| Title : Discovery of long-chain salicylketoxime derivatives as monoacylglycerol lipase (MAGL) inhibitors - Bononi_2018_Eur.J.Med.Chem_157_817 |
| Author(s) : Bononi G , Granchi C , Lapillo M , Giannotti M , Nieri D , Fortunato S , Boustani ME , Caligiuri I , Poli G , Carlson KE , Kim SH , Macchia M , Martinelli A , Rizzolio F , Chicca A , Katzenellenbogen JA , Minutolo F , Tuccinardi T |
| Ref : Eur Journal of Medicinal Chemistry , 157 :817 , 2018 |
| Abstract : |
| PubMedSearch : Bononi_2018_Eur.J.Med.Chem_157_817 |
| PubMedID: 30144699 |
| Title : Rational Development of MAGL Inhibitors - Granchi_2018_Methods.Mol.Biol_1824_335 |
| Author(s) : Granchi C , Rizzolio F , Caligiuri I , Macchia M , Martinelli A , Minutolo F , Tuccinardi T |
| Ref : Methods Mol Biol , 1824 :335 , 2018 |
| Abstract : |
| PubMedSearch : Granchi_2018_Methods.Mol.Biol_1824_335 |
| PubMedID: 30039417 |
| Title : Discovery of 1,5-Diphenylpyrazole-3-Carboxamide Derivatives as Potent, Reversible, and Selective Monoacylglycerol Lipase (MAGL) Inhibitors - Aghazadeh Tabrizi_2018_J.Med.Chem_61_1340 |
| Author(s) : Aghazadeh Tabrizi M , Baraldi PG , Baraldi S , Ruggiero E , De Stefano L , Rizzolio F , Di Cesare Mannelli L , Ghelardini C , Chicca A , Lapillo M , Gertsch J , Manera C , Macchia M , Martinelli A , Granchi C , Minutolo F , Tuccinardi T |
| Ref : Journal of Medicinal Chemistry , 61 :1340 , 2018 |
| Abstract : |
| PubMedSearch : Aghazadeh Tabrizi_2018_J.Med.Chem_61_1340 |
| PubMedID: 29309142 |
| Title : 4-Aryliden-2-methyloxazol-5(4H)-one as a new scaffold for selective reversible MAGL inhibitors - Granchi_2016_J.Enzyme.Inhib.Med.Chem_31_137 |
| Author(s) : Granchi C , Rizzolio F , Bordoni V , Caligiuri I , Manera C , Macchia M , Minutolo F , Martinelli A , Giordano A , Tuccinardi T |
| Ref : J Enzyme Inhib Med Chem , 31 :137 , 2016 |
| Abstract : |
| PubMedSearch : Granchi_2016_J.Enzyme.Inhib.Med.Chem_31_137 |
| PubMedID: 25669350 |
| Title : Structural Optimization of 4-Chlorobenzoylpiperidine Derivatives for the Development of Potent, Reversible, and Selective Monoacylglycerol Lipase (MAGL) Inhibitors - Granchi_2016_J.Med.Chem_59_10299 |
| Author(s) : Granchi C , Rizzolio F , Palazzolo S , Carmignani S , Macchia M , Saccomanni G , Manera C , Martinelli A , Minutolo F , Tuccinardi T |
| Ref : Journal of Medicinal Chemistry , 59 :10299 , 2016 |
| Abstract : |
| PubMedSearch : Granchi_2016_J.Med.Chem_59_10299 |
| PubMedID: 27809504 |
| Title : Identification and characterization of a new reversible MAGL inhibitor - Tuccinardi_2014_Bioorg.Med.Chem_22_3285 |
| Author(s) : Tuccinardi T , Granchi C , Rizzolio F , Caligiuri I , Battistello V , Toffoli G , Minutolo F , Macchia M , Martinelli A |
| Ref : Bioorganic & Medicinal Chemistry , 22 :3285 , 2014 |
| Abstract : |
| PubMedSearch : Tuccinardi_2014_Bioorg.Med.Chem_22_3285 |
| PubMedID: 24853323 |
| Title : The genome and transcriptome of Haemonchus contortus, a key model parasite for drug and vaccine discovery - Laing_2013_Genome.Biol_14_R88 |
| Author(s) : Laing R , Kikuchi T , Martinelli A , Tsai IJ , Beech RN , Redman E , Holroyd N , Bartley DJ , Beasley H , Britton C , Curran D , Devaney E , Gilabert A , Hunt M , Jackson F , Johnston SL , Kryukov I , Li K , Morrison AA , Reid AJ , Sargison N , Saunders GI , Wasmuth JD , Wolstenholme A , Berriman M , Gilleard JS , Cotton JA |
| Ref : Genome Biol , 14 :R88 , 2013 |
| Abstract : |
| PubMedSearch : Laing_2013_Genome.Biol_14_R88 |
| PubMedID: 23985316 |
| Gene_locus related to this paper: haeco-u6nsf0 , haeco-u6psa2 , haeco-u6pu58 |
| Title : Lipase immobilization on differently functionalized vinyl-based amphiphilic polymers: influence of phase segregation on the enzyme hydrolytic activity - Bellusci_2012_Biomacromolecules_13_805 |
| Author(s) : Bellusci M , Francolini I , Martinelli A , D'Ilario L , Piozzi A |
| Ref : Biomacromolecules , 13 :805 , 2012 |
| Abstract : |
| PubMedSearch : Bellusci_2012_Biomacromolecules_13_805 |
| PubMedID: 22295868 |