Christophe J

References (42)

Title : New functionally selective muscarinic agonists - Lambrecht_1993_Life.Sci_52(5-6)_481
Author(s) : Lambrecht G , Moser U , Grimm U , Pfaff O , Hermanni U , Hildebrandt C , Waelbroeck M , Christophe J , Mutschler E
Ref : Life Sciences , 52 :481 , 1993
Abstract :
PubMedSearch : Lambrecht_1993_Life.Sci_52(5-6)_481
PubMedID: 7680092

Title : Thermodynamics of antagonist binding to rat muscarinic M2 receptors: antimuscarinics of the pridinol, sila-pridinol, diphenidol and sila-diphenidol type - Waelbroeck_1993_Br.J.Pharmacol_109_360
Author(s) : Waelbroeck M , Camus J , Tastenoy M , Lambrecht G , Mutschler E , Kropfgans M , Sperlich J , Wiesenberger F , Tacke R , Christophe J
Ref : British Journal of Pharmacology , 109 :360 , 1993
Abstract :
PubMedSearch : Waelbroeck_1993_Br.J.Pharmacol_109_360
PubMedID: 8102927

Title : Poster: Binding to an allosteric site on muscarinic receptors -
Author(s) : Waelbroeck M , Camus J , Christophe J
Ref : Life Sciences , 52(5-6) :576 , 1993
PubMedID:

Title : Binding properties of nine 4-diphenyl-acetoxy-N-methyl-piperidine (4-DAMP) analogues to M1, M2, M3 and putative M4 muscarinic receptor subtypes - Waelbroeck_1992_Br.J.Pharmacol_105_97
Author(s) : Waelbroeck M , Camus J , Tastenoy M , Christophe J
Ref : British Journal of Pharmacology , 105 :97 , 1992
Abstract :
PubMedSearch : Waelbroeck_1992_Br.J.Pharmacol_105_97
PubMedID: 1596694

Title : Stereoselective interaction of procyclidine, hexahydro-difenidol, hexbutinol and oxyphencyclimine, and of related antagonists, with four muscarinic receptors - Waelbroeck_1992_Eur.J.Pharmacol_227_33
Author(s) : Waelbroeck M , Camus J , Tastenoy M , Mutschler E , Strohmann C , Tacke R , Schjelderup L , Aasen A , Lambrecht G , Christophe J
Ref : European Journal of Pharmacology , 227 :33 , 1992
Abstract :
PubMedSearch : Waelbroeck_1992_Eur.J.Pharmacol_227_33
PubMedID: 1426023

Title : Inactivation of brain cortex muscarinic receptors by 4-diphenylacetoxy-1-(2-chloroethyl) piperidine mustard - Waelbroeck_1992_Biochem.Pharmacol_44_285
Author(s) : Waelbroeck M , Renzetti AR , Tastenoy M , Barlow RB , Christophe J
Ref : Biochemical Pharmacology , 44 :285 , 1992
Abstract :
PubMedSearch : Waelbroeck_1992_Biochem.Pharmacol_44_285
PubMedID: 1642642

Title : Binding affinities of hexahydro-difenidol and hexahydro-sila-difenidol analogues at four muscarinic receptor subtypes: constitutional and stereochemical aspects - Waelbroeck_1991_Eur.J.Pharmacol_206_95
Author(s) : Waelbroeck M , Camus J , Tastenoy M , Mutschler E , Strohmann C , Tacke R , Lambrecht G , Christophe J
Ref : European Journal of Pharmacology , 206 :95 , 1991
Abstract :
PubMedSearch : Waelbroeck_1991_Eur.J.Pharmacol_206_95
PubMedID: 2065719

Title : Stereoselectivity of (R)- and (S)-hexahydro-difenidol binding to neuroblastoma M1, cardiac M2, pancreatic M3, and striatum M4 muscarinic receptors - Waelbroeck_1991_Chirality_3_118
Author(s) : Waelbroeck M , Camus J , Tastenoy M , Mutschler E , Strohmann C , Tacke R , Lambrecht G , Christophe J
Ref : Chirality , 3 :118 , 1991
Abstract :
PubMedSearch : Waelbroeck_1991_Chirality_3_118
PubMedID: 1863523

