| Title : In vitro kinetic profiling by enzymatic approaches to select FAPIs with a long residence time - Verhulst_2026_Eur.J.Med.Chem_304_118494 |
| Author(s) : Verhulst E , Brzeminski P , de Groot A , Wals JW , Michiels R , Fabisiak A , Thys J , Grintsevich S , Van Rymenant Y , Peeters S , Lambregts S , Sim Y , Verstraete R , Van Wielendaele P , Berg M , Elvas F , Van Ostade X , Rosch F , Lambeir AM , De Winter H , Van der Veken P , De Meester I |
| Ref : Eur Journal of Medicinal Chemistry , 304 :118494 , 2026 |
| Abstract : |
| PubMedSearch : Verhulst_2026_Eur.J.Med.Chem_304_118494 |
| PubMedID: 41455278 |
| Gene_locus related to this paper: human-FAP |
| Title : Fibroblast activation protein on human natural killer cells: insights from natural killer cell activation and crosstalk with cancer-associated fibroblasts - Van Rymenant_2025_J.Leukoc.Biol_117_ |
| Author(s) : Van Rymenant Y , de Groot A , Dirkx L , Verhulst E , De Loose J , Pintelon I , Verhezen T , De Waele J , Thys S , De Wever O , Tanc M , Caljon G , Van der Veken P , De Meester I |
| Ref : J Leukoc Biol , 117 : , 2025 |
| Abstract : |
| PubMedSearch : Van Rymenant_2025_J.Leukoc.Biol_117_ |
| PubMedID: 40638797 |
| Gene_locus related to this paper: human-FAP |
| Title : Synthesis and Preclinical Evaluation of Druglike (18)F-Labeled Fibroblast Activation Protein (FAP) Inhibitors with Enhanced Tumor Retention - Adhikari_2025_Bioconjug.Chem_36_1887 |
| Author(s) : Adhikari K , Grintsevich S , de Groot A , Verhulst E , Van Rymenant Y , Vangestel C , Lauwerys L , Miranda A , De Meester I , Van der Veken P , Elvas F |
| Ref : Bioconjug Chem , 36 :1887 , 2025 |
| Abstract : |
| PubMedSearch : Adhikari_2025_Bioconjug.Chem_36_1887 |
| PubMedID: 40790340 |
| Title : Active site-directed probes targeting dipeptidyl peptidases 8 and 9 - Espadinha_2024_Eur.J.Med.Chem_270_116389 |
| Author(s) : Espadinha M , De Loose J , Corthaut S , Thys S , Van Rymenant Y , Verhulst E , Benramdane S , Filippi N , Augustyns K , Van Wielendaele P , Pintelon I , De Meester I , Van der Veken P |
| Ref : Eur Journal of Medicinal Chemistry , 270 :116389 , 2024 |
| Abstract : |
| PubMedSearch : Espadinha_2024_Eur.J.Med.Chem_270_116389 |
| PubMedID: 38593588 |
| Gene_locus related to this paper: human-DPP8 , human-DPP9 |
| Title : Next generation fibroblast activation protein (FAP) targeting PET tracers - The tetrazine ligation allows an easy and convenient way to (18)F-labeled (4-quinolinoyl)glycyl-2-cyanopyrrolidines - Poulie_2023_Eur.J.Med.Chem_262_115862 |
| Author(s) : Poulie CBM , Shalgunov V , Elvas F , Van Rymenant Y , Moon ES , Battisti UM , De Loose J , De Meester I , Rosch F , Van der Veken P , Herth MM |
| Ref : Eur Journal of Medicinal Chemistry , 262 :115862 , 2023 |
| Abstract : |
| PubMedSearch : Poulie_2023_Eur.J.Med.Chem_262_115862 |
| PubMedID: 37883899 |
| Title : Novel Generation of FAP Inhibitor-Based Homodimers for Improved Application in Radiotheranostics - Martin_2023_Cancers.(Basel)_15_ |
| Author(s) : Martin M , Ballal S , Yadav MP , Bal C , Van Rymenant Y , De Loose J , Verhulst E , De Meester I , Van der Veken P , Roesch F |
| Ref : Cancers (Basel) , 15 : , 2023 |
| Abstract : |
| PubMedSearch : Martin_2023_Cancers.(Basel)_15_ |
| PubMedID: 36980775 |
| Title : Vildagliptin-Derived Dipeptidyl Peptidase 9 (DPP9) Inhibitors: Identification of a DPP8\/9-Specific Lead - Benramdane_2022_ChemMedChem__e202200097 |
| Author(s) : Benramdane S , De Loose J , Beyens O , Van Rymenant Y , Vliegen G , Augustyns K , De Winter H , De Meester I , Van der Veken P |
| Ref : ChemMedChem , :e202200097 , 2022 |
| Abstract : |
| PubMedSearch : Benramdane_2022_ChemMedChem__e202200097 |
| PubMedID: 35760756 |
| Title : Fibroblast Activation Protein (FAP) targeting homodimeric FAP inhibitor radiotheranostics: a step to improve tumor uptake and retention time - Moon_2021_Am.J.Nucl.Med.Mol.Imaging_11_476 |
| Author(s) : Moon ES , Ballal S , Yadav MP , Bal C , Van Rymenant Y , Stephan S , Bracke A , Van der Veken P , De Meester I , Roesch F |
| Ref : Am J Nucl Med Mol Imaging , 11 :476 , 2021 |
| Abstract : |
| PubMedSearch : Moon_2021_Am.J.Nucl.Med.Mol.Imaging_11_476 |
| PubMedID: 35003886 |
| Title : In Vitro Evaluation of the Squaramide-Conjugated Fibroblast Activation Protein Inhibitor-Based Agents AAZTA(5).SA.FAPi and DOTA.SA.FAPi - Moon_2021_Molecules_26_3482 |
| Author(s) : Moon ES , Van Rymenant Y , Battan S , De Loose J , Bracke A , Van der Veken P , De Meester I , Rosch F |
| Ref : Molecules , 26 :3482 , 2021 |
| Abstract : |
| PubMedSearch : Moon_2021_Molecules_26_3482 |
| PubMedID: 34201111 |
| Gene_locus related to this paper: human-FAP |