| Title : Iso- and Benzisothiazolinone Inhibitors of Monoacylglycerol Lipase: Exploring On-Target Activity Through Scaffold Decoration and In Situ Warhead Generation - Rocca_2026_ChemMedChem_21_e70414 |
| Author(s) : Rocca E , Bedini A , Scalvini L , Galvani F , Castelli R , Sarcone L , Recchia A , Fanini F , Tran A , Rivara S , Spadoni G , Piomelli D , Mor M |
| Ref : ChemMedChem , 21 :e70414 , 2026 |
| Abstract : |
| PubMedSearch : Rocca_2026_ChemMedChem_21_e70414 |
| PubMedID: 42638513 |
| Title : Development of potent and selective FAAH inhibitors with improved drug-like properties as potential tools to treat neuroinflammatory conditions - Papa_2022_Eur.J.Med.Chem_246_114952 |
| Author(s) : Papa A , Pasquini S , Galvani F , Cammarota M , Contri C , Carullo G , Gemma S , Ramunno A , Lamponi S , Gorelli B , Saponara S , Varani K , Mor M , Campiani G , Boscia F , Vincenzi F , Lodola A , Butini S |
| Ref : Eur Journal of Medicinal Chemistry , 246 :114952 , 2022 |
| Abstract : |
| PubMedSearch : Papa_2022_Eur.J.Med.Chem_246_114952 |
| PubMedID: 36462439 |
| Title : Mechanistic Modeling of Monoglyceride Lipase Covalent Modification Elucidates the Role of Leaving Group Expulsion and Discriminates Inhibitors with High and Low Potency - Galvani_2022_J.Chem.Inf.Model__ |
| Author(s) : Galvani F , Scalvini L , Rivara S , Lodola A , Mor M |
| Ref : J Chem Inf Model , : , 2022 |
| Abstract : |
| PubMedSearch : Galvani_2022_J.Chem.Inf.Model__ |
| PubMedID: 35580195 |
| Gene_locus related to this paper: human-MGLL |