Title : Binding kinetics of quinuclidinyl benzilate and methyl-quinuclidinyl benzilate enantiomers at neuronal (M1), cardiac (M2), and pancreatic (M3) muscarinic receptors - Waelbroeck_1991_Mol.Pharmacol_40_413
Author(s) : Waelbroeck M , Tastenoy M , Camus J , Christophe J
Ref : Molecular Pharmacology , 40 :413 , 1991
Abstract :
PubMedSearch : Waelbroeck_1991_Mol.Pharmacol_40_413
PubMedID: 1896027

Title : Stereoselectivity of procyclidine binding to muscarinic receptor subtypes M1, M2 and M4 - Waelbroeck_1990_Eur.J.Pharmacol_189_135
Author(s) : Waelbroeck M , Camus J , Tastenoy M , Lambrecht G , Mutschler E , Tacke R , Christophe J
Ref : European Journal of Pharmacology , 189 :135 , 1990
Abstract :
PubMedSearch : Waelbroeck_1990_Eur.J.Pharmacol_189_135
PubMedID: 2253700

Title : Stereoselective inhibition of muscarinic receptor subtypes by the enantiomers of hexahydro-difenidol and acetylenic analogues - Feifel_1990_Br.J.Pharmacol_99_455
Author(s) : Feifel R , Wagner-Roder M , Strohmann C , Tacke R , Waelbroeck M , Christophe J , Mutschler E , Lambrecht G
Ref : British Journal of Pharmacology , 99 :455 , 1990
Abstract :
PubMedSearch : Feifel_1990_Br.J.Pharmacol_99_455
PubMedID: 2331578

Title : Binding of selective antagonists to four muscarinic receptors (M1 to M4) in rat forebrain - Waelbroeck_1990_Mol.Pharmacol_38_267
Author(s) : Waelbroeck M , Tastenoy M , Camus J , Christophe J
Ref : Molecular Pharmacology , 38 :267 , 1990
Abstract :
PubMedSearch : Waelbroeck_1990_Mol.Pharmacol_38_267
PubMedID: 2385234

Title : Bretylium tosylate binds preferentially to muscarinic receptors labelled with [3H]oxotremorine M (SH or 'high affinity' receptors) in rat heart and brain cortex - Gillard_1989_Eur.J.Pharmacol_160_117
Author(s) : Gillard M , Brunner F , Waelbroeck M , Svoboda M , Christophe J
Ref : European Journal of Pharmacology , 160 :117 , 1989
Abstract :
PubMedSearch : Gillard_1989_Eur.J.Pharmacol_160_117
PubMedID: 2714357

Title : Determination of the association and dissociation rate constants of muscarinic antagonists on rat pancreas: rank order of potency varies with time - Waelbroeck_1989_Mol.Pharmacol_36_405
Author(s) : Waelbroeck M , Camus J , Christophe J
Ref : Molecular Pharmacology , 36 :405 , 1989
Abstract :
PubMedSearch : Waelbroeck_1989_Mol.Pharmacol_36_405
PubMedID: 2779525

Title : Binding and functional properties of antimuscarinics of the hexocyclium\/sila-hexocyclium and hexahydro-diphenidol\/hexahydro-sila-diphenidol type to muscarinic receptor subtypes - Waelbroeck_1989_Br.J.Pharmacol_98_197
Author(s) : Waelbroeck M , Tastenoy M , Camus J , Christophe J , Strohmann C , Linoh H , Zilch H , Tacke R , Mutschler E , Lambrecht G
Ref : British Journal of Pharmacology , 98 :197 , 1989
Abstract :
PubMedSearch : Waelbroeck_1989_Br.J.Pharmacol_98_197
PubMedID: 2804545

Title : Affinity profiles of hexahydro-sila-difenidol analogues at muscarinic receptor subtypes - Lambrecht_1989_Eur.J.Pharmacol_168_71
Author(s) : Lambrecht G , Feifel R , Wagner-Roder M , Strohmann C , Zilch H , Tacke R , Waelbroeck M , Christophe J , Boddeke HW , Mutschler E
Ref : European Journal of Pharmacology , 168 :71 , 1989
Abstract :
PubMedSearch : Lambrecht_1989_Eur.J.Pharmacol_168_71
PubMedID: 2583233

