| Title : 5-methyl-2-carboxamidepyrrole-based novel dual mPGES-1\/sEH inhibitors as promising anticancer candidates - Colarusso_2025_Arch.Pharm.(Weinheim)_358_e2400708 |
| Author(s) : Colarusso E , Lauro G , Potenza M , Galatello P , Garigliota MLD , Ferraro MG , Piccolo M , Chini MG , Irace C , Campiglia P , Hoffstetter RK , Werz O , Ramunno A , Bifulco G |
| Ref : Arch Pharm (Weinheim) , 358 :e2400708 , 2025 |
| Abstract : |
| PubMedSearch : Colarusso_2025_Arch.Pharm.(Weinheim)_358_e2400708 |
| PubMedID: 39692230 |
| Title : 5-methyl-2-carboxamidepyrrole-based novel dual mPGES-1\/sEH inhibitors as promising anticancer candidates - Colarusso_2025_Arch.Pharm.(Weinheim)_358_e2400708 |
| Author(s) : Colarusso E , Lauro G , Potenza M , Galatello P , Garigliota MLD , Ferraro MG , Piccolo M , Chini MG , Irace C , Campiglia P , Hoffstetter RK , Werz O , Ramunno A , Bifulco G |
| Ref : Arch Pharm (Weinheim) , 358 :e2400708 , 2025 |
| Abstract : |
| PubMedSearch : Colarusso_2025_Arch.Pharm.(Weinheim)_358_e2400708 |
| PubMedID: 39692230 |
| Title : 5-methyl-2-carboxamidepyrrole-based novel dual mPGES-1\/sEH inhibitors as promising anticancer candidates - Colarusso_2025_Arch.Pharm.(Weinheim)_358_e2400708 |
| Author(s) : Colarusso E , Lauro G , Potenza M , Galatello P , Garigliota MLD , Ferraro MG , Piccolo M , Chini MG , Irace C , Campiglia P , Hoffstetter RK , Werz O , Ramunno A , Bifulco G |
| Ref : Arch Pharm (Weinheim) , 358 :e2400708 , 2025 |
| Abstract : |
| PubMedSearch : Colarusso_2025_Arch.Pharm.(Weinheim)_358_e2400708 |
| PubMedID: 39692230 |
| Title : Development of Potent and Selective Monoacylglycerol Lipase Inhibitors. SARs, Structural Analysis, and Biological Characterization - Butini_2024_J.Med.Chem__ |
| Author(s) : Butini S , Grether U , Jung KM , Ligresti A , Allara M , Postmus AGJ , Maramai S , Brogi S , Papa A , Carullo G , Sykes D , Veprintsev D , Federico S , Grillo A , Di Guglielmo B , Ramunno A , Stevens AF , Heer D , Lamponi S , Gemma S , Benz J , Di Marzo V , van der Stelt M , Piomelli D , Campiani G |
| Ref : Journal of Medicinal Chemistry , : , 2024 |
| Abstract : |
| PubMedSearch : Butini_2024_J.Med.Chem__ |
| PubMedID: 38241614 |
| Gene_locus related to this paper: human-MGLL |
| Title : Development of Potent and Selective Monoacylglycerol Lipase Inhibitors. SARs, Structural Analysis, and Biological Characterization - Butini_2024_J.Med.Chem__ |
| Author(s) : Butini S , Grether U , Jung KM , Ligresti A , Allara M , Postmus AGJ , Maramai S , Brogi S , Papa A , Carullo G , Sykes D , Veprintsev D , Federico S , Grillo A , Di Guglielmo B , Ramunno A , Stevens AF , Heer D , Lamponi S , Gemma S , Benz J , Di Marzo V , van der Stelt M , Piomelli D , Campiani G |
| Ref : Journal of Medicinal Chemistry , : , 2024 |
| Abstract : |
| PubMedSearch : Butini_2024_J.Med.Chem__ |
| PubMedID: 38241614 |
| Gene_locus related to this paper: human-MGLL |
| Title : Development of Potent and Selective Monoacylglycerol Lipase Inhibitors. SARs, Structural Analysis, and Biological Characterization - Butini_2024_J.Med.Chem__ |
| Author(s) : Butini S , Grether U , Jung KM , Ligresti A , Allara M , Postmus AGJ , Maramai S , Brogi S , Papa A , Carullo G , Sykes D , Veprintsev D , Federico S , Grillo A , Di Guglielmo B , Ramunno A , Stevens AF , Heer D , Lamponi S , Gemma S , Benz J , Di Marzo V , van der Stelt M , Piomelli D , Campiani G |
| Ref : Journal of Medicinal Chemistry , : , 2024 |
| Abstract : |
| PubMedSearch : Butini_2024_J.Med.Chem__ |
| PubMedID: 38241614 |
| Gene_locus related to this paper: human-MGLL |
| Title : Development of potent and selective FAAH inhibitors with improved drug-like properties as potential tools to treat neuroinflammatory conditions - Papa_2022_Eur.J.Med.Chem_246_114952 |
| Author(s) : Papa A , Pasquini S , Galvani F , Cammarota M , Contri C , Carullo G , Gemma S , Ramunno A , Lamponi S , Gorelli B , Saponara S , Varani K , Mor M , Campiani G , Boscia F , Vincenzi F , Lodola A , Butini S |
| Ref : Eur Journal of Medicinal Chemistry , 246 :114952 , 2022 |
| Abstract : |
| PubMedSearch : Papa_2022_Eur.J.Med.Chem_246_114952 |
| PubMedID: 36462439 |
| Title : Development of potent and selective FAAH inhibitors with improved drug-like properties as potential tools to treat neuroinflammatory conditions - Papa_2022_Eur.J.Med.Chem_246_114952 |
| Author(s) : Papa A , Pasquini S , Galvani F , Cammarota M , Contri C , Carullo G , Gemma S , Ramunno A , Lamponi S , Gorelli B , Saponara S , Varani K , Mor M , Campiani G , Boscia F , Vincenzi F , Lodola A , Butini S |
| Ref : Eur Journal of Medicinal Chemistry , 246 :114952 , 2022 |
| Abstract : |
| PubMedSearch : Papa_2022_Eur.J.Med.Chem_246_114952 |
| PubMedID: 36462439 |
| Title : Development of potent and selective FAAH inhibitors with improved drug-like properties as potential tools to treat neuroinflammatory conditions - Papa_2022_Eur.J.Med.Chem_246_114952 |
| Author(s) : Papa A , Pasquini S , Galvani F , Cammarota M , Contri C , Carullo G , Gemma S , Ramunno A , Lamponi S , Gorelli B , Saponara S , Varani K , Mor M , Campiani G , Boscia F , Vincenzi F , Lodola A , Butini S |
| Ref : Eur Journal of Medicinal Chemistry , 246 :114952 , 2022 |
| Abstract : |
| PubMedSearch : Papa_2022_Eur.J.Med.Chem_246_114952 |
| PubMedID: 36462439 |
| Title : 3-(2-Aminoethyl)pyridine analogs as alpha4beta2 nicotinic cholinergic receptor ligands - Dukat_2005_Bioorg.Med.Chem.Lett_15_4308 |
| Author(s) : Dukat M , Ramunno A , Banzi R , Damaj MI , Martin B , Glennon RA |
| Ref : Bioorganic & Medicinal Chemistry Lett , 15 :4308 , 2005 |
| Abstract : |
| PubMedSearch : Dukat_2005_Bioorg.Med.Chem.Lett_15_4308 |
| PubMedID: 16039854 |
| Title : 6-(2-Phenylethyl)nicotine: a novel nicotinic cholinergic receptor ligand - Ramunno_2005_Bioorg.Med.Chem.Lett_15_3237 |
| Author(s) : Ramunno A , Dukat M , Lee M , Young R , El-Zahabi M , Damaj MI , Martin B , Glennon RA |
| Ref : Bioorganic & Medicinal Chemistry Lett , 15 :3237 , 2005 |
| Abstract : |
| PubMedSearch : Ramunno_2005_Bioorg.Med.Chem.Lett_15_3237 |
| PubMedID: 15925512 |
| Title : 3-(2-Aminoethyl)pyridine analogs as alpha4beta2 nicotinic cholinergic receptor ligands - Dukat_2005_Bioorg.Med.Chem.Lett_15_4308 |
| Author(s) : Dukat M , Ramunno A , Banzi R , Damaj MI , Martin B , Glennon RA |
| Ref : Bioorganic & Medicinal Chemistry Lett , 15 :4308 , 2005 |
| Abstract : |
| PubMedSearch : Dukat_2005_Bioorg.Med.Chem.Lett_15_4308 |
| PubMedID: 16039854 |
| Title : 3-(2-Aminoethyl)pyridine analogs as alpha4beta2 nicotinic cholinergic receptor ligands - Dukat_2005_Bioorg.Med.Chem.Lett_15_4308 |
| Author(s) : Dukat M , Ramunno A , Banzi R , Damaj MI , Martin B , Glennon RA |
| Ref : Bioorganic & Medicinal Chemistry Lett , 15 :4308 , 2005 |
| Abstract : |
| PubMedSearch : Dukat_2005_Bioorg.Med.Chem.Lett_15_4308 |
| PubMedID: 16039854 |
| Title : 6-(2-Phenylethyl)nicotine: a novel nicotinic cholinergic receptor ligand - Ramunno_2005_Bioorg.Med.Chem.Lett_15_3237 |
| Author(s) : Ramunno A , Dukat M , Lee M , Young R , El-Zahabi M , Damaj MI , Martin B , Glennon RA |
| Ref : Bioorganic & Medicinal Chemistry Lett , 15 :3237 , 2005 |
| Abstract : |
| PubMedSearch : Ramunno_2005_Bioorg.Med.Chem.Lett_15_3237 |
| PubMedID: 15925512 |
| Title : 6-(2-Phenylethyl)nicotine: a novel nicotinic cholinergic receptor ligand - Ramunno_2005_Bioorg.Med.Chem.Lett_15_3237 |
| Author(s) : Ramunno A , Dukat M , Lee M , Young R , El-Zahabi M , Damaj MI , Martin B , Glennon RA |
| Ref : Bioorganic & Medicinal Chemistry Lett , 15 :3237 , 2005 |
| Abstract : |
| PubMedSearch : Ramunno_2005_Bioorg.Med.Chem.Lett_15_3237 |
| PubMedID: 15925512 |