Title : A thiocarbamate inhibitor of endothelial lipase raises HDL cholesterol levels in mice - Greco_2013_Bioorg.Med.Chem.Lett_23_2595 |
Author(s) : Greco MN , Connelly MA , Leo GC , Olson MW , Powell E , Huang Z , Hawkins M , Smith C , Schalk-Hihi C , Darrow AL , Xin H , Lang W , Damiano BP , Hlasta DJ |
Ref : Bioorganic & Medicinal Chemistry Lett , 23 :2595 , 2013 |
Abstract : |
PubMedSearch : Greco_2013_Bioorg.Med.Chem.Lett_23_2595 |
PubMedID: 23528297 |
Title : Screening and characterization of human monoglyceride lipase active site inhibitors using orthogonal binding and functional assays - Clemente_2012_J.Biomol.Screen_17_629 |
Author(s) : Clemente JC , Nulton E , Nelen M , Todd MJ , Maguire D , Schalk-Hihi C , Kuo LC , Zhang SP , Flores CM , Kranz JK |
Ref : J Biomol Screen , 17 :629 , 2012 |
Abstract : |
PubMedSearch : Clemente_2012_J.Biomol.Screen_17_629 |
PubMedID: 22496098 |
Title : A novel fluorogenic substrate for the measurement of endothelial lipase activity - Darrow_2011_J.Lipid.Res_52_374 |
Author(s) : Darrow AL , Olson MW , Xin H , Burke SL , Smith C , Schalk-Hihi C , Williams R , Bayoumy SS , Deckman IC , Todd MJ , Damiano BP , Connelly MA |
Ref : J Lipid Res , 52 :374 , 2011 |
Abstract : |
PubMedSearch : Darrow_2011_J.Lipid.Res_52_374 |
PubMedID: 21062953 |
Gene_locus related to this paper: human-LIPG |
Title : Crystal structure of a soluble form of human monoglyceride lipase in complex with an inhibitor at 1.35 A resolution - Schalk-Hihi_2011_Protein.Sci_20_670 |
Author(s) : Schalk-Hihi C , Schubert C , Alexander R , Bayoumy S , Clemente JC , Deckman I , Desjarlais RL , Dzordzorme KC , Flores CM , Grasberger B , Kranz JK , Lewandowski F , Liu L , Ma H , Maguire D , Macielag MJ , McDonnell ME , Mezzasalma Haarlander T , Miller R , Milligan C , Reynolds C , Kuo LC |
Ref : Protein Science , 20 :670 , 2011 |
Abstract : |
PubMedSearch : Schalk-Hihi_2011_Protein.Sci_20_670 |
PubMedID: 21308848 |
Gene_locus related to this paper: human-MGLL |