Title : Poster: Stereoselective interaction of trihexyphenidyl and related compounds with muscarinic receptors - |
Author(s) : Gross J , Pfaff O , Rachel D , Tacke R , Leis A , Ruhlmann K , Waelbroeck M , Mutschler E , Lambrecht G |
Ref : Life Sciences , 64 :593 , 1999 |
PubMedID: |
Title : Binding and functional properties of hexocyclium and sila-hexocyclium derivatives to muscarinic receptor subtypes - Waelbroeck_1994_Br.J.Pharmacol_112_505 |
Author(s) : Waelbroeck M , Camus J , Tastenoy M , Feifel R , Mutschler E , Tacke R , Strohmann C , Rafeiner K , Rodrigues de Miranda JF , Lambrecht G |
Ref : British Journal of Pharmacology , 112 :505 , 1994 |
Abstract : |
PubMedSearch : Waelbroeck_1994_Br.J.Pharmacol_112_505 |
PubMedID: 8075869 |
Title : Characterization of muscarinic receptors mediating vasodilation in rat perfused kidney - Eltze_1993_Eur.J.Pharmacol_238_343 |
Author(s) : Eltze M , Ullrich B , Mutschler E , Moser U , Bungardt E , Friebe T , Gubitz C , Tacke R , Lambrecht G |
Ref : European Journal of Pharmacology , 238 :343 , 1993 |
Abstract : |
PubMedSearch : Eltze_1993_Eur.J.Pharmacol_238_343 |
PubMedID: 8405103 |
Title : Thermodynamics of antagonist binding to rat muscarinic M2 receptors: antimuscarinics of the pridinol, sila-pridinol, diphenidol and sila-diphenidol type - Waelbroeck_1993_Br.J.Pharmacol_109_360 |
Author(s) : Waelbroeck M , Camus J , Tastenoy M , Lambrecht G , Mutschler E , Kropfgans M , Sperlich J , Wiesenberger F , Tacke R , Christophe J |
Ref : British Journal of Pharmacology , 109 :360 , 1993 |
Abstract : |
PubMedSearch : Waelbroeck_1993_Br.J.Pharmacol_109_360 |
PubMedID: 8102927 |
Title : Poster: Functional characterization of muscarinic receptors in rabbit peripheral lung - |
Author(s) : Vockert E , Egerer HP , Tacke R , Lambrecht G , Mutschler E |
Ref : Life Sciences , 52(5-6) :551 , 1993 |
PubMedID: |
Title : Poster: Characterization of the vasodilatory muscarinic receptor in perfused rat kidney by the use of agonists and antagonists - |
Author(s) : Eltze M , Mutschler E , Moser U , Friebe T , Gubitz C , Tacke R , Lambrecht G |
Ref : Life Sciences , 52(5-6) :579 , 1993 |
PubMedID: |
Title : Stereoselective interaction of procyclidine, hexahydro-difenidol, hexbutinol and oxyphencyclimine, and of related antagonists, with four muscarinic receptors - Waelbroeck_1992_Eur.J.Pharmacol_227_33 |
Author(s) : Waelbroeck M , Camus J , Tastenoy M , Mutschler E , Strohmann C , Tacke R , Schjelderup L , Aasen A , Lambrecht G , Christophe J |
Ref : European Journal of Pharmacology , 227 :33 , 1992 |
Abstract : |
PubMedSearch : Waelbroeck_1992_Eur.J.Pharmacol_227_33 |
PubMedID: 1426023 |
Title : Characterization of muscarinic receptors mediating vasodilation in guinea-pig ileum submucosal arterioles by the use of computer-assisted videomicroscopy - Bungardt_1992_Eur.J.Pharmacol_213_53 |
Author(s) : Bungardt E , Vockert E , Feifel R , Moser U , Tacke R , Mutschler E , Lambrecht G , Surprenant A |
Ref : European Journal of Pharmacology , 213 :53 , 1992 |
Abstract : |
PubMedSearch : Bungardt_1992_Eur.J.Pharmacol_213_53 |
PubMedID: 1499657 |
Title : Binding affinities of hexahydro-difenidol and hexahydro-sila-difenidol analogues at four muscarinic receptor subtypes: constitutional and stereochemical aspects - Waelbroeck_1991_Eur.J.Pharmacol_206_95 |
Author(s) : Waelbroeck M , Camus J , Tastenoy M , Mutschler E , Strohmann C , Tacke R , Lambrecht G , Christophe J |
