Title : Design and synthesis of cyanamides as potent and selective N-acylethanolamine acid amidase inhibitors - Malamas_2020_Bioorg.Med.Chem_28_115195 |
Author(s) : Malamas MS , Farah SI , Lamani M , Pelekoudas DN , Perry NT , Rajarshi G , Miyabe CY , Chandrashekhar H , West J , Pavlopoulos S , Makriyannis A |
Ref : Bioorganic & Medicinal Chemistry , 28 :115195 , 2020 |
Abstract : |
PubMedSearch : Malamas_2020_Bioorg.Med.Chem_28_115195 |
PubMedID: 31761726 |
Title : Effects of Distal Mutations on the Structure, Dynamics and Catalysis of Human Monoacylglycerol Lipase - Tyukhtenko_2018_Sci.Rep_8_1719 |
Author(s) : Tyukhtenko S , Rajarshi G , Karageorgos I , Zvonok N , Gallagher ES , Huang H , Vemuri K , Hudgens JW , Ma X , Nasr ML , Pavlopoulos S , Makriyannis A |
Ref : Sci Rep , 8 :1719 , 2018 |
Abstract : |
PubMedSearch : Tyukhtenko_2018_Sci.Rep_8_1719 |
PubMedID: 29379013 |
Gene_locus related to this paper: human-MGLL |
Title : Specific Inter-residue Interactions as Determinants of Human Monoacylglycerol Lipase Catalytic Competency: A ROLE FOR GLOBAL CONFORMATIONAL CHANGES - Tyukhtenko_2016_J.Biol.Chem_291_2556 |
Author(s) : Tyukhtenko S , Karageorgos I , Rajarshi G , Zvonok N , Pavlopoulos S , Janero DR , Makriyannis A |
Ref : Journal of Biological Chemistry , 291 :2556 , 2016 |
Abstract : |
PubMedSearch : Tyukhtenko_2016_J.Biol.Chem_291_2556 |
PubMedID: 26555264 |