Title : A Carrier Free Delivery System of a Monoacylglycerol Lipase Hydrophobic Inhibitor - Adeel_2021_Int.J.Pharm__121374 |
Author(s) : Adeel M , Saorin G , Boccalon G , Sfriso AA , Parisi S , Moro I , Palazzolo S , Caligiuri I , Granchi C , Corona G , Cemazar M , Canzonieri V , Tuccinardi T , Rizzolio F |
Ref : Int J Pharm , :121374 , 2021 |
Abstract : Adeel_2021_Int.J.Pharm__121374 |
ESTHER : Adeel_2021_Int.J.Pharm__121374 |
PubMedSearch : Adeel_2021_Int.J.Pharm__121374 |
PubMedID: 34906647 |
Title : Design, synthesis and biological evaluation of second-generation benzoylpiperidine derivatives as reversible monoacylglycerol lipase (MAGL) inhibitors - Granchi_2020_Eur.J.Med.Chem_209_112857 |
Author(s) : Granchi C , Bononi G , Ferrisi R , Gori E , Mantini G , Glasmacher S , Poli G , Palazzolo S , Caligiuri I , Rizzolio F , Canzonieri V , Perin T , Gertsch J , Sodi A , Giovannetti E , Macchia M , Minutolo F , Tuccinardi T , Chicca A |
Ref : Eur Journal of Medicinal Chemistry , 209 :112857 , 2020 |
Abstract : Granchi_2020_Eur.J.Med.Chem_209_112857 |
ESTHER : Granchi_2020_Eur.J.Med.Chem_209_112857 |
PubMedSearch : Granchi_2020_Eur.J.Med.Chem_209_112857 |
PubMedID: 33045662 |
Gene_locus related to this paper: human-MGLL |
Title : Structural Optimization of 4-Chlorobenzoylpiperidine Derivatives for the Development of Potent, Reversible, and Selective Monoacylglycerol Lipase (MAGL) Inhibitors - Granchi_2016_J.Med.Chem_59_10299 |
Author(s) : Granchi C , Rizzolio F , Palazzolo S , Carmignani S , Macchia M , Saccomanni G , Manera C , Martinelli A , Minutolo F , Tuccinardi T |
Ref : Journal of Medicinal Chemistry , 59 :10299 , 2016 |
Abstract : Granchi_2016_J.Med.Chem_59_10299 |
ESTHER : Granchi_2016_J.Med.Chem_59_10299 |
PubMedSearch : Granchi_2016_J.Med.Chem_59_10299 |
PubMedID: 27809504 |