Title : Discovery and development of a potent and highly selective small molecule muscarinic acetylcholine receptor subtype I (mAChR 1 or M1) antagonist in vitro and in vivo probe - Weaver_2009_Curr.Top.Med.Chem_9_1217 |
Author(s) : Weaver CD , Sheffler DJ , Lewis LM , Bridges TM , Williams R , Nalywajko NT , Kennedy JP , Mulder MM , Jadhav S , Aldrich LA , Jones CK , Marlo JE , Niswender CM , Mock MM , Zheng F , Conn PJ , Lindsley CW |
Ref : Curr Top Med Chem , 9 :1217 , 2009 |
Abstract : Weaver_2009_Curr.Top.Med.Chem_9_1217 |
ESTHER : Weaver_2009_Curr.Top.Med.Chem_9_1217 |
PubMedSearch : Weaver_2009_Curr.Top.Med.Chem_9_1217 |
PubMedID: 19807667 |
Title : Discovery and characterization of novel allosteric potentiators of M1 muscarinic receptors reveals multiple modes of activity - Marlo_2009_Mol.Pharmacol_75_577 |
Author(s) : Marlo JE , Niswender CM , Days EL , Bridges TM , Xiang Y , Rodriguez AL , Shirey JK , Brady AE , Nalywajko T , Luo Q , Austin CA , Williams MB , Kim K , Williams R , Orton D , Brown HA , Lindsley CW , Weaver CD , Conn PJ |
Ref : Molecular Pharmacology , 75 :577 , 2009 |
Abstract : Marlo_2009_Mol.Pharmacol_75_577 |
ESTHER : Marlo_2009_Mol.Pharmacol_75_577 |
PubMedSearch : Marlo_2009_Mol.Pharmacol_75_577 |
PubMedID: 19047481 |
Title : Discovery of the first highly M5-preferring muscarinic acetylcholine receptor ligand, an M5 positive allosteric modulator derived from a series of 5-trifluoromethoxy N-benzyl isatins - Bridges_2009_J.Med.Chem_52_3445 |
Author(s) : Bridges TM , Marlo JE , Niswender CM , Jones CK , Jadhav SB , Gentry PR , Plumley HC , Weaver CD , Conn PJ , Lindsley CW |
Ref : Journal of Medicinal Chemistry , 52 :3445 , 2009 |
Abstract : Bridges_2009_J.Med.Chem_52_3445 |
ESTHER : Bridges_2009_J.Med.Chem_52_3445 |
PubMedSearch : Bridges_2009_J.Med.Chem_52_3445 |
PubMedID: 19438238 |