Author(s) : Arumugam N , Almansour AI , Kumar RS , Kotresha D , Saiswaroop R , Venketesh S
Ref : Bioorganic & Medicinal Chemistry , 27 :2621 , 2019
Abstract : Arumugam_2019_Bioorg.Med.Chem_27_2621
ESTHER : Arumugam_2019_Bioorg.Med.Chem_27_2621
PubMedSearch : Arumugam_2019_Bioorg.Med.Chem_27_2621
PubMedID: 30952387

Title : Ionic liquid-enabled synthesis, cholinesterase inhibitory activity, and molecular docking study of highly functionalized tetrasubstituted pyrrolidines - Kumar_2018_Bioorg.Chem_77_263
Author(s) : Kumar RS , Almansour AI , Arumugam N , Althomili DMQ , Altaf M , Basiri A , D K , Sai Manohar T , S V
Ref : Bioorg Chem , 77 :263 , 2018
Abstract : Kumar_2018_Bioorg.Chem_77_263
ESTHER : Kumar_2018_Bioorg.Chem_77_263
PubMedSearch : Kumar_2018_Bioorg.Chem_77_263
PubMedID: 29421701

Title : Highly functionalized 2-amino-4H-pyrans as potent cholinesterase inhibitors - Kumar_2018_Bioorg.Chem_81_134
Author(s) : Kumar RS , Almansour AI , Arumugam N , Al-Thamili DM , Basiri A , Kotresha D , Manohar TS , Venketesh S , Asad M , Asiri AM
Ref : Bioorg Chem , 81 :134 , 2018
Abstract : Kumar_2018_Bioorg.Chem_81_134
ESTHER : Kumar_2018_Bioorg.Chem_81_134
PubMedSearch : Kumar_2018_Bioorg.Chem_81_134
PubMedID: 30121001

Title : Synthesis and cholinesterase inhibitory activity study of new piperidone grafted spiropyrrolidines - Basiri_2017_Bioorg.Chem_75_210
Author(s) : Basiri A , Abd Razik BM , Ezzat MO , Kia Y , Kumar RS , Almansour AI , Arumugam N , Murugaiyah V
Ref : Bioorg Chem , 75 :210 , 2017
Abstract : Basiri_2017_Bioorg.Chem_75_210
ESTHER : Basiri_2017_Bioorg.Chem_75_210
PubMedSearch : Basiri_2017_Bioorg.Chem_75_210
PubMedID: 28987876

Title : A facile ionic liquid promoted synthesis, cholinesterase inhibitory activity and molecular modeling study of novel highly functionalized spiropyrrolidines - Almansour_2015_Molecules_20_2296
Author(s) : Almansour AI , Kumar RS , Arumugam N , Basiri A , Kia Y , Ali MA , Farooq M , Murugaiyah V
Ref : Molecules , 20 :2296 , 2015
Abstract : Almansour_2015_Molecules_20_2296
ESTHER : Almansour_2015_Molecules_20_2296
PubMedSearch : Almansour_2015_Molecules_20_2296
PubMedID: 25642838

Title : An efficient ionic liquid mediated synthesis, cholinesterase inhibitory activity and molecular modeling study of novel piperidone embedded alpha,beta-unsaturated ketones - Kia_2014_Med.Chem_10_512
Author(s) : Kia Y , Osman H , Kumar RS , Murugaiyah V , Basiri A , Khaw KY , Rosli MM
Ref : Med Chem , 10 :512 , 2014
Abstract : Kia_2014_Med.Chem_10_512
ESTHER : Kia_2014_Med.Chem_10_512
PubMedSearch : Kia_2014_Med.Chem_10_512
PubMedID: 24138113

Title : An expedient synthesis and screening for antiacetylcholinesterase activity of piperidine embedded novel pentacyclic cage compounds - Kumar_2014_Med.Chem_10_228
Author(s) : Kumar RS , Almansour AI , Arumugam N , Osman H , Ali MA , Basiri A , Kia Y
Ref : Med Chem , 10 :228 , 2014
Abstract : Kumar_2014_Med.Chem_10_228
ESTHER : Kumar_2014_Med.Chem_10_228
PubMedSearch : Kumar_2014_Med.Chem_10_228
PubMedID: 23627271