Title : Stereoselectivity of the interaction of muscarinic antagonists with their receptors - Waelbroeck_1989_Trends.Pharmacol.Sci_Suppl_65
Author(s) : Waelbroeck M , Tastenoy M , Camus J , Feifel R , Mutschler E , Strohmann C , Tacke R , Lambrecht G , Christophe J
Ref : Trends in Pharmacological Sciences , Suppl :65 , 1989
Abstract :
PubMedSearch : Waelbroeck_1989_Trends.Pharmacol.Sci_Suppl_65
PubMedID: 2694526

Title : 80\% of muscarinic receptors expressed by the NB-OK 1 human neuroblastoma cell line show high affinity for pirenzepine and are comparable to rat hippocampus M1 receptors - Waelbroeck_1988_FEBS.Lett_226_287
Author(s) : Waelbroeck M , Camus J , Tastenoy M , Christophe J
Ref : FEBS Letters , 226 :287 , 1988
Abstract :
PubMedSearch : Waelbroeck_1988_FEBS.Lett_226_287
PubMedID: 3338559

Title : Characterization of muscarinic receptors in human pancreatic membranes - Waelbroeck_1988_Pancreas_3_627
Author(s) : Waelbroeck M , Camus J , Tastenoy M , de Neef P , Scemama JL , Fourmy D , Vaysse N , Pradayrol L , Robberecht P , Christophe J
Ref : Pancreas , 3 :627 , 1988
Abstract :
PubMedSearch : Waelbroeck_1988_Pancreas_3_627
PubMedID: 3222245

Title : Effects of d-tubocurarine on rat cardiac muscarinic receptors: a comparison with gallamine - Waelbroeck_1988_J.Recept.Res_8_787
Author(s) : Waelbroeck M , Robberecht P , de Neef P , Christophe J
Ref : J Recept Res , 8 :787 , 1988
Abstract :
PubMedSearch : Waelbroeck_1988_J.Recept.Res_8_787
PubMedID: 3193402

Title : Stereoselectivity of the enantiomers of trihexyphenidyl and its methiodide at muscarinic receptor subtypes - Lambrecht_1988_Eur.J.Pharmacol_155_167
Author(s) : Lambrecht G , Feifel R , Moser U , Aasen AJ , Waelbroeck M , Christophe J , Mutschler E
Ref : European Journal of Pharmacology , 155 :167 , 1988
Abstract :
PubMedSearch : Lambrecht_1988_Eur.J.Pharmacol_155_167
PubMedID: 3243330

Title : Functional characterization of muscarinic receptors in rat parotid acini - Dehaye_1988_Eur.J.Pharmacol_151_427
Author(s) : Dehaye JP , Marino A , Soukias Y , Poloczek P , Winand J , Christophe J
Ref : European Journal of Pharmacology , 151 :427 , 1988
Abstract :
PubMedSearch : Dehaye_1988_Eur.J.Pharmacol_151_427
PubMedID: 2463925

Title : Muscarinic receptor heterogeneity in rat central nervous system. II. Brain receptors labeled by [3H]oxotremorine-M correspond to heterogeneous M2 receptors with very high affinity for agonists - Gillard_1987_Mol.Pharmacol_32_100
Author(s) : Gillard M , Waelbroeck M , Christophe J
Ref : Molecular Pharmacology , 32 :100 , 1987
Abstract :
PubMedSearch : Gillard_1987_Mol.Pharmacol_32_100
PubMedID: 3600611

Title : Different antagonist binding properties of rat pancreatic and cardiac muscarinic receptors - Waelbroeck_1987_Life.Sci_41_2235
Author(s) : Waelbroeck M , Camus J , Winand J , Christophe J
Ref : Life Sciences , 41 :2235 , 1987
Abstract :
PubMedSearch : Waelbroeck_1987_Life.Sci_41_2235
PubMedID: 3118122

