| Title : Selective and Orally Bioavailable Dipeptidyl Peptidase 9 Inhibitors with Potent Pyroptosis Induction Properties - Filippi_2025_J.Med.Chem__ |
| Author(s) : Filippi N , Mertens K , De Loose J , Benramdane S , Hermans R , Espadinha M , Dirkx L , Feijens PB , Nozal V , Verhulst E , Peeters S , Gomard T , Corthaut S , Augustyns K , Caljon G , Schols D , De Meester I , Van der Veken P |
| Ref : Journal of Medicinal Chemistry , : , 2025 |
| Abstract : |
| PubMedSearch : Filippi_2025_J.Med.Chem__ |
| PubMedID: 41160575 |
| Gene_locus related to this paper: human-DPP9 |
| Title : Cosolvent Molecular Dynamics Applied to DPP4, DPP8 and DPP9: Reproduction of Important Binding Features and Use in Inhibitor Design - Beyens_2024_J.Chem.Inf.Model_64_7650 |
| Author(s) : Beyens O , Corthaut S , Peeters S , Van der Veken P , De Meester I , De Winter H |
| Ref : J Chem Inf Model , 64 :7650 , 2024 |
| Abstract : |
| PubMedSearch : Beyens_2024_J.Chem.Inf.Model_64_7650 |
| PubMedID: 39332821 |
| Title : Active site-directed probes targeting dipeptidyl peptidases 8 and 9 - Espadinha_2024_Eur.J.Med.Chem_270_116389 |
| Author(s) : Espadinha M , De Loose J , Corthaut S , Thys S , Van Rymenant Y , Verhulst E , Benramdane S , Filippi N , Augustyns K , Van Wielendaele P , Pintelon I , De Meester I , Van der Veken P |
| Ref : Eur Journal of Medicinal Chemistry , 270 :116389 , 2024 |
| Abstract : |
| PubMedSearch : Espadinha_2024_Eur.J.Med.Chem_270_116389 |
| PubMedID: 38593588 |
| Gene_locus related to this paper: human-DPP8 , human-DPP9 |
| Title : An interdisciplinary approach provides insights into the pronounced selectivity of compound 42 for DPP9 - Beyens_2024_ChemMedChem__e202400700 |
| Author(s) : Beyens O , Corthaut S , Lambeir AM , Van der Veken P , Sterckx YG , De Meester I , De Winter H |
| Ref : ChemMedChem , :e202400700 , 2024 |
| Abstract : |
| PubMedSearch : Beyens_2024_ChemMedChem__e202400700 |
| PubMedID: 39552560 |
| Gene_locus related to this paper: human-DPP8 , human-DPP9 |