Title : Inhibitory Activity of 4-Benzylidene Oxazolones Derivatives of Cinnamic Acid on Human Acetylcholinesterase and Cognitive Improvements in a Mouse Model - Ramirez-Ruiz_2023_Molecules_28_ |
Author(s) : Ramirez-Ruiz AM , Avila-Cossio ME , Estolano-Cobian A , Cornejo-Bravo JM , Martinez AL , Cordova-Guerrero I , Cota-Ramirez BR , Carranza-Ambriz KP , Rivero IA , Serrano-Medina A |
Ref : Molecules , 28 : , 2023 |
Abstract : |
PubMedSearch : Ramirez-Ruiz_2023_Molecules_28_ |
PubMedID: 37959813 |
Title : Novel thienocycloalkylpyridazinones as useful scaffolds for acetylcholinesterase inhibition and serotonin 5-HT(6) receptor interaction - Asproni_2023_Bioorg.Med.Chem_84_117256 |
Author(s) : Asproni B , Catto M , Loriga G , Murineddu G , Corona P , Purgatorio R , Cichero E , Fossa P , Scarano N , Martinez AL , Brea J , Pinna GA |
Ref : Bioorganic & Medicinal Chemistry , 84 :117256 , 2023 |
Abstract : |
PubMedSearch : Asproni_2023_Bioorg.Med.Chem_84_117256 |
PubMedID: 37003157 |
Title : Synthesis, In Vitro Profiling, and In Vivo Evaluation of Benzohomoadamantane-Based Ureas for Visceral Pain: A New Indication for Soluble Epoxide Hydrolase Inhibitors - Codony_2022_J.Med.Chem_65_13660 |
Author(s) : Codony S , Entrena JM , Calvo-Tusell C , Jora B , Gonzalez-Cano R , Osuna S , Corpas R , Morisseau C , Perez B , Barniol-Xicota M , Grinan-Ferre C , Perez C , Rodriguez-Franco MI , Martinez AL , Loza MI , Pallas M , Verhelst SHL , Sanfeliu C , Feixas F , Hammock BD , Brea J , Cobos EJ , Vazquez S |
Ref : Journal of Medicinal Chemistry , 65 :13660 , 2022 |
Abstract : |
PubMedSearch : Codony_2022_J.Med.Chem_65_13660 |
PubMedID: 36222708 |
Title : Synthesis and biological evaluation of dantrolene-like hydrazide and hydrazone analogues as multitarget agents for neurodegenerative diseases - Bolognino_2021_ChemMedChem__ |
Author(s) : Bolognino I , Giangregorio N , Tonazzi A , Martinez AL , Altomare CD , Loza MI , Sablone S , Cellamare S , Catto M |
Ref : ChemMedChem , : , 2021 |
Abstract : |
PubMedSearch : Bolognino_2021_ChemMedChem__ |
PubMedID: 34047061 |