Title : Chemical Proteomic Profiling of Human Methyltransferases - Horning_2016_J.Am.Chem.Soc_138_13335 |
Author(s) : Horning BD , Suciu RM , Ghadiri DA , Ulanovskaya OA , Matthews ML , Lum KM , Backus KM , Brown SJ , Rosen H , Cravatt BF |
Ref : Journal of the American Chemical Society , 138 :13335 , 2016 |
Abstract : |
PubMedSearch : Horning_2016_J.Am.Chem.Soc_138_13335 |
PubMedID: 27689866 |
Title : Characterization of a Selective, Reversible Inhibitor of Lysophospholipase 2 (LYPLA2) - Adibekian_2013_Probe.Report__4 |
Author(s) : Adibekian A , Martin BR , Chang JW , Hsu KL , Tsuboi K , Bachovchin DA , Speers AE , Brown SJ , Spicer T , Fernandez-Vega V , Ferguson J , Cravatt BF , Hodder P , Rosen H |
Ref : Probe Report , : , 2013 |
Abstract : |
PubMedSearch : Adibekian_2013_Probe.Report__4 |
PubMedID: 24624468 |
Gene_locus related to this paper: human-LYPLA2 |
Title : Characterization of a Selective, Reversible Inhibitor of Lysophospholipase 1 (LYPLA1) - Adibekian_2013_Probe.Report__3 |
Author(s) : Adibekian A , Martin BR , Chang JW , Hsu KL , Tsuboi K , Bachovchin DA , Speers AE , Brown SJ , Spicer T , Fernandez-Vega V , Ferguson J , Cravatt BF , Hodder P , Rosen H |
Ref : Probe Report , : , 2013 |
Abstract : |
PubMedSearch : Adibekian_2013_Probe.Report__3 |
PubMedID: 24624465 |
Title : Selective inhibitors and tailored activity probes for lipoprotein-associated phospholipase A(2) - Nagano_2013_Bioorg.Med.Chem.Lett_23_839 |
Author(s) : Nagano JM , Hsu KL , Whitby LR , Niphakis MJ , Speers AE , Brown SJ , Spicer T , Fernandez-Vega V , Ferguson J , Hodder P , Srinivasan P , Gonzalez TD , Rosen H , Bahnson BJ , Cravatt BF |
Ref : Bioorganic & Medicinal Chemistry Lett , 23 :839 , 2013 |
Abstract : |
PubMedSearch : Nagano_2013_Bioorg.Med.Chem.Lett_23_839 |
PubMedID: 23260346 |
Title : Optimization and characterization of a triazole urea inhibitor for diacylglycerol lipase beta (DAGL-beta) - Hsu_2012_Probe.Report__ |
Author(s) : Hsu KL , Tsuboi K , Speers AE , Brown SJ , Spicer T , Fernandez-Vega V , Ferguson J , Cravatt BF , Hodder P , Rosen H |
Ref : Probe Report , : , 2012 |
Abstract : |
PubMedSearch : Hsu_2012_Probe.Report__ |
PubMedID: 23658950 |
Gene_locus related to this paper: human-ABHD6 |
Title : Confirming target engagement for reversible inhibitors in vivo by kinetically tuned activity-based probes - Adibekian_2012_J.Am.Chem.Soc_134_10345 |
Author(s) : Adibekian A , Martin BR , Chang JW , Hsu KL , Tsuboi K , Bachovchin DA , Speers AE , Brown SJ , Spicer T , Fernandez-Vega V , Ferguson J , Hodder PS , Rosen H , Cravatt BF |
Ref : J Am Chem Soc , 134 :10345 , 2012 |
Abstract : |
PubMedSearch : Adibekian_2012_J.Am.Chem.Soc_134_10345 |
PubMedID: 22690931 |
Title : Optimization and characterization of a triazole urea inhibitor for alpha\/beta hydrolase domain-containing protein 11 (ABHD11): anti-probe for LYPLA1\/LYPLA2 dual inhibitor ML211 - Adibekian_2011_Probe.Report__1 |
Author(s) : Adibekian A , Hsu KL , Speers AE , Brown SJ , Spicer T , Fernandez-Vega V , Ferguson J , Cravatt BF , Hodder P , Rosen H |
Ref : Probe Report , : , 2011 |
Abstract : |
PubMedSearch : Adibekian_2011_Probe.Report__1 |
PubMedID: 23658953 |
Title : Optimization and characterization of a triazole urea dual inhibitor for lysophospholipase 1 (LYPLA1) and lysophospholipase 2 (LYPLA2) - Adibekian_2011_Probe.Report__5 |
Author(s) : Adibekian A , Martin BR , Speers AE , Brown SJ , Spicer T , Fernandez-Vega V , Ferguson J , Cravatt BF , Hodder P , Rosen H |
Ref : Probe Report , : , 2011 |
Abstract : |
PubMedSearch : Adibekian_2011_Probe.Report__5 |
PubMedID: 23658947 |
Title : Optimization and characterization of a triazole urea inhibitor for platelet-activating factor acetylhydrolase type 2 (PAFAH2) - Adibekian_2011_Probe.Report__2 |
Author(s) : Adibekian A , Hsu KL , Speers AE , Monillas ES , Brown SJ , Spicer T , Fernandez-Vega V , Ferguson J , Bahnson BJ , Cravatt BF , Hodder P , Rosen H |
