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| Title : Poster: A study of M1 receptor coupling to inhibitory G proteins in CHO cells via GTPS binding determined with anti-G protein antibodies - |
| Author(s) : DeLapp NW , McClure D , McKinzie J , Silbernagel A , Sawyer BD , Felder CC |
| Ref : Life Sciences , 64 :569 , 1999 |
| PubMedID: |
| Title : Direct pharmacological comparison of the muscarinic receptors mediating relaxation and contraction in the rabbit thoracic aorta - Sawyer_1999_Gen.Pharmacol_32_445 |
| Author(s) : Sawyer BD , Bymaster FP , Calligaro DO , Falcone J , Mitch CH , Ward JS , Whitesitt CA , Shannon HE |
| Ref : General Pharmacology , 32 :445 , 1999 |
| Abstract : Sawyer_1999_Gen.Pharmacol_32_445 |
| ESTHER : Sawyer_1999_Gen.Pharmacol_32_445 |
| PubMedSearch : Sawyer_1999_Gen.Pharmacol_32_445 |
| PubMedID: 10323485 |
| Title : Poster: An anti-G protein scintillation proximity assay for M1-M5 receptor-mediated GTPS binding - |
| Author(s) : McKinzie JH , Sawyer BD , Felder CC , Falcone J , Silbernagel A , McClure D , DeLapp NW |
| Ref : Life Sciences , 64 :570 , 1999 |
| PubMedID: |
| Title : Poster: Comparison of GTP-gamma-35S and 3H-NMS binding in CHO cells stably expressing human M1-M5 muscarinic receptors using scintillation proximity assays - |
| Author(s) : Sawyer BD , Silbernagel A , McKinzie JB , Falcone J , DeLapp NW , Felder CC |
| Ref : Life Sciences , 64 :568 , 1999 |
| PubMedID: |
| Title : Conformationally constrained analogues of the muscarinic agonist 3-(4-(methylthio)-1,2,5-thiadiazol-3-yl)-1,2,5,6-tetrahydro-1-methylpyr idine. Synthesis, receptor affinity, and antinociceptive activity - Sauerberg_1998_J.Med.Chem_41_109 |
| Author(s) : Sauerberg P , Olesen PH , Sheardown MJ , Rimvall K , Thogersen H , Shannon HE , Sawyer BD , Ward JS , Bymaster FP , DeLapp NW , Calligaro DO , Swedberg MD |
| Ref : Journal of Medicinal Chemistry , 41 :109 , 1998 |
| Abstract : Sauerberg_1998_J.Med.Chem_41_109 |
| ESTHER : Sauerberg_1998_J.Med.Chem_41_109 |
| PubMedSearch : Sauerberg_1998_J.Med.Chem_41_109 |
| PubMedID: 9438027 |
| Title : Pharmacology of butylthio[2.2.2] (LY297802\/NNC11-1053): a novel analgesic with mixed muscarinic receptor agonist and antagonist activity - Shannon_1997_J.Pharmacol.Exp.Ther_281_884 |
| Author(s) : Shannon HE , Sheardown MJ , Bymaster FP , Calligaro DO , DeLapp NW , Gidda J , Mitch CH , Sawyer BD , Stengel PW , Ward JS , Wong DT , Olesen PH , Suzdak PD , Sauerberg P , Swedberg MD |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 281 :884 , 1997 |
| Abstract : Shannon_1997_J.Pharmacol.Exp.Ther_281_884 |
| ESTHER : Shannon_1997_J.Pharmacol.Exp.Ther_281_884 |
| PubMedSearch : Shannon_1997_J.Pharmacol.Exp.Ther_281_884 |
| PubMedID: 9152398 |
| Title : Detrusor regeneration in the rat using porcine small intestinal submucosal grafts: functional innervation and receptor expression - Vaught_1996_J.Urol_155_374 |
| Author(s) : Vaught JD , Kropp BP , Sawyer BD , Rippy MK , Badylak SF , Shannon HE , Thor KB |
| Ref : J Urol , 155 :374 , 1996 |
| Abstract : Vaught_1996_J.Urol_155_374 |
| ESTHER : Vaught_1996_J.Urol_155_374 |
| PubMedSearch : Vaught_1996_J.Urol_155_374 |
| PubMedID: 7490890 |
| Title : Poster: 3-(3-Hexyloxypyrazinyl)quinuclidine as a functionally selective M1 agonist - |
| Author(s) : Ward JS , Merritt L , Calligaro DO , Bymaster FP , Shannon HE , Sawyer BD , Mitch CH , Sheardown MJ , Olesen PH , Suzdak PD , Swedberg MD , Sauerberg P |
| Ref : Life Sciences , 56(11-12) :1003 , 1995 |
| PubMedID: |
| Title : Poster: Sidechain steric bulk and muscarinic agonist sar in alkoxy-TZTP's - |
| Author(s) : Mitch CH , Bymaster FP , Calligaro DO , Quimby SJ , Sawyer BD , Ward JS , Olesen PH , Sauerberg P , Sheardown MJ , Suzdak PD , Swedberg MD , Shannon HE |
| Ref : Life Sciences , 56(11-12) :1004 , 1995 |
| PubMedID: |