Title : Muscarinic receptor heterogeneity in rat central nervous system. I. Binding of four selective antagonists to three muscarinic receptor subclasses: a comparison with M2 cardiac muscarinic receptors of the C type - Waelbroeck_1987_Mol.Pharmacol_32_91
Author(s) : Waelbroeck M , Gillard M , Robberecht P , Christophe J
Ref : Molecular Pharmacology , 32 :91 , 1987
Abstract :
PubMedSearch : Waelbroeck_1987_Mol.Pharmacol_32_91
PubMedID: 3600616

Title : In vitro effects of gallamine on dissociation kinetics of (3H)N-methylscopolamine and (3H)pirenzepine from rat brain muscarinic receptors - Gillard_1986_J.Recept.Res_6_47
Author(s) : Gillard M , Waelbroeck M , Christophe J
Ref : J Recept Res , 6 :47 , 1986
Abstract :
PubMedSearch : Gillard_1986_J.Recept.Res_6_47
PubMedID: 3754901

Title : Propylbenzilylcholine mustard is selective for rat heart muscarinic receptors having a low affinity for agonists - Christophe_1986_Br.J.Pharmacol_88_63
Author(s) : Christophe J , de Neef P , Robberecht P , Waelbroeck M
Ref : British Journal of Pharmacology , 88 :63 , 1986
Abstract :
PubMedSearch : Christophe_1986_Br.J.Pharmacol_88_63
PubMedID: 3708224

Title : Kinetic studies of [3H]-N-methylscopolamine binding to muscarinic receptors in the rat central nervous system: evidence for the existence of three classes of binding sites - Waelbroeck_1986_Mol.Pharmacol_30_305
Author(s) : Waelbroeck M , Gillard M , Robberecht P , Christophe J
Ref : Molecular Pharmacology , 30 :305 , 1986
Abstract :
PubMedSearch : Waelbroeck_1986_Mol.Pharmacol_30_305
PubMedID: 3762520

Title : Secoverine is a non-selective muscarinic antagonist on rat heart and brain receptors - Brunner_1986_Eur.J.Pharmacol_127_17
Author(s) : Brunner F , Waelbroeck M , Christophe J
Ref : European Journal of Pharmacology , 127 :17 , 1986
Abstract :
PubMedSearch : Brunner_1986_Eur.J.Pharmacol_127_17
PubMedID: 3758175

Title : Effects of temperature and ethanol on agonist and antagonist binding to rat heart muscarinic receptors in the absence and presence of GTP - Waelbroeck_1985_Biochem.J_231_469
Author(s) : Waelbroeck M , Robberecht P , Chatelain P , de Neef P , Christophe J
Ref : Biochemical Journal , 231 :469 , 1985
Abstract :
PubMedSearch : Waelbroeck_1985_Biochem.J_231_469
PubMedID: 4062907

Title : Inhibitory effects of quinidine on rat heart muscarinic receptors - Waelbroeck_1984_Life.Sci_35_1069
Author(s) : Waelbroeck M , de Neef P , Robberecht P , Christophe J
Ref : Life Sciences , 35 :1069 , 1984
Abstract :
PubMedSearch : Waelbroeck_1984_Life.Sci_35_1069
PubMedID: 6482646

Title : Effects of verapamil on the binding properties of rat heart muscarinic receptors: evidence for an allosteric site - Waelbroeck_1984_Biochem.Biophys.Res.Commun_121_340
Author(s) : Waelbroeck M , Robberecht P , de Neef P , Christophe J
Ref : Biochemical & Biophysical Research Communications , 121 :340 , 1984
Abstract :
PubMedSearch : Waelbroeck_1984_Biochem.Biophys.Res.Commun_121_340
PubMedID: 6732812

Title : Multiple effects of short-chain alcohols on binding to rat heart muscarinic receptors - Waelbroeck_1984_Biochem.J_219_563
Author(s) : Waelbroeck M , Robberecht P , de Neef P , Christophe J
Ref : Biochemical Journal , 219 :563 , 1984
Abstract :
PubMedSearch : Waelbroeck_1984_Biochem.J_219_563
PubMedID: 6743233

