Peters D

General

Full name : Peters Dan

First name : Dan

Mail : Aniona ApS, Baltorpvej 154, DK-2750 Ballerup

Zip Code :

City :

Country : Denmark

Email : info@danpet.eu

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References (25)

Title : Radiosynthesis and in vitro validation of (3)H-NS14492 as a novel high affinity alpha7 nicotinic receptor radioligand - Magnussen_2015_Eur.J.Pharmacol_762_35
Author(s) : Magnussen JH , Ettrup A , Donat CK , Peters D , Pedersen MH , Knudsen GM , Mikkelsen JD
Ref : European Journal of Pharmacology , 762 :35 , 2015
PubMedID: 25941084

Title : Engineered alpha4beta2 nicotinic acetylcholine receptors as models for measuring agonist binding and effect at the orthosteric low-affinity alpha4-alpha4 interface - Ahring_2015_Neuropharmacol_92_135
Author(s) : Ahring PK , Olsen JA , Nielsen EO , Peters D , Pedersen MH , Rohde LA , Kastrup JS , Shahsavar A , Indurthi DC , Chebib M , Gajhede M , Balle T
Ref : Neuropharmacology , 92 :135 , 2015
PubMedID: 25595102

Title : Poster: Exploring the structure activity relationships of halogen containing N-(pyridin-3-yl)-piperazines and homopiperazines at alpha4beta2 nAChRs -
Author(s) : Rudner-Varga V , Ahring PK , Indurthi D , Peters D , Orton H , Kanizaj N , McLeod MD , Chebib M , Balle T
Ref : Biochemical Pharmacology , 97 :623 , 2015
PubMedID:

Title : Poster: Radiosynthesis and in vitro validation of [3H]NS14492 as a novel high affinity alpha7 nicotinic receptor radioligand -
Author(s) : Donat CK , Magnussen JH , Ettrup A , Peters D , Pedersen MH , Knudsen GM , Mikkelsen JD
Ref : Biochemical Pharmacology , 97 :629 , 2015
PubMedID:

Title : A Promising PET Tracer for Imaging of alpha(7) Nicotinic Acetylcholine Receptors in the Brain: Design, Synthesis, and in Vivo Evaluation of a Dibenzothiophene-Based Radioligand - Teodoro_2015_Molecules_20_18387
Author(s) : Teodoro R , Scheunemann M , Deuther-Conrad W , Wenzel B , Fasoli FM , Gotti C , Kranz M , Donat CK , Patt M , Hillmer A , Zheng MQ , Peters D , Steinbach J , Sabri O , Huang Y , Brust P
Ref : Molecules , 20 :18387 , 2015
PubMedID: 26473809

Title : Biophysical and pharmacological characterization of alpha6-containing nicotinic acetylcholine receptors expressed in HEK293 cells - Rasmussen_2014_Brain.Res_1542_1
Author(s) : Rasmussen AH , Strobaek D , Dyhring T , Jensen ML , Peters D , Grunnet M , Timmermann DB , Ahring PK
Ref : Brain Research , 1542 :1 , 2014
PubMedID: 24157862

Title : Two distinct allosteric binding sites at alpha4beta2 nicotinic acetylcholine receptors revealed by NS206 and NS9283 give unique insights to binding activity-associated linkage at Cys-loop receptors - Olsen_2013_J.Biol.Chem_288_35997
Author(s) : Olsen JA , Kastrup JS , Peters D , Gajhede M , Balle T , Ahring PK
Ref : Journal of Biological Chemistry , 288 :35997 , 2013
PubMedID: 24169695

Title : Molecular determinants of subtype-selective efficacies of cytisine and the novel compound NS3861 at heteromeric nicotinic acetylcholine receptors - Harpsoe_2013_J.Biol.Chem_288_2559
Author(s) : Harpsoe K , Hald H , Timmermann DB , Jensen ML , Dyhring T , Nielsen EO , Peters D , Balle T , Gajhede M , Kastrup JS , Ahring PK
Ref : Journal of Biological Chemistry , 288 :2559 , 2013
PubMedID: 23229547

Title : Augmentation of cognitive function by NS9283, a stoichiometry-dependent positive allosteric modulator of alpha2- and alpha4-containing nicotinic acetylcholine receptors - Timmermann_2012_Br.J.Pharmacol_167_164
Author(s) : Timmermann DB , Sandager-Nielsen K , Dyhring T , Smith M , Jacobsen AM , Nielsen EO , Grunnet M , Christensen JK , Peters D , Kohlhaas KL , Olsen GM , Ahring PK
Ref : British Journal of Pharmacology , 167 :164 , 2012
PubMedID: 22506660

Title : Intersubunit bridge formation governs agonist efficacy at nicotinic acetylcholine alpha4beta2 receptors: unique role of halogen bonding revealed - Rohde_2012_J.Biol.Chem_287_4248
Author(s) : Rohde LA , Ahring PK , Jensen ML , Nielsen EO , Peters D , Helgstrand C , Krintel C , Harpsoe K , Gajhede M , Kastrup JS , Balle T
Ref : Journal of Biological Chemistry , 287 :4248 , 2012
PubMedID: 22170047

Title : Poster: Differential allosteric modulation of high- and low-sensitivity forms of the alpha4\/beta2 nAChR: Evidence for distinct modulator binding sites -
Author(s) : Timmermann DB , Grunnet M , Peters D , Ahring PK
Ref : Biochemical Pharmacology , 82 :1031 , 2011
PubMedID:

Title : Unraveling the high- and low-sensitivity agonist responses of nicotinic acetylcholine receptors - Harpsoe_2011_J.Neurosci_31_10759
Author(s) : Harpsoe K , Ahring PK , Christensen JK , Jensen ML , Peters D , Balle T
Ref : Journal of Neuroscience , 31 :10759 , 2011
PubMedID: 21795528

Title : Poster: The (alpha4)3(\/beta2)2 nAChR has a benzodiazepine-like modulatory binding site in the alphaalpha-subunit interface as revealed by studies with NS9283 -
Author(s) : Ahring PK , Peters D , Christensen JK , Jensen ML , Harpsoe K , Balle T
Ref : Biochemical Pharmacology , 82 :1029 , 2011
PubMedID:

Title : 11C-NS14492 as a novel PET radioligand for imaging cerebral alpha7 nicotinic acetylcholine receptors: in vivo evaluation and drug occupancy measurements - Ettrup_2011_J.Nucl.Med_52_1449
Author(s) : Ettrup A , Mikkelsen JD , Lehel S , Madsen J , Nielsen EO , Palner M , Timmermann DB , Peters D , Knudsen GM
Ref : J Nucl Med , 52 :1449 , 2011
PubMedID: 21828113

Title : In vitro pharmacological characterization of a novel selective alpha7 neuronal nicotinic acetylcholine receptor agonist ABT-107 - Malysz_2010_J.Pharmacol.Exp.Ther_334_863
Author(s) : Malysz J , Anderson DJ , Gronlien JH , Ji J , Bunnelle WH , Hakerud M , Thorin-Hagene K , Ween H , Helfrich R , Hu M , Gubbins E , Gopalakrishnan S , Puttfarcken PS , Briggs CA , Li J , Meyer MD , Dyhring T , Ahring PK , Nielsen EO , Peters D , Timmermann DB , Gopalakrishnan M
Ref : Journal of Pharmacology & Experimental Therapeutics , 334 :863 , 2010
PubMedID: 20504915

Title : Syntheses and structure-activity relationship (SAR) studies of 2,5-diazabicyclo[2.2.1]heptanes as novel alpha7 neuronal nicotinic receptor (NNR) ligands - Li_2010_Bioorg.Med.Chem.Lett_20_3636
Author(s) : Li T , Bunnelle WH , Ryther KB , Anderson DJ , Malysz J , Helfrich R , Gronlien JH , Hakerud M , Peters D , Schrimpf MR , Gopalakrishnan M , Ji J
Ref : Bioorganic & Medicinal Chemistry Lett , 20 :3636 , 2010
PubMedID: 20472430

Title : Alpha7 nicotinic acetylcholine receptor activation ameliorates scopolamine-induced behavioural changes in a modified continuous Y-maze task in mice - Redrobe_2009_Eur.J.Pharmacol_602_58
Author(s) : Redrobe JP , Nielsen EO , Christensen JK , Peters D , Timmermann DB , Olsen GM
Ref : European Journal of Pharmacology , 602 :58 , 2009
PubMedID: 18848931

Title : Poster: In vitro pharmacological profile of a novel alpha4\/beta2 positive allosteric modulator NS9283 (A-969933) -
Author(s) : Malysz J , Dyhring T , Ahring PK , Olsen GM , Peters D , Gronlien JH , Wetterstrand C , Ween H , Haakerud M , Thorin-Hagene K , Andersen E , Anderson DJ , Hu M , Kroeger PE , Lee CHL , Gopalakrishnan M , Timmermann DB
Ref : Biochemical Pharmacology , 78 :919 , 2009
PubMedID:

Title : Complementary three-dimensional quantitative structure-activity relationship modeling of binding affinity and functional potency: a study on alpha4beta2 nicotinic ligands - Tosco_2009_J.Med.Chem_52_2311
Author(s) : Tosco P , Ahring PK , Dyhring T , Peters D , Harpsoe K , Liljefors T , Balle T
Ref : Journal of Medicinal Chemistry , 52 :2311 , 2009
PubMedID: 19301898

Title : Role of channel activation in cognitive enhancement mediated by alpha7 nicotinic acetylcholine receptors - Briggs_2009_Br.J.Pharmacol_158_1486
Author(s) : Briggs CA , Gronlien JH , Curzon P , Timmermann DB , Ween H , Thorin-Hagene K , Kerr P , Anderson DJ , Malysz J , Dyhring T , Olsen GM , Peters D , Bunnelle WH , Gopalakrishnan M
Ref : British Journal of Pharmacology , 158 :1486 , 2009
PubMedID: 19845675

Title : Molecular imaging of alpha7 nicotinic acetylcholine receptors: design and evaluation of the potent radioligand [18F]NS10743 - Deuther-Conrad_2009_Eur.J.Nucl.Med.Mol.Imaging_36_791
Author(s) : Deuther-Conrad W , Fischer S , Hiller A , Nielsen EO , Timmermann DB , Steinbach J , Sabri O , Peters D , Brust P
Ref : Eur J Nucl Med Mol Imaging , 36 :791 , 2009
PubMedID: 19137292

Title : The selective alpha7 nicotinic acetylcholine receptor agonist A-582941 activates immediate early genes in limbic regions of the forebrain: Differential effects in the juvenile and adult rat - Thomsen_2008_Neurosci_154_741
Author(s) : Thomsen MS , Mikkelsen JD , Timmermann DB , Peters D , Hay-Schmidt A , Martens H , Hansen HH
Ref : Neuroscience , 154 :741 , 2008
PubMedID: 18495359

Title : An allosteric modulator of the alpha7 nicotinic acetylcholine receptor possessing cognition-enhancing properties in vivo - Timmermann_2007_J.Pharmacol.Exp.Ther_323_294
Author(s) : Timmermann DB , Gronlien JH , Kohlhaas KL , Nielsen EO , Dam E , Jorgensen TD , Ahring PK , Peters D , Holst D , Christensen JK , Malysz J , Briggs CA , Gopalakrishnan M , Olsen GM
Ref : Journal of Pharmacology & Experimental Therapeutics , 323 :294 , 2007
PubMedID: 17625074

Title : Alpha-7 nicotinic acetylcholine receptor agonists selectively activate limbic regions of the rat forebrain: an effect similar to antipsychotics - Hansen_2007_J.Neurosci.Res_85_1810
Author(s) : Hansen HH , Timmermann DB , Peters D , Walters C , Damaj MI , Mikkelsen JD
Ref : Journal of Neuroscience Research , 85 :1810 , 2007
PubMedID: 17455307

Title : New ligands with affinity for the alpha4beta2 subtype of nicotinic acetylcholine receptors. Synthesis, receptor binding, and 3D-QSAR modeling - Audouze_2006_J.Med.Chem_49_3159
Author(s) : Audouze K , Nielsen EO , Olsen GM , Ahring P , Jorgensen TD , Peters D , Liljefors T , Balle T
Ref : Journal of Medicinal Chemistry , 49 :3159 , 2006
PubMedID: 16722635