| Title : Poster: Muscarinic receptor characterization and evaluation of a series of novel muscarinic ligands in the isolated rabbit thoracic aorta - |
| Author(s) : Sawyer BD , Shannon HE , Ward JS , Mitch CH , Sheardown MJ , Olesen PH , Sauerberg P |
| Ref : Life Sciences , 56(11-12) :1004 , 1995 |
| PubMedID: |
| Title : Functionally selective M1 muscarinic agonists. 3. Side chains and azacycles contributing to functional muscarinic selectivity among pyrazinylazacycles - Ward_1995_J.Med.Chem_38_3469 |
| Author(s) : Ward JS , Merritt L , Calligaro DO , Bymaster FP , Shannon HE , Sawyer BD , Mitch CH , Deeter JB , Peters SC , Sheardown MJ , Olesen PH , Swedberg MD , Sauerberg P |
| Ref : Journal of Medicinal Chemistry , 38 :3469 , 1995 |
| Abstract : Ward_1995_J.Med.Chem_38_3469 |
| ESTHER : Ward_1995_J.Med.Chem_38_3469 |
| PubMedSearch : Ward_1995_J.Med.Chem_38_3469 |
| PubMedID: 7658434 |
| Title : Xanomeline: a novel muscarinic receptor agonist with functional selectivity for M1 receptors - Shannon_1994_J.Pharmacol.Exp.Ther_269_271 |
| Author(s) : Shannon HE , Bymaster FP , Calligaro DO , Greenwood B , Mitch CH , Sawyer BD , Ward JS , Wong DT , Olesen PH , Sheardown MJ |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 269 :271 , 1994 |
| Abstract : Shannon_1994_J.Pharmacol.Exp.Ther_269_271 |
| ESTHER : Shannon_1994_J.Pharmacol.Exp.Ther_269_271 |
| PubMedSearch : Shannon_1994_J.Pharmacol.Exp.Ther_269_271 |
| PubMedID: 7909557 |
| Title : Poster: Alkoxy sar around the functionally M1 selective agonist hexyloxy-TZTP - |
| Author(s) : Sauerberg P , Olesen PH , Sheardown MJ , Suzdak PD , Swedberg MD , Mitch CH , Ward JS , Calligaro DO , Sawyer BD , Bymaster FP , Shannon HE |
| Ref : Life Sciences , 52(5-6) :549 , 1993 |
| PubMedID: |
| Title : Poster: Synthesis and structure-activity relationship of 3-(pyrazinyl)- 1, 2, 5, 6-tetrahydro-1-methylpyridines. Construction of a molecular model for the M-1 pharmacophore - |
| Author(s) : Ward JS , Merritt L , Klimkowski VJ , Lamb ML , Mitch CH , Bymaster FP , Sawyer BD , Shannon HE , Olesen PH , Honore T , Sheardown MJ , Sauerberg P |
| Ref : Life Sciences , 52(5-6) :549 , 1993 |
| PubMedID: |
| Title : Poster: 3-hexyloxy analogs of TZTP are potent and selective M1 agonists in brain of rat in vivo - |
| Author(s) : Bymaster FP , Wong DT , Mitch CH , Ward JS , Calligaro DO , Shannon HE , Sawyer BD , Quimby SJ , Sheardown MJ , Olesen PH , Suzdak PD , Sauerberg P |
| Ref : Life Sciences , 52(5-6) :593 , 1993 |
| PubMedID: |
| Title : Muscarinic M1 receptor agonist actions of muscarinic receptor agonists in rabbit vas deferens - Shannon_1993_Eur.J.Pharmacol_232_47 |
| Author(s) : Shannon HE , Sawyer BD , Bemis KG , Bymaster FP , Health I , Mitch CH , Ward JS |
| Ref : European Journal of Pharmacology , 232 :47 , 1993 |
| Abstract : Shannon_1993_Eur.J.Pharmacol_232_47 |
| ESTHER : Shannon_1993_Eur.J.Pharmacol_232_47 |
| PubMedSearch : Shannon_1993_Eur.J.Pharmacol_232_47 |
| PubMedID: 8458395 |
| Title : Poster: Hexyloxy-TZTP: A potent and selective M1 agonist in-vitro - |
| Author(s) : Mitch CH , Bymaster FP , Calligaro DO , Quimby SJ , Sawyer BD , Shannon HE , Ward JS , Olesen PH , Sauerberg P , Sheardown MJ , Suzdak PD |
| Ref : Life Sciences , 52(5-6) :550 , 1993 |
| PubMedID: |
| Title : Novel functional M1 selective muscarinic agonists. 2. Synthesis and structure-activity relationships of 3-pyrazinyl-1,2,5,6-tetrahydro-1-methylpyridines. Construction of a molecular model for the M1 pharmacophore - Ward_1992_J.Med.Chem_35_4011 |
| Author(s) : Ward JS , Merritt L , Klimkowski VJ , Lamb ML , Mitch CH , Bymaster FP , Sawyer BD , Shannon HE , Olesen PH , Honore T , Sheardown MJ , Sauerberg P |
| Ref : Journal of Medicinal Chemistry , 35 :4011 , 1992 |
| Abstract : Ward_1992_J.Med.Chem_35_4011 |
| ESTHER : Ward_1992_J.Med.Chem_35_4011 |
| PubMedSearch : Ward_1992_J.Med.Chem_35_4011 |
| PubMedID: 1433209 |