| Title : Design and Synthesis of Highly Potent and Specific ABHD6 Inhibitors - Malamas_2021_ChemMedChem__ |
| Author(s) : Malamas MS , Lamani M , Farah SI , Mohammad KA , Miyabe CY , Rajarshi G , Wu S , Zvonok N , Chandrashekhar H , Wood J , Makriyannis A |
| Ref : ChemMedChem , : , 2021 |
| Abstract : |
| PubMedSearch : Malamas_2021_ChemMedChem__ |
| PubMedID: 34486233 |
| Gene_locus related to this paper: human-ABHD6 , mouse-ABHD6 |
| Title : Design and synthesis of cyanamides as potent and selective N-acylethanolamine acid amidase inhibitors - Malamas_2020_Bioorg.Med.Chem_28_115195 |
| Author(s) : Malamas MS , Farah SI , Lamani M , Pelekoudas DN , Perry NT , Rajarshi G , Miyabe CY , Chandrashekhar H , West J , Pavlopoulos S , Makriyannis A |
| Ref : Bioorganic & Medicinal Chemistry , 28 :115195 , 2020 |
| Abstract : |
| PubMedSearch : Malamas_2020_Bioorg.Med.Chem_28_115195 |
| PubMedID: 31761726 |
| Title : Conformational gating, dynamics and allostery in human monoacylglycerol lipase - Tyukhtenko_2020_Sci.Rep_10_18531 |
| Author(s) : Tyukhtenko S , Ma X , Rajarshi G , Karageorgos I , Anderson KW , Hudgens JW , Guo JJ , Nasr ML , Zvonok N , Vemuri K , Wagner G , Makriyannis A |
| Ref : Sci Rep , 10 :18531 , 2020 |
| Abstract : |
| PubMedSearch : Tyukhtenko_2020_Sci.Rep_10_18531 |
| PubMedID: 33116203 |
| Gene_locus related to this paper: human-MGLL |
| Title : Synthesis and evaluation of potent and selective MGL inhibitors as a glaucoma treatment - Alapafuja_2019_Bioorg.Med.Chem_27_55 |
| Author(s) : Alapafuja SO , Malamas MS , Shukla V , Zvonok A , Miller S , Daily L , Rajarshi G , Miyabe CY , Chandrashekhar H , Wood J , Tyukhtenko S , Straiker A , Makriyannis A |
| Ref : Bioorganic & Medicinal Chemistry , 27 :55 , 2019 |
| Abstract : |
| PubMedSearch : Alapafuja_2019_Bioorg.Med.Chem_27_55 |
| PubMedID: 30446439 |
| Title : Effects of Distal Mutations on the Structure, Dynamics and Catalysis of Human Monoacylglycerol Lipase - Tyukhtenko_2018_Sci.Rep_8_1719 |
| Author(s) : Tyukhtenko S , Rajarshi G , Karageorgos I , Zvonok N , Gallagher ES , Huang H , Vemuri K , Hudgens JW , Ma X , Nasr ML , Pavlopoulos S , Makriyannis A |
| Ref : Sci Rep , 8 :1719 , 2018 |
| Abstract : |
| PubMedSearch : Tyukhtenko_2018_Sci.Rep_8_1719 |
| PubMedID: 29379013 |
| Gene_locus related to this paper: human-MGLL |
| Title : Specific Inter-residue Interactions as Determinants of Human Monoacylglycerol Lipase Catalytic Competency: A ROLE FOR GLOBAL CONFORMATIONAL CHANGES - Tyukhtenko_2016_J.Biol.Chem_291_2556 |
| Author(s) : Tyukhtenko S , Karageorgos I , Rajarshi G , Zvonok N , Pavlopoulos S , Janero DR , Makriyannis A |
| Ref : Journal of Biological Chemistry , 291 :2556 , 2016 |
| Abstract : |
| PubMedSearch : Tyukhtenko_2016_J.Biol.Chem_291_2556 |
| PubMedID: 26555264 |