Title : Design, synthesis and biological evaluation of second-generation benzoylpiperidine derivatives as reversible monoacylglycerol lipase (MAGL) inhibitors - Granchi_2020_Eur.J.Med.Chem_209_112857 |
Author(s) : Granchi C , Bononi G , Ferrisi R , Gori E , Mantini G , Glasmacher S , Poli G , Palazzolo S , Caligiuri I , Rizzolio F , Canzonieri V , Perin T , Gertsch J , Sodi A , Giovannetti E , Macchia M , Minutolo F , Tuccinardi T , Chicca A |
Ref : Eur Journal of Medicinal Chemistry , 209 :112857 , 2020 |
Abstract : Granchi_2020_Eur.J.Med.Chem_209_112857 |
ESTHER : Granchi_2020_Eur.J.Med.Chem_209_112857 |
PubMedSearch : Granchi_2020_Eur.J.Med.Chem_209_112857 |
PubMedID: 33045662 |
Gene_locus related to this paper: human-MGLL |
Gene_locus related to this paper: human-MGLL |
Granchi C, Bononi G, Ferrisi R, Gori E, Mantini G, Glasmacher S, Poli G, Palazzolo S, Caligiuri I, Rizzolio F, Canzonieri V, Perin T, Gertsch J, Sodi A, Giovannetti E, Macchia M, Minutolo F, Tuccinardi T, Chicca A (2020)
Design, synthesis and biological evaluation of second-generation benzoylpiperidine derivatives as reversible monoacylglycerol lipase (MAGL) inhibitors
Eur Journal of Medicinal Chemistry
209 :112857
Granchi C, Bononi G, Ferrisi R, Gori E, Mantini G, Glasmacher S, Poli G, Palazzolo S, Caligiuri I, Rizzolio F, Canzonieri V, Perin T, Gertsch J, Sodi A, Giovannetti E, Macchia M, Minutolo F, Tuccinardi T, Chicca A (2020)
Eur Journal of Medicinal Chemistry
209 :112857