Ref : European Journal of Pharmacology , 206 :95 , 1991 |
Abstract : |
PubMedSearch : Waelbroeck_1991_Eur.J.Pharmacol_206_95 |
PubMedID: 2065719 |
Title : Stereoselectivity of (R)- and (S)-hexahydro-difenidol binding to neuroblastoma M1, cardiac M2, pancreatic M3, and striatum M4 muscarinic receptors - Waelbroeck_1991_Chirality_3_118 |
Author(s) : Waelbroeck M , Camus J , Tastenoy M , Mutschler E , Strohmann C , Tacke R , Lambrecht G , Christophe J |
Ref : Chirality , 3 :118 , 1991 |
Abstract : |
PubMedSearch : Waelbroeck_1991_Chirality_3_118 |
PubMedID: 1863523 |
Title : Selective labelling of muscarinic M1 receptors in calf superior cervical ganglia by [3H](+\/-)-telenzepine - Feifel_1991_Eur.J.Pharmacol_195_115 |
Author(s) : Feifel R , Rodrigues de Miranda JF , Strohmann C , Tacke R , Aasen AJ , Mutschler E , Lambrecht G |
Ref : European Journal of Pharmacology , 195 :115 , 1991 |
Abstract : |
PubMedSearch : Feifel_1991_Eur.J.Pharmacol_195_115 |
PubMedID: 2065706 |
Title : Pharmacological characterization of the vascular muscarinic receptors mediating relaxation and contraction in rabbit aorta - Jaiswal_1991_J.Pharmacol.Exp.Ther_258_842 |
Author(s) : Jaiswal N , Lambrecht G , Mutschler E , Tacke R , Malik KU |
Ref : Journal of Pharmacology & Experimental Therapeutics , 258 :842 , 1991 |
Abstract : |
PubMedSearch : Jaiswal_1991_J.Pharmacol.Exp.Ther_258_842 |
PubMedID: 1716312 |
Title : Antagonist binding profiles of five cloned human muscarinic receptor subtypes - Dorje_1991_J.Pharmacol.Exp.Ther_256_727 |
Author(s) : Dorje F , Wess J , Lambrecht G , Tacke R , Mutschler E , Brann MR |
Ref : Journal of Pharmacology & Experimental Therapeutics , 256 :727 , 1991 |
Abstract : |
PubMedSearch : Dorje_1991_J.Pharmacol.Exp.Ther_256_727 |
PubMedID: 1994002 |
Title : Human gastric mucosa expresses glandular M3 subtype of muscarinic receptors - Pfeiffer_1990_Dig.Dis.Sci_35_1468 |
Author(s) : Pfeiffer A , Hanack C , Kopp R , Tacke R , Moser U , Mutschler E , Lambrecht G , Herawi M |
Ref : Digestive Diseases & Sciences , 35 :1468 , 1990 |
Abstract : |
PubMedSearch : Pfeiffer_1990_Dig.Dis.Sci_35_1468 |
PubMedID: 2253531 |
Title : Muscarinic receptor subtypes in rat pancreatic islets: binding and functional studies - Verspohl_1990_Eur.J.Pharmacol_178_303 |
Author(s) : Verspohl EJ , Tacke R , Mutschler E , Lambrecht G |
Ref : European Journal of Pharmacology , 178 :303 , 1990 |
Abstract : |
PubMedSearch : Verspohl_1990_Eur.J.Pharmacol_178_303 |
PubMedID: 2187704 |
Title : Muscarinic receptors mediating acid secretion in isolated rat gastric parietal cells are of M3 type - Pfeiffer_1990_Gastroenterology_98_218 |
Author(s) : Pfeiffer A , Rochlitz H , Noelke B , Tacke R , Moser U , Mutschler E , Lambrecht G |
Ref : Gastroenterology , 98 :218 , 1990 |
Abstract : |
PubMedSearch : Pfeiffer_1990_Gastroenterology_98_218 |
PubMedID: 2293581 |
Title : Selective antagonists provide evidence that M1 muscarinic receptors may mediate carbachol-induced drinking in the rat - Polidori_1990_Eur.J.Pharmacol_179_159 |
Author(s) : Polidori C , Massi M , Lambrecht G , Mutschler E , Tacke R , Melchiorre C |
Ref : European Journal of Pharmacology , 179 :159 , 1990 |
Abstract : |
PubMedSearch : Polidori_1990_Eur.J.Pharmacol_179_159 |
PubMedID: 2364977 |
Title : Stereoselectivity of procyclidine binding to muscarinic receptor subtypes M1, M2 and M4 - Waelbroeck_1990_Eur.J.Pharmacol_189_135 |