Title : Characterization of muscarinic cholinergic receptors on rat pancreatic acini by N-[3H]methylscopolamine binding. Their relationship with calcium 45 efflux and amylase secretion - Dehaye_1984_J.Biol.Chem_259_294
Author(s) : Dehaye JP , Winand J , Poloczek P , Christophe J
Ref : Journal of Biological Chemistry , 259 :294 , 1984
Abstract :
PubMedSearch : Dehaye_1984_J.Biol.Chem_259_294
PubMedID: 6200472

Title : A comparison between muscarinic receptor occupancy, adenylate cyclase inhibition, and inotropic response in human heart - Delhaye_1984_Naunyn.Schmiedebergs.Arch.Pharmacol_325_170
Author(s) : Delhaye M , De Smet JM , Taton G , de Neef P , Camus JC , Fontaine J , Waelbroeck M , Robberecht P , Christophe J
Ref : Naunyn Schmiedebergs Arch Pharmacol , 325 :170 , 1984
Abstract :
PubMedSearch : Delhaye_1984_Naunyn.Schmiedebergs.Arch.Pharmacol_325_170
PubMedID: 6717612

Title : Effects of a chemical sympathectomy on cardiac muscarinic receptors in normotensive (WKY) and spontaneously hypertensive (SHR) rats -
Author(s) : Waelbroeck M , Robberecht P , Christophe J , Chatelain P , Huu AN , Roba J
Ref : Biochemical Pharmacology , 32 :1805 , 1983
PubMedID: 6409110

Title : Effect of pH on binding of agonists and antagonists to rat heart muscarinic receptors - Asselin_1983_Biochem.J_216_11
Author(s) : Asselin J , Waelbroeck M , Robberecht P , de Neef P , Christophe J
Ref : Biochemical Journal , 216 :11 , 1983
Abstract :
PubMedSearch : Asselin_1983_Biochem.J_216_11
PubMedID: 6651771

Title : Increased number of high-affinity muscarinic receptors in rat heart after phenylhydrazine treatment - Chatelain_1983_Eur.J.Pharmacol_91_279
Author(s) : Chatelain P , Waelbroeck M , de Neef P , Robberecht P , Christophe J
Ref : European Journal of Pharmacology , 91 :279 , 1983
Abstract :
PubMedSearch : Chatelain_1983_Eur.J.Pharmacol_91_279
PubMedID: 6225652

Title : Inhibitory effects of pirenzepine on muscarinic stimulation of rat pancreas - Dehaye_1983_Eur.J.Pharmacol_92_259
Author(s) : Dehaye JP , Winand J , Hermans L , Poloczek P , Christophe J
Ref : European Journal of Pharmacology , 92 :259 , 1983
Abstract :
PubMedSearch : Dehaye_1983_Eur.J.Pharmacol_92_259
PubMedID: 6605251

Title : Rat cardiac muscarinic receptors. I. Effects of guanine nucleotides on high- and low-affinity binding sites - Waelbroeck_1982_Mol.Pharmacol_21_581
Author(s) : Waelbroeck M , Robberecht P , Chatelain P , Christophe J
Ref : Molecular Pharmacology , 21 :581 , 1982
Abstract :
PubMedSearch : Waelbroeck_1982_Mol.Pharmacol_21_581
PubMedID: 7110116

Title : Rat cardiac muscarinic receptors. II. Influence of thyroid status and cardiac hypertrophy - Robberecht_1982_Mol.Pharmacol_21_589
Author(s) : Robberecht P , Waelbroeck M , Claeys M , Huu AN , Chatelain P , Christophe J
Ref : Molecular Pharmacology , 21 :589 , 1982
Abstract :
PubMedSearch : Robberecht_1982_Mol.Pharmacol_21_589
PubMedID: 6213844

Title : Guanine nucleotide binding sites, responsible for adenylate cyclase activation and carbamylcholine binding inhibition, show similar properties in rat heart membranes - Waelbroeck_1981_J.Cyclic.Nucleotide.Res_7_173
Author(s) : Waelbroeck M , Robberecht P , Chatelain P , Christophe J
Ref : J Cyclic Nucleotide Res , 7 :173 , 1981
Abstract :
PubMedSearch : Waelbroeck_1981_J.Cyclic.Nucleotide.Res_7_173
PubMedID: 7287969