| Title : Design of Benzoxathiazin-3-one 1,1-Dioxides as a New Class of Irreversible Serine Hydrolase Inhibitors: Discovery of a Uniquely Selective PNPLA4 Inhibitor - Kornahrens_2017_J.Am.Chem.Soc_139_7052 |
| Author(s) : Kornahrens AF , Cognetta AB, 3rd , Brody DM , Matthews ML , Cravatt BF , Boger DL |
| Ref : Journal of the American Chemical Society , 139 :7052 , 2017 |
| Abstract : |
| PubMedSearch : Kornahrens_2017_J.Am.Chem.Soc_139_7052 |
| PubMedID: 28498651 |
| Title : Chemical Proteomic Profiling of Human Methyltransferases - Horning_2016_J.Am.Chem.Soc_138_13335 |
| Author(s) : Horning BD , Suciu RM , Ghadiri DA , Ulanovskaya OA , Matthews ML , Lum KM , Backus KM , Brown SJ , Rosen H , Cravatt BF |
| Ref : Journal of the American Chemical Society , 138 :13335 , 2016 |
| Abstract : |
| PubMedSearch : Horning_2016_J.Am.Chem.Soc_138_13335 |
| PubMedID: 27689866 |
| Title : Design of activated serine-containing catalytic triads with atomic-level accuracy - Rajagopalan_2014_Nat.Chem.Biol_10_386 |
| Author(s) : Rajagopalan S , Wang C , Yu K , Kuzin AP , Richter F , Lew S , Miklos AE , Matthews ML , Seetharaman J , Su M , Hunt JF , Cravatt BF , Baker D |
| Ref : Nat Chemical Biology , 10 :386 , 2014 |
| Abstract : |
| PubMedSearch : Rajagopalan_2014_Nat.Chem.Biol_10_386 |
| PubMedID: 24705591 |
| Title : Highly selective inhibitors of monoacylglycerol lipase bearing a reactive group that is bioisosteric with endocannabinoid substrates - Chang_2012_Chem.Biol_19_579 |
| Author(s) : Chang JW , Niphakis MJ , Lum KM , Cognetta AB, 3rd , Wang C , Matthews ML , Niessen S , Buczynski MW , Parsons LH , Cravatt BF |
| Ref : Chemical Biology , 19 :579 , 2012 |
| Abstract : |
| PubMedSearch : Chang_2012_Chem.Biol_19_579 |
| PubMedID: 22542104 |
| Gene_locus related to this paper: human-MGLL |