Title : Delta-containing GABA(A) receptors in pain management: Promising targets for novel analgesics - Luo_2021_Neuropharmacol_195_108675 |
Author(s) : Luo Y , Kusay AS , Jiang T , Chebib M , Balle T |
Ref : Neuropharmacology , 195 :108675 , 2021 |
Abstract : |
PubMedSearch : Luo_2021_Neuropharmacol_195_108675 |
PubMedID: 34153311 |
Title : Novel Approach for the Search for Chemical Scaffolds with Dual Activity with Acetylcholinesterase and the alpha7 Nicotinic Acetylcholine Receptor-A Perspective for the Treatment of Neurodegenerative Disorders - Kowal_2019_Molecules_24_ |
Author(s) : Kowal NM , Indurthi DC , Ahring PK , Chebib M , Olafsdottir ES , Balle T |
Ref : Molecules , 24 : , 2019 |
Abstract : |
PubMedSearch : Kowal_2019_Molecules_24_ |
PubMedID: 30691196 |
Title : Galantamine is not a positive allosteric modulator of human alpha4beta2 or alpha7 nicotinic acetylcholine receptors - Kowal_2018_Br.J.Pharmacol_175_2911 |
Author(s) : Kowal NM , Ahring PK , Liao VWY , Indurti DC , Harvey BS , O'Connor SM , Chebib M , Olafsdottir ES , Balle T |
Ref : British Journal of Pharmacology , 175 :2911 , 2018 |
Abstract : |
PubMedSearch : Kowal_2018_Br.J.Pharmacol_175_2911 |
PubMedID: 29669164 |
Title : Pinnatoxins E, F and G target multiple nicotinic receptor subtypes - Hellyer_2015_J.Neurochem_135_479 |
Author(s) : Hellyer SD , Indurthi DC , Balle T , Runder-Varga V , Selwood AI , Tyndall JD , Chebib M , Rhodes L , Kerr DS |
Ref : Journal of Neurochemistry , 135 :479 , 2015 |
Abstract : |
PubMedSearch : Hellyer_2015_J.Neurochem_135_479 |
PubMedID: 26173951 |
Title : Poster: Exploring the structure activity relationships of halogen containing N-(pyridin-3-yl)-piperazines and homopiperazines at alpha4beta2 nAChRs - |
Author(s) : Rudner-Varga V , Ahring PK , Indurthi D , Peters D , Orton H , Kanizaj N , McLeod MD , Chebib M , Balle T |
Ref : Biochemical Pharmacology , 97 :623 , 2015 |
PubMedID: |
Title : Engineered alpha4beta2 nicotinic acetylcholine receptors as models for measuring agonist binding and effect at the orthosteric low-affinity alpha4-alpha4 interface - Ahring_2015_Neuropharmacol_92_135 |
Author(s) : Ahring PK , Olsen JA , Nielsen EO , Peters D , Pedersen MH , Rohde LA , Kastrup JS , Shahsavar A , Indurthi DC , Chebib M , Gajhede M , Balle T |
Ref : Neuropharmacology , 92 :135 , 2015 |
Abstract : |
PubMedSearch : Ahring_2015_Neuropharmacol_92_135 |
PubMedID: 25595102 |
Title : Poster: Exploiting ligand selectivity to understand allosteric receptor opening - |
Author(s) : Indurthi DC , Balle T , Ahring PK , Chebib M , Lewis TM , Absalom NL |
Ref : Biochemical Pharmacology , 97 :624 , 2015 |
PubMedID: |
Title : Presence of multiple binding sites on alpha9alpha10 nAChR receptors alludes to stoichiometric-dependent action of the alpha-conotoxin, Vc1.1 - Indurthi_2014_Biochem.Pharmacol_89_131 |
Author(s) : Indurthi DC , Pera E , Kim HL , Chu C , McLeod MD , McIntosh JM , Absalom NL , Chebib M |
