Galati S

Title : Watermelon: setup and validation of an in silico fragment-based approach - Di Stefano_2024_J.Enzyme.Inhib.Med.Chem_39_2356179

Author(s) : Di Stefano M , Galati S , Piazza L , Gado F , Granchi C , Macchia M , Giordano A , Tuccinardi T , Poli G

Ref : J Enzyme Inhib Med Chem , 39 :2356179 , 2024

Abstract :

PubMedSearch : Di Stefano_2024_J.Enzyme.Inhib.Med.Chem_39_2356179

PubMedID: 38864179

Title : Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors - Di Stefano_2023_Eur.J.Med.Chem_263_115916

Author(s) : Di Stefano M , Masoni S , Bononi G , Poli G , Galati S , Gado F , Manzi S , Vagaggini C , Brai A , Caligiuri I , Asif K , Rizzolio F , Macchia M , Chicca A , Sodi A , Di Bussolo V , Minutolo F , Meier P , Gertsch J , Granchi C , Dreassi E , Tuccinardi T

Ref : Eur Journal of Medicinal Chemistry , 263 :115916 , 2023

Abstract :

PubMedSearch : Di Stefano_2023_Eur.J.Med.Chem_263_115916

PubMedID: 37976705

Galati S

References (2)

1. Watermelon: setup and validation of an in silico fragment-based approach - Di Stefano_2024_J.Enzyme.Inhib.Med.Chem_39_2356179

2. Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors - Di Stefano_2023_Eur.J.Med.Chem_263_115916