Title : Development of Potent and Selective Monoacylglycerol Lipase Inhibitors. SARs, Structural Analysis, and Biological Characterization - Butini_2024_J.Med.Chem__ |
Author(s) : Butini S , Grether U , Jung KM , Ligresti A , Allara M , Postmus AGJ , Maramai S , Brogi S , Papa A , Carullo G , Sykes D , Veprintsev D , Federico S , Grillo A , Di Guglielmo B , Ramunno A , Stevens AF , Heer D , Lamponi S , Gemma S , Benz J , Di Marzo V , van der Stelt M , Piomelli D , Campiani G |
Ref : Journal of Medicinal Chemistry , : , 2024 |
Abstract : |
PubMedSearch : Butini_2024_J.Med.Chem__ |
PubMedID: 38241614 |
Gene_locus related to this paper: human-MGLL |
Title : A Comparative Study between Lycorine and Galantamine Abilities to Interact with AMYLOID beta and Reduce In Vitro Neurotoxicity - Kola_2023_Int.J.Mol.Sci_24_ |
Author(s) : Kola A , Lamponi S , Curro F , Valensin D |
Ref : Int J Mol Sci , 24 : , 2023 |
Abstract : |
PubMedSearch : Kola_2023_Int.J.Mol.Sci_24_ |
PubMedID: 36768823 |
Title : Development of potent and selective FAAH inhibitors with improved drug-like properties as potential tools to treat neuroinflammatory conditions - Papa_2022_Eur.J.Med.Chem_246_114952 |
Author(s) : Papa A , Pasquini S , Galvani F , Cammarota M , Contri C , Carullo G , Gemma S , Ramunno A , Lamponi S , Gorelli B , Saponara S , Varani K , Mor M , Campiani G , Boscia F , Vincenzi F , Lodola A , Butini S |
Ref : Eur Journal of Medicinal Chemistry , 246 :114952 , 2022 |
Abstract : |
PubMedSearch : Papa_2022_Eur.J.Med.Chem_246_114952 |
PubMedID: 36462439 |
Title : Development and Pharmacological Characterization of Selective Blockers of 2-Arachidonoyl Glycerol Degradation with Efficacy in Rodent Models of Multiple Sclerosis and Pain - Brindisi_2016_J.Med.Chem_59_2612 |
Author(s) : Brindisi M , Maramai S , Gemma S , Brogi S , Grillo A , Di Cesare Mannelli L , Gabellieri E , Lamponi S , Saponara S , Gorelli B , Tedesco D , Bonfiglio T , Landry C , Jung KM , Armirotti A , Luongo L , Ligresti A , Piscitelli F , Bertucci C , Dehouck MP , Campiani G , Maione S , Ghelardini C , Pittaluga A , Piomelli D , Di Marzo V , Butini S |
Ref : Journal of Medicinal Chemistry , 59 :2612 , 2016 |
Abstract : |
PubMedSearch : Brindisi_2016_J.Med.Chem_59_2612 |
PubMedID: 26888301 |
Title : Disease-Modifying Anti-Alzheimer's Drugs: Inhibitors of Human Cholinesterases Interfering with beta-Amyloid Aggregation - Brogi_2014_CNS.Neurosci.Ther_20_624 |
Author(s) : Brogi S , Butini S , Maramai S , Colombo R , Verga L , Lanni C , De Lorenzi E , Lamponi S , Andreassi M , Bartolini M , Andrisano V , Novellino E , Campiani G , Brindisi M , Gemma S |
Ref : CNS Neurosci Ther , 20 :624 , 2014 |
Abstract : |
PubMedSearch : Brogi_2014_CNS.Neurosci.Ther_20_624 |
PubMedID: 24935788 |