Ref : Probe Report , : , 2011 |
Abstract : |
PubMedSearch : Adibekian_2011_Probe.Report__2 |
PubMedID: 23658960 |
Title : Probe Development Efforts to Identify Novel Inhibitors of Protein Phosphatase Methylesterase-1 (PME-1) - Bachovchin_2010_Probe.Report__1 |
Author(s) : Bachovchin DA , Speers AE , Brown SJ , Spicer TP , Fernandez V , Ferguson J , Mohr JT , Murphy J , Fu GC , Cravatt BF , Hodder PS , Rosen H |
Ref : Probe Report , : , 2010 |
Abstract : |
PubMedSearch : Bachovchin_2010_Probe.Report__1 |
PubMedID: 22834039 |
Title : Probe Report for PME-1 Inhibitors - Bachovchin_2010_Probe.Report__2 |
Author(s) : Bachovchin DA , Speers AE , Zuhl AM , Brown SJ , Cravatt BF , Fernandez V , Spicer T , Mercer BA , Ferguson J , Hodder P , Rosen HR |
Ref : Probe Report , : , 2010 |
Abstract : |
PubMedSearch : Bachovchin_2010_Probe.Report__2 |
PubMedID: 21433379 |
Title : Oxime esters as selective, covalent inhibitors of the serine hydrolase retinoblastoma-binding protein 9 (RBBP9) - Bachovchin_2010_Bioorg.Med.Chem.Lett_20_2254 |
Author(s) : Bachovchin DA , Wolfe MR , Masuda K , Brown SJ , Spicer TP , Fernandez-Vega V , Chase P , Hodder PS , Rosen H , Cravatt BF |
Ref : Bioorganic & Medicinal Chemistry Lett , 20 :2254 , 2010 |
Abstract : |
PubMedSearch : Bachovchin_2010_Bioorg.Med.Chem.Lett_20_2254 |
PubMedID: 20207142 |
Gene_locus related to this paper: human-RBBP9 |
Title : Probe Report for RBBP9 Inhibitors - Probe 2 - Bachovchin_2010_Probe.Report.1__ |
Author(s) : Bachovchin DA , Speers AE , Brown SJ , Cravatt BF , Spicer T , Mercer BA , Ferguson J , Hodder P , Rosen HR |
Ref : Probe Report , : , 2010 |
Abstract : |
PubMedSearch : Bachovchin_2010_Probe.Report.1__ |
PubMedID: 21433382 |
Gene_locus related to this paper: human-RBBP9 |
Title : Probe Report for RBBP9 Inhibitors - Probe 1 - Brown_2010_Probe.Report__ |
Author(s) : Brown SJ , Bachovchin DA , Cravatt BF , Fernandez-Vega V , Spicer T , Mercer BA , Hodder P , Rosen HR |
Ref : Probe Report , : , 2010 |
Abstract : |
PubMedSearch : Brown_2010_Probe.Report__ |
PubMedID: 21433353 |
Gene_locus related to this paper: human-RBBP9 |
Title : Identification of selective inhibitors of uncharacterized enzymes by high-throughput screening with fluorescent activity-based probes - Bachovchin_2009_Nat.Biotechnol_27_387 |
Author(s) : Bachovchin DA , Brown SJ , Rosen H , Cravatt BF |
Ref : Nat Biotechnol , 27 :387 , 2009 |
Abstract : |
PubMedSearch : Bachovchin_2009_Nat.Biotechnol_27_387 |
PubMedID: 19329999 |
Gene_locus related to this paper: human-ABHD11 |
Title : Striatal A2 receptor regulates apomorphine-induced turning in rats with unilateral dopamine denervation - Brown_1991_Psychopharmacology.(Berl)_103_78 |
Author(s) : Brown SJ , Gill R , Evenden JL , Iversen SD , Richardson PJ |
Ref : Psychopharmacology (Berl) , 103 :78 , 1991 |
Abstract : |
PubMedSearch : Brown_1991_Psychopharmacology.(Berl)_103_78 |
PubMedID: 1900945 |
Title : Both A1 and A2a purine receptors regulate striatal acetylcholine release - Brown_1990_J.Neurochem_55_31 |
Author(s) : Brown SJ , James S , Reddington M , Richardson PJ |
Ref : Journal of Neurochemistry , 55 :31 , 1990 |
Abstract : |
PubMedSearch : Brown_1990_J.Neurochem_55_31 |
PubMedID: 2355224 |
Title : Ectoenzymes control adenosine modulation of immunoisolated cholinergic synapses - Richardson_1987_Nature_327_232 |
Author(s) : Richardson PJ , Brown SJ , Bailyes EM , Luzio JP |
Ref : Nature , 327 :232 , 1987 |
Abstract : |
PubMedSearch : Richardson_1987_Nature_327_232 |
PubMedID: 3033519 |
Title : ATP release from affinity-purified rat cholinergic nerve terminals - Richardson_1987_J.Neurochem_48_622 |
Author(s) : Richardson PJ , Brown SJ |
Ref : Journal of Neurochemistry , 48 :622 , 1987 |
Abstract : |
PubMedSearch : Richardson_1987_J.Neurochem_48_622 |
PubMedID: 2432187 |