8PTQ
Name : Crystal structure of human monoacylglycerol lipase in complex with compound 5l
Revelation date : 31-Jan-2024
Family : Monoglyceridelipase_lysophospholip
Gene_locus : human-MGLL
PDB file : ESTHER: header of PDB entry RCSB: Full entry
Comment
Butini, S.,Benz, J.,Grether, U.,Leibrock, L.,Papa, A.,Maramai, S.,Carullo, G.,Federico, S.,Grillo, A.,Di Guglielmo, B.,Lamponi, S.,Gemma, S.,Campiani, G.
Ligand : Ligand in structure: Ligplot
References (1)
| Title : Development of Potent and Selective Monoacylglycerol Lipase Inhibitors. SARs, Structural Analysis, and Biological Characterization - Butini_2024_J.Med.Chem__ |
| Author(s) : Butini S , Grether U , Jung KM , Ligresti A , Allara M , Postmus AGJ , Maramai S , Brogi S , Papa A , Carullo G , Sykes D , Veprintsev D , Federico S , Grillo A , Di Guglielmo B , Ramunno A , Stevens AF , Heer D , Lamponi S , Gemma S , Benz J , Di Marzo V , van der Stelt M , Piomelli D , Campiani G |
| Ref : Journal of Medicinal Chemistry , : , 2024 |
| Abstract : |
| PubMedSearch : Butini_2024_J.Med.Chem__ |
| PubMedID: 38241614 |
| Gene_locus related to this paper: human-MGLL |
Representative scheme of Prolylcarboxypeptidase structure and an image from PDBsum server
Databases
PDB-Sum : 8PTQ Previously Class, Architecture, Topology and Homologous superfamily - PDB-Sum server
FSSP : 8PTQ Fold classification based on Structure-Structure alignment of Proteins - FSSP server
SCOP : 8PTQ Structural Classification Of Protein - SCOP server
PROTEOPEDIA : 8PTQ 3D, interactive encyclopedia of proteins - PROTEOPEDIA server