Title : Competitive activity-based protein profiling identifies aza-beta-lactams as a versatile chemotype for serine hydrolase inhibition - Zuhl_2012_J.Am.Chem.Soc_134_5068 |
Author(s) : Zuhl AM , Mohr JT , Bachovchin DA , Niessen S , Hsu KL , Berlin JM , Dochnahl M , Lopez-Alberca MP , Fu GC , Cravatt BF |
Ref : J Am Chem Soc , 134 :5068 , 2012 |
Abstract : |
PubMedSearch : Zuhl_2012_J.Am.Chem.Soc_134_5068 |
PubMedID: 22400490 |
Gene_locus related to this paper: human-ABHD10 |
Title : Academic cross-fertilization by public screening yields a remarkable class of protein phosphatase methylesterase-1 inhibitors - Bachovchin_2011_Proc.Natl.Acad.Sci.U.S.A_108_6811 |
Author(s) : Bachovchin DA , Mohr JT , Speers AE , Wang C , Berlin JM , Spicer TP , Fernandez-Vega V , Chase P , Hodder PS , Schurer SC , Nomura DK , Rosen H , Fu GC , Cravatt BF |
Ref : Proc Natl Acad Sci U S A , 108 :6811 , 2011 |
Abstract : |
PubMedSearch : Bachovchin_2011_Proc.Natl.Acad.Sci.U.S.A_108_6811 |
PubMedID: 21398589 |
Gene_locus related to this paper: human-PPME1 |
Title : Probe Development Efforts to Identify Novel Inhibitors of Protein Phosphatase Methylesterase-1 (PME-1) - Bachovchin_2010_Probe.Report__1 |
Author(s) : Bachovchin DA , Speers AE , Brown SJ , Spicer TP , Fernandez V , Ferguson J , Mohr JT , Murphy J , Fu GC , Cravatt BF , Hodder PS , Rosen H |
Ref : Probe Report , : , 2010 |
Abstract : |
PubMedSearch : Bachovchin_2010_Probe.Report__1 |
PubMedID: 22834039 |