Ref : Biochemical Pharmacology , 89 :131 , 2014 |
Abstract : |
PubMedSearch : Indurthi_2014_Biochem.Pharmacol_89_131 |
PubMedID: 24548457 |
Title : Covalent trapping of methyllycaconitine at the alpha4-alpha4 interface of the alpha4beta2 nicotinic acetylcholine receptor: antagonist binding site and mode of receptor inhibition revealed - Absalom_2013_J.Biol.Chem_288_26521 |
Author(s) : Absalom NL , Quek G , Lewis TM , Qudah T , von Arenstorff I , Ambrus JI , Harpsoe K , Karim N , Balle T , McLeod MD , Chebib M |
Ref : Journal of Biological Chemistry , 288 :26521 , 2013 |
Abstract : |
PubMedSearch : Absalom_2013_J.Biol.Chem_288_26521 |
PubMedID: 23893416 |
Title : Poster: An additional binding site for methyllycaconitine (MLA) and analogs occurs at the alpha4-alpha4 interface of the (alpha4)3(beta2)2 nAChR - |
Author(s) : Chebib M , Absalom NL , Quek G , Indurthi DC , Lewis TM , Qudah T , von Arenstorff I , Halliday JI , Ambrus JI , Harpsoe K , Karim N , Balle T , McLeod MD |
Ref : Biochemical Pharmacology , 86 :1225 , 2013 |
PubMedID: |
Title : Covalent attachment of antagonists to the alpha7 nicotinic acetylcholine receptor: synthesis and reactivity of substituted maleimides - Ambrus_2012_Chem.Commun.(Camb)_48_6699 |
Author(s) : Ambrus JI , Halliday JI , Kanizaj N , Absalom N , Harpsoe K , Balle T , Chebib M , McLeod MD |
Ref : Chem Commun (Camb) , 48 :6699 , 2012 |
Abstract : |
PubMedSearch : Ambrus_2012_Chem.Commun.(Camb)_48_6699 |
PubMedID: 22627701 |
Title : Identifying the binding site of novel methyllycaconitine (MLA) analogs at alpha4beta2 nicotinic acetylcholine receptors - Quek_2010_ACS.Chem.Neurosci_1_796 |
Author(s) : Quek GX , Lin D , Halliday JI , Absalom N , Ambrus JI , Thompson AJ , Lochner M , Lummis SC , McLeod MD , Chebib M |
Ref : ACS Chem Neurosci , 1 :796 , 2010 |
Abstract : |
PubMedSearch : Quek_2010_ACS.Chem.Neurosci_1_796 |
PubMedID: 22778816 |
Title : Poster: Probing the non-competitive binding site within the n-terminal region of alpha4\/beta2 nicotinic receptors - |
Author(s) : Quek GXJ , Halliday JI , McLeod MD , Chebib M |
Ref : Biochemical Pharmacology , 78 :905 , 2009 |
PubMedID: |
Title : Alpha9 nicotinic acetylcholine receptors and the treatment of pain - McIntosh_2009_Biochem.Pharmacol_78(7)_693 |
Author(s) : McIntosh JM , Absalom N , Chebib M , Elgoyhen AB , Vincler M |
Ref : Biochemical Pharmacology , 78 :693 , 2009 |
Abstract : |
PubMedSearch : McIntosh_2009_Biochem.Pharmacol_78(7)_693 |
PubMedID: 19477168 |
Title : The beta-amyloid protein of Alzheimer's disease binds to membrane lipids but does not bind to the alpha7 nicotinic acetylcholine receptor - Small_2007_J.Neurochem_101_1527 |
Author(s) : Small DH , Maksel D , Kerr ML , Ng J , Hou X , Chu C , Mehrani H , Unabia S , Azari MF , Loiacono R , Aguilar MI , Chebib M |
Ref : Journal of Neurochemistry , 101 :1527 , 2007 |
Abstract : |
PubMedSearch : Small_2007_J.Neurochem_101_1527 |
PubMedID: 17286584 |