Title : Cholinesterase inhibitory activity versus aromatic core multiplicity: A facile green synthesis and molecular docking study of novel piperidone embedded thiazolopyrimidines - Basiri_2014_Bioorg.Med.Chem_22_906
Author(s) : Basiri A , Murugaiyah V , Osman H , Kumar RS , Kia Y , Hooda A , Parsons RB
Ref : Bioorganic & Medicinal Chemistry , 22 :906 , 2014
Abstract : Basiri_2014_Bioorg.Med.Chem_22_906
ESTHER : Basiri_2014_Bioorg.Med.Chem_22_906
PubMedSearch : Basiri_2014_Bioorg.Med.Chem_22_906
PubMedID: 24369842

Title : Ionic liquid mediated synthesis of mono- and bis-spirooxindole-hexahydropyrrolidines as cholinesterase inhibitors and their molecular docking studies - Kia_2014_Bioorg.Med.Chem_22_1318
Author(s) : Kia Y , Osman H , Kumar RS , Basiri A , Murugaiyah V
Ref : Bioorganic & Medicinal Chemistry , 22 :1318 , 2014
Abstract : Kia_2014_Bioorg.Med.Chem_22_1318
ESTHER : Kia_2014_Bioorg.Med.Chem_22_1318
PubMedSearch : Kia_2014_Bioorg.Med.Chem_22_1318
PubMedID: 24461561

Title : Synthesis and discovery of novel piperidone-grafted mono- and bis-spirooxindole-hexahydropyrrolizines as potent cholinesterase inhibitors - Kia_2013_Bioorg.Med.Chem_21_1696
Author(s) : Kia Y , Osman H , Kumar RS , Murugaiyah V , Basiri A , Perumal S , Wahab HA , Bing CS
Ref : Bioorganic & Medicinal Chemistry , 21 :1696 , 2013
Abstract : Kia_2013_Bioorg.Med.Chem_21_1696
ESTHER : Kia_2013_Bioorg.Med.Chem_21_1696
PubMedSearch : Kia_2013_Bioorg.Med.Chem_21_1696
PubMedID: 23454132

Title : An expedient, ionic liquid mediated multi-component synthesis of novel piperidone grafted cholinesterase enzymes inhibitors and their molecular modeling study - Basiri_2013_Eur.J.Med.Chem_67C_221
Author(s) : Basiri A , Murugaiyah V , Osman H , Kumar RS , Kia Y , Awang KB , Ali MA
Ref : Eur Journal of Medicinal Chemistry , 67C :221 , 2013
Abstract : Basiri_2013_Eur.J.Med.Chem_67C_221
ESTHER : Basiri_2013_Eur.J.Med.Chem_67C_221
PubMedSearch : Basiri_2013_Eur.J.Med.Chem_67C_221
PubMedID: 23871902

Title : AChE inhibitor: a regio- and stereo-selective 1,3-dipolar cycloaddition for the synthesis of novel substituted 5,6-dimethoxy spiro[5.3']-oxindole-spiro-[6.3'']-2,3-dihydro-1H-inden-1''-one-7-(substituted aryl)-tetrahydro-1H-pyrrolo[1,2-c][1,3]thiazole - Ashraf_2012_Bioorg.Med.Chem.Lett_22_508
Author(s) : Ashraf Ali M , Ismail R , Choon TS , Kumar RS , Osman H , Arumugam N , Almansour AI , Elumalai K , Singh A
Ref : Bioorganic & Medicinal Chemistry Lett , 22 :508 , 2012
Abstract : Ashraf_2012_Bioorg.Med.Chem.Lett_22_508
ESTHER : Ashraf_2012_Bioorg.Med.Chem.Lett_22_508
PubMedSearch : Ashraf_2012_Bioorg.Med.Chem.Lett_22_508
PubMedID: 22142546

Title : Substituted spiro [2.3'] oxindolespiro [3.2'']-5,6-dimethoxy-indane-1''-one-pyrrolidine analogue as inhibitors of acetylcholinesterase - Ali_2010_Bioorg.Med.Chem.Lett_20_7064
Author(s) : Ali MA , Ismail R , Choon TS , Yoon YK , Wei AC , Pandian S , Kumar RS , Osman H , Manogaran E
Ref : Bioorganic & Medicinal Chemistry Lett , 20 :7064 , 2010
Abstract : Ali_2010_Bioorg.Med.Chem.Lett_20_7064
ESTHER : Ali_2010_Bioorg.Med.Chem.Lett_20_7064
PubMedSearch : Ali_2010_Bioorg.Med.Chem.Lett_20_7064
PubMedID: 20951037