| Title : Fragment-Based Discovery of Fenamic Acids as Pan-Species Inhibitors of the Soluble Epoxide Hydrolase Phosphatase Domain - Zhu_2026_ACS.Chem.Biol_21_2053 |
| Author(s) : Zhu WF , Feugray G , Brunst S , Messaoudi H , Yang M , Martinez-Conde N , Kramer A , Weizel L , Ehrler JMH , Kramer JS , Kaiser A , Al-Tarrass M , Pereira T , Valet M , Brunel V , Schubert-Zsilavecz M , Knapp S , Lillich FF , Hernandez-Olmos V , Duflot T , Hiesinger K , Qian H , Proschak A , Bellien J , Proschak E |
| Ref : ACS Chemical Biology , 21 :2053 , 2026 |
| Abstract : |
| PubMedSearch : Zhu_2026_ACS.Chem.Biol_21_2053 |
| PubMedID: 42631699 |
| Title : Computed Tomography Perfusion and Angiography for Death by Neurologic Criteria - Chasse_2025_JAMA.Neurol__ |
| Author(s) : Chasse M , Shankar JJS , Fergusson DA , English SW , Dhanani S , Lauzier F , Turgeon AF , Ball I , Darvesh S , Neves Briard J , Essig M , Boucher-Roy D , Titova P , Lebrasseur M , Couillard P , Kramer A , D'Aragon F , Hannouche M , Tampieri D , Meade MO , Menon BK , Green R , Baker AJ , Burns KEA , Zarychanski R , Shahin J , Boyd JG , Binnie A , Gibson A , Wang HT , Shemie S |
| Ref : JAMA Neurol , : , 2025 |
| Abstract : |
| PubMedSearch : Chasse_2025_JAMA.Neurol__ |
| PubMedID: 40512483 |
| Title : Novel alpha-7 nicotinic acetylcholine receptor agonists containing a urea moiety: identification and characterization of the potent, selective, and orally efficacious agonist 1-[6-(4-fluorophenyl)pyridin-3-yl]-3-(4-piperidin-1-ylbutyl) urea (SEN34625\/WYE-103914) - Ghiron_2010_J.Med.Chem_53_4379 |
| Author(s) : Ghiron C , Haydar SN , Aschmies S , Bothmann H , Castaldo C , Cocconcelli G , Comery TA , Di L , Dunlop J , Lock T , Kramer A , Kowal D , Jow F , Grauer S , Harrison B , La Rosa S , Maccari L , Marquis KL , Micco I , Nencini A , Quinn J , Robichaud AJ , Roncarati R , Scali C , Terstappen GC , Turlizzi E , Valacchi M , Varrone M , Zanaletti R , Zanelli U |
| Ref : Journal of Medicinal Chemistry , 53 :4379 , 2010 |
| Abstract : |
| PubMedSearch : Ghiron_2010_J.Med.Chem_53_4379 |
| PubMedID: 20465311 |
| Title : Old and new pharmacology: positive allosteric modulation of the alpha7 nicotinic acetylcholine receptor by the 5-hydroxytryptamine(2B\/C) receptor antagonist SB-206553 (3,5-dihydro-5-methyl-N-3-pyridinylbenzo[1,2-b:4,5-b']di pyrrole-1(2H)-carboxamide) - Dunlop_2009_J.Pharmacol.Exp.Ther_328_766 |
| Author(s) : Dunlop J , Lock T , Jow B , Sitzia F , Grauer S , Jow F , Kramer A , Bowlby MR , Randall A , Kowal D , Gilbert A , Comery TA , Larocque J , Soloveva V , Brown J , Roncarati R |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 328 :766 , 2009 |
| Abstract : |
| PubMedSearch : Dunlop_2009_J.Pharmacol.Exp.Ther_328_766 |
| PubMedID: 19050173 |
| Title : Poster: In vitro pharmacological characterization and pro-cognitive effects of the selective alpha-7 nicotinic agonist WYE-103914 - |
| Author(s) : Dunlop J , Comery TA , Lock T , Kramer A , Kowal D , Yeola S , Jow F , Aschmies S , Lin Q , Beyer CE , Brennan J , Kelley C , Roncarati R , Scali C , Haydar S , Ghiron C , Marquis KL , Harrison B , Robichaud A , Terstappen GC |
| Ref : Biochemical Pharmacology , 78 :911 , 2009 |
| PubMedID: |
| Title : Functional properties of alpha7 nicotinic acetylcholine receptors co-expressed with RIC-3 in a stable recombinant CHO-K1 cell line - Roncarati_2008_Assay.Drug.Dev.Technol_6_181 |
| Author(s) : Roncarati R , Seredenina T , Jow B , Jow F , Papini S , Kramer A , Bothmann H , Dunlop J , Terstappen GC |
| Ref : Assay Drug Dev Technol , 6 :181 , 2008 |
| Abstract : |
| PubMedSearch : Roncarati_2008_Assay.Drug.Dev.Technol_6_181 |
| PubMedID: 18471073 |