Author(s) : Waelbroeck M , Camus J , Tastenoy M , Lambrecht G , Mutschler E , Tacke R , Christophe J |
Ref : European Journal of Pharmacology , 189 :135 , 1990 |
Abstract : |
PubMedSearch : Waelbroeck_1990_Eur.J.Pharmacol_189_135 |
PubMedID: 2253700 |
Title : Stereoselective inhibition of muscarinic receptor subtypes by the enantiomers of hexahydro-difenidol and acetylenic analogues - Feifel_1990_Br.J.Pharmacol_99_455 |
Author(s) : Feifel R , Wagner-Roder M , Strohmann C , Tacke R , Waelbroeck M , Christophe J , Mutschler E , Lambrecht G |
Ref : British Journal of Pharmacology , 99 :455 , 1990 |
Abstract : |
PubMedSearch : Feifel_1990_Br.J.Pharmacol_99_455 |
PubMedID: 2331578 |
Title : Pharmacokinetic properties of the antimuscarinic drug [3H]-hexahydro-sila-difenidol in the rat - Rettenmayr_1990_Naunyn.Schmiedebergs.Arch.Pharmacol_342_146 |
Author(s) : Rettenmayr NM , Rodrigues de Miranda JF , Rijntjes NV , Russel FG , van Ginneken CA , Strohmann C , Tacke R , Lambrecht G , Mutschler E |
Ref : Naunyn Schmiedebergs Arch Pharmacol , 342 :146 , 1990 |
Abstract : |
PubMedSearch : Rettenmayr_1990_Naunyn.Schmiedebergs.Arch.Pharmacol_342_146 |
PubMedID: 2234099 |
Title : Novel pharmacological profile of muscarinic receptors mediating contraction of the guinea-pig uterus - Dorje_1990_Naunyn.Schmiedebergs.Arch.Pharmacol_342_284 |
Author(s) : Dorje F , Friebe T , Tacke R , Mutschler E , Lambrecht G |
Ref : Naunyn Schmiedebergs Arch Pharmacol , 342 :284 , 1990 |
Abstract : |
PubMedSearch : Dorje_1990_Naunyn.Schmiedebergs.Arch.Pharmacol_342_284 |
PubMedID: 2280796 |
Title : Poster: [3H]-(+\/-}-Telenzepine selectively labels muscarinic M1-receptors in calf superior cervical ganglia - |
Author(s) : Feifel R , Rodrigues de Miranda JF , Strohmann C , Tacke R , Lambrecht G , Mutschler E |
Ref : Trends in Pharmacological Sciences , Suppl :110 , 1989 |
PubMedID: |
Title : Human HT-29 colon carcinoma cells contain muscarinic M3 receptors coupled to phosphoinositide metabolism - Kopp_1989_Eur.J.Pharmacol_172_397 |
Author(s) : Kopp R , Lambrecht G , Mutschler E , Moser U , Tacke R , Pfeiffer A |
Ref : European Journal of Pharmacology , 172 :397 , 1989 |
Abstract : |
PubMedSearch : Kopp_1989_Eur.J.Pharmacol_172_397 |
PubMedID: 2555210 |
Title : Pharmacology of hexahydro-difenidol, hexahydro-sila-difenidol and related selective muscarinic antagonists - Lambrecht_1989_Trends.Pharmacol.Sci_Suppl_60 |
Author(s) : Lambrecht G , Feifel R , Moser U , Wagner-Roder M , Choo LK , Camus J , Tastenoy M , Waelbroeck M , Strohmann C , Tacke R |
Ref : Trends in Pharmacological Sciences , Suppl :60 , 1989 |
Abstract : |
PubMedSearch : Lambrecht_1989_Trends.Pharmacol.Sci_Suppl_60 |
PubMedID: 2694525 |
Title : Poster: Antimuscarinic potencies of olefinic analogues related to hexahydro-difenidol at three muscarinic receptor subtypes - |
Author(s) : Choo LK , Wagner M , Unterhalt B , Middelberg C , Tacke R , Strohmann C , Tafel A , Mutschler E , Lambrecht G |
Ref : Trends in Pharmacological Sciences , Suppl :113 , 1989 |
PubMedID: |
Title : Poster: Pharmacophore model for antimuscarinic agents related to difenidol and siladifenidol - a molecular modeling study - |
Author(s) : Bruggmann J , Holtje HD , Mutschler E , Lambrecht G , Tacke R |
Ref : Trends in Pharmacological Sciences , Suppl :114 , 1989 |
PubMedID: |
Title : Binding and functional properties of antimuscarinics of the hexocyclium\/sila-hexocyclium and hexahydro-diphenidol\/hexahydro-sila-diphenidol type to muscarinic receptor subtypes - Waelbroeck_1989_Br.J.Pharmacol_98_197 |
Author(s) : Waelbroeck M , Tastenoy M , Camus J , Christophe J , Strohmann C , Linoh H , Zilch H , Tacke R , Mutschler E , Lambrecht G |
Ref : British Journal of Pharmacology , 98 :197 , 1989 |
Abstract : |
PubMedSearch : Waelbroeck_1989_Br.J.Pharmacol_98_197 |
PubMedID: 2804545 |
Title : Affinity profiles of hexahydro-sila-difenidol analogues at muscarinic receptor subtypes - Lambrecht_1989_Eur.J.Pharmacol_168_71 |
Author(s) : Lambrecht G , Feifel R , Wagner-Roder M , Strohmann C , Zilch H , Tacke R , Waelbroeck M , Christophe J , Boddeke HW , Mutschler E |
Ref : European Journal of Pharmacology , 168 :71 , 1989 |
Abstract : |
PubMedSearch : Lambrecht_1989_Eur.J.Pharmacol_168_71 |
PubMedID: 2583233 |
Title : Different muscarine receptors mediate the prejunctional inhibition of [3H]-noradrenaline release in rat or guinea-pig iris and the contraction of the rabbit iris sphincter muscle - Fuder_1989_Naunyn.Schmiedebergs.Arch.Pharmacol_340_597 |
Author(s) : Fuder H , Schopf J , Unckell J , Wesner MT , Melchiorre C , Tacke R , Mutschler E , Lambrecht G |
Ref : Naunyn Schmiedebergs Arch Pharmacol , 340 :597 , 1989 |
Abstract : |
PubMedSearch : Fuder_1989_Naunyn.Schmiedebergs.Arch.Pharmacol_340_597 |
PubMedID: 2615852 |
Title : Stereoselectivity of the interaction of muscarinic antagonists with their receptors - Waelbroeck_1989_Trends.Pharmacol.Sci_Suppl_65 |
Author(s) : Waelbroeck M , Tastenoy M , Camus J , Feifel R , Mutschler E , Strohmann C , Tacke R , Lambrecht G , Christophe J |
Ref : Trends in Pharmacological Sciences , Suppl :65 , 1989 |
Abstract : |
PubMedSearch : Waelbroeck_1989_Trends.Pharmacol.Sci_Suppl_65 |
PubMedID: 2694526 |
Title : Poster: High affinity pirenzepine receptors in chicken atria are different from Ml type - |
Author(s) : Tietz H , Lindmar R , Loffelholz K , Strohmann C , Tacke R , Lambrecht G , Mutschler E |
Ref : Trends in Pharmacological Sciences , Suppl :107 , 1989 |
PubMedID: |
Title : Presynaptic muscarinic receptors mediating inhibition of neurogenic contractions in rabbit vas deferens are of the ganglionic M1-type - Eltz_1988_Eur.J.Pharmacol_158_233 |
Author(s) : Eltz M , Gmelin G , Wess J , Strohmann C , Tacke R , Mutschler E , Lambrecht G |
Ref : European Journal of Pharmacology , 158 :233 , 1988 |
Abstract : |
PubMedSearch : Eltz_1988_Eur.J.Pharmacol_158_233 |
PubMedID: 2472963 |
Title : p-fluoro-hexahydro-sila-difenidol: the first M2 beta-selective muscarinic antagonist - |
Author(s) : Lambrecht G , Feifel R , Forth B , Strohmann C , Tacke R , Mutschler E |
Ref : European Journal of Pharmacology , 152 :193 , 1988 |
PubMedID: 3208832 |
Title : o-Methoxy-sila-hexocyclium: a new quaternary M1-selective muscarinic antagonist - |
Author(s) : Lambrecht G , Gmelin G , Rafeiner K , Strohmann C , Tacke R , Mutschler E |
Ref : European Journal of Pharmacology , 151 :155 , 1988 |
PubMedID: 3416923 |
Title : Poster: Hexahydrosiladifenidol: a selective antagonist at muscarinic M2 receptor subtypes - |
Author(s) : Lambrecht G , Moser U , Wess J , Riotte J , Fuder H , Kilbinger H , Milller H , Linoh H , Tacke R , Zilch H , Mutschler E |
Ref : Trends in Pharmacological Sciences , Suppl :91 , 1986 |
PubMedID: |