| Title : Next generation thiazolyl ketone inhibitors of cytosolic phospholipase A(2) alpha for targeted cancer therapy - Ashcroft_2025_Nat.Commun_16_164 |
| Author(s) : Ashcroft FJ , Bourboula A , Mahammad N , Barbayianni E , Feuerherm AJ , Nguyen TT , Hayashi D , Kokotou MG , Alevizopoulos K , Dennis EA , Kokotos G , Johansen B |
| Ref : Nat Commun , 16 :164 , 2025 |
| Abstract : |
| PubMedSearch : Ashcroft_2025_Nat.Commun_16_164 |
| PubMedID: 39747052 |
| Title : A Lipidomic Approach to Studying the Downregulation of Free Fatty Acids by Cytosolic Phospholipase A(2) Inhibitors - Bourboula_2025_Biomolecules_15_ |
| Author(s) : Bourboula A , Mantzourani C , Chalatsa I , Machalia C , Emmanouilidou E , Kokotou MG , Kokotos G |
| Ref : Biomolecules , 15 : , 2025 |
| Abstract : |
| PubMedSearch : Bourboula_2025_Biomolecules_15_ |
| PubMedID: 40427519 |
| Title : Phospholipase A2 enzymes: physical structure, biological function, disease implication, chemical inhibition, and therapeutic intervention - |
| Author(s) : Dennis EA , Cao J , Hsu YH , Magrioti V , Kokotos G |
| Ref : Chem Rev , 111 :6130 , 2011 |
| PubMedID: 21910409 |
| Gene_locus related to this paper: human-PLA2G15 |
| Title : A novel monoacylglycerol lipase inhibitor with analgesic and anti-inflammatory activity - Magrioti_2008_Bioorg.Med.Chem.Lett_18_5424 |
| Author(s) : Magrioti V , Naxakis G , Hadjipavlou-Litina D , Makriyannis A , Kokotos G |
| Ref : Bioorganic & Medicinal Chemistry Lett , 18 :5424 , 2008 |
| Abstract : |
| PubMedSearch : Magrioti_2008_Bioorg.Med.Chem.Lett_18_5424 |
| PubMedID: 18819796 |
| Title : Enzymatic removal of carboxyl protecting groups. III. Fast removal of allyl and chloroethyl esters by Bacillus subtilis esterase (BS2) - Fotakopoulou_2007_J.Org.Chem_72_782 |
| Author(s) : Fotakopoulou I , Barbayianni E , Constantinou-Kokotou V , Bornscheuer UT , Kokotos G |
| Ref : J Org Chem , 72 :782 , 2007 |
| Abstract : |
| PubMedSearch : Fotakopoulou_2007_J.Org.Chem_72_782 |
| PubMedID: 17253795 |
| Title : Enzymatic removal of carboxyl protecting groups. 1. Cleavage of the tert-butyl moiety - Schmidt_2005_J.Org.Chem_70_3737 |
| Author(s) : Schmidt M , Barbayianni E , Fotakopoulou I , Hohne M , Constantinou-Kokotou V , Bornscheuer UT , Kokotos G |
| Ref : J Org Chem , 70 :3737 , 2005 |
| Abstract : |
| PubMedSearch : Schmidt_2005_J.Org.Chem_70_3737 |
| PubMedID: 15845019 |
| Gene_locus related to this paper: canan-lipasA |
| Title : Enzymatic removal of carboxyl protecting groups. 2. Cleavage of the benzyl and methyl moieties - Barbayianni_2005_J.Org.Chem_70_8730 |
| Author(s) : Barbayianni E , Fotakopoulou I , Schmidt M , Constantinou-Kokotou V , Bornscheuer UT , Kokotos G |
| Ref : J Org Chem , 70 :8730 , 2005 |
| Abstract : |
| PubMedSearch : Barbayianni_2005_J.Org.Chem_70_8730 |
| PubMedID: 16238302 |
| Title : Novel trifluoromethyl ketones as potent gastric lipase inhibitors - Kokotos_2003_Chembiochem_4_90 |
| Author(s) : Kokotos G , Kotsovolou S , Verger R |
| Ref : Chembiochem , 4 :90 , 2003 |
| Abstract : |
| PubMedSearch : Kokotos_2003_Chembiochem_4_90 |
| PubMedID: 12512081 |
| Title : Synthesis of lipophilic aldehydes and study of their inhibition effect on human digestive lipases - Kotsovolou_2002_Org.Lett_4_2625 |
| Author(s) : Kotsovolou S , Verger R , Kokotos G |
| Ref : Org Lett , 4 :2625 , 2002 |
| Abstract : |
| PubMedSearch : Kotsovolou_2002_Org.Lett_4_2625 |
| PubMedID: 12153194 |
| Title : Synthetic routes and lipase-inhibiting activity of long-chain alpha-keto amides - Chiou_2001_Lipids_36_535 |
| Author(s) : Chiou A , Verger R , Kokotos G |
| Ref : Lipids , 36 :535 , 2001 |
| Abstract : |
| PubMedSearch : Chiou_2001_Lipids_36_535 |
| PubMedID: 11432468 |
| Title : New fluorogenic substrates for the study of secondary specificity of prolyl oligopeptidase - Noula_1997_J.Pept.Res_49_46 |
| Author(s) : Noula C , Kokotos G , Barth T , Tzougraki C |
| Ref : J Pept Res , 49 :46 , 1997 |
| Abstract : |
| PubMedSearch : Noula_1997_J.Pept.Res_49_46 |
| PubMedID: 9128099 |