Full name : Valant Celine
First name : Celine
Mail : Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville VIC 3052
Zip Code :
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Country : Australia
Email : celine.valant@monash.edu
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| Title : Probing structural requirements of positive allosteric modulators of the m4 muscarinic receptor - Huynh_2013_J.Med.Chem_56_8196 |
| Author(s) : Huynh T , Valant C , Crosby IT , Sexton PM , Christopoulos A , Capuano B |
| Ref : Journal of Medicinal Chemistry , 56 :8196 , 2013 |
| Abstract : Huynh_2013_J.Med.Chem_56_8196 |
| ESTHER : Huynh_2013_J.Med.Chem_56_8196 |
| PubMedSearch : Huynh_2013_J.Med.Chem_56_8196 |
| PubMedID: 24074052 |
| Title : Reverse engineering of the selective agonist TBPB unveils both orthosteric and allosteric modes of action at the M(1) muscarinic acetylcholine receptor - Keov_2013_Mol.Pharmacol_84_425 |
| Author(s) : Keov P , Valant C , Devine SM , Lane JR , Scammells PJ , Sexton PM , Christopoulos A |
| Ref : Molecular Pharmacology , 84 :425 , 2013 |
| Abstract : Keov_2013_Mol.Pharmacol_84_425 |
| ESTHER : Keov_2013_Mol.Pharmacol_84_425 |
| PubMedSearch : Keov_2013_Mol.Pharmacol_84_425 |
| PubMedID: 23798605 |
| Title : Structural basis for modulation of a G-protein-coupled receptor by allosteric drugs - Dror_2013_Nature_503_295 |
| Author(s) : Dror RO , Green HF , Valant C , Borhani DW , Valcourt JR , Pan AC , Arlow DH , Canals M , Lane JR , Rahmani R , Baell JB , Sexton PM , Christopoulos A , Shaw DE |
| Ref : Nature , 503 :295 , 2013 |
| Abstract : Dror_2013_Nature_503_295 |
| ESTHER : Dror_2013_Nature_503_295 |
| PubMedSearch : Dror_2013_Nature_503_295 |
| PubMedID: 24121438 |
| Title : Activation and allosteric modulation of a muscarinic acetylcholine receptor - Kruse_2013_Nature_504_101 |
| Author(s) : Kruse AC , Ring AM , Manglik A , Hu J , Hu K , Eitel K , Hubner H , Pardon E , Valant C , Sexton PM , Christopoulos A , Felder CC , Gmeiner P , Steyaert J , Weis WI , Garcia KC , Wess J , Kobilka BK |
| Ref : Nature , 504 :101 , 2013 |
| Abstract : Kruse_2013_Nature_504_101 |
| ESTHER : Kruse_2013_Nature_504_101 |
| PubMedSearch : Kruse_2013_Nature_504_101 |
| PubMedID: 24256733 |
| Title : Synthesis and pharmacological profiling of analogues of benzyl quinolone carboxylic acid (BQCA) as allosteric modulators of the M1 muscarinic receptor - Mistry_2013_J.Med.Chem_56_5151 |
| Author(s) : Mistry SN , Valant C , Sexton PM , Capuano B , Christopoulos A , Scammells PJ |
| Ref : Journal of Medicinal Chemistry , 56 :5151 , 2013 |
| Abstract : Mistry_2013_J.Med.Chem_56_5151 |
| ESTHER : Mistry_2013_J.Med.Chem_56_5151 |
| PubMedSearch : Mistry_2013_J.Med.Chem_56_5151 |
| PubMedID: 23718562 |
| Title : Allosteric modulation of endogenous metabolites as an avenue for drug discovery - Wootten_2012_Mol.Pharmacol_82_281 |
| Author(s) : Wootten D , Savage EE , Valant C , May LT , Sloop KW , Ficorilli J , Showalter AD , Willard FS , Christopoulos A , Sexton PM |
| Ref : Molecular Pharmacology , 82 :281 , 2012 |
| Abstract : Wootten_2012_Mol.Pharmacol_82_281 |
| ESTHER : Wootten_2012_Mol.Pharmacol_82_281 |
| PubMedSearch : Wootten_2012_Mol.Pharmacol_82_281 |
| PubMedID: 22576254 |
| Title : Probe dependence in the allosteric modulation of a G protein-coupled receptor: implications for detection and validation of allosteric ligand effects - Valant_2012_Mol.Pharmacol_81_41 |
| Author(s) : Valant C , Felder CC , Sexton PM , Christopoulos A |
| Ref : Molecular Pharmacology , 81 :41 , 2012 |
| Abstract : Valant_2012_Mol.Pharmacol_81_41 |
| ESTHER : Valant_2012_Mol.Pharmacol_81_41 |
| PubMedSearch : Valant_2012_Mol.Pharmacol_81_41 |
| PubMedID: 21989256 |
| Title : Determination of adenosine A1 receptor agonist and antagonist pharmacology using Saccharomyces cerevisiae: implications for ligand screening and functional selectivity - Stewart_2009_J.Pharmacol.Exp.Ther_331_277 |
| Author(s) : Stewart GD , Valant C , Dowell SJ , Mijaljica D , Devenish RJ , Scammells PJ , Sexton PM , Christopoulos A |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 331 :277 , 2009 |
| Abstract : Stewart_2009_J.Pharmacol.Exp.Ther_331_277 |
| ESTHER : Stewart_2009_J.Pharmacol.Exp.Ther_331_277 |
| PubMedSearch : Stewart_2009_J.Pharmacol.Exp.Ther_331_277 |
| PubMedID: 19641164 |
| Title : A novel mechanism of G protein-coupled receptor functional selectivity. Muscarinic partial agonist McN-A-343 as a bitopic orthosteric\/allosteric ligand - Valant_2008_J.Biol.Chem_283_29312 |
| Author(s) : Valant C , Gregory KJ , Hall NE , Scammells PJ , Lew MJ , Sexton PM , Christopoulos A |
| Ref : Journal of Biological Chemistry , 283 :29312 , 2008 |
| Abstract : Valant_2008_J.Biol.Chem_283_29312 |
| ESTHER : Valant_2008_J.Biol.Chem_283_29312 |
| PubMedSearch : Valant_2008_J.Biol.Chem_283_29312 |
| PubMedID